IL95279A - 4-]ציקלואלקילן-1- )אימידאזוליל או טריאזוליל( מתיל[- בנזוניטרילים ותולדותיהם, תהליכים להכנתם ותכשירי רוקחות המכילים אותם - Google Patents
4-]ציקלואלקילן-1- )אימידאזוליל או טריאזוליל( מתיל[- בנזוניטרילים ותולדותיהם, תהליכים להכנתם ותכשירי רוקחות המכילים אותםInfo
- Publication number
- IL95279A IL95279A IL9527990A IL9527990A IL95279A IL 95279 A IL95279 A IL 95279A IL 9527990 A IL9527990 A IL 9527990A IL 9527990 A IL9527990 A IL 9527990A IL 95279 A IL95279 A IL 95279A
- Authority
- IL
- Israel
- Prior art keywords
- methyl
- imidazolyl
- benzonitrile
- cycloalkylene
- triazolyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE3926365A DE3926365A1 (de) | 1989-08-04 | 1989-08-04 | Cycloalkylenazole, verfahren zu deren herstellung, pharmazeutische praeparate, die diese enthalten sowie ihre verwendung zur herstellung von arzneimitteln |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL95279A0 IL95279A0 (en) | 1991-06-30 |
| IL95279A true IL95279A (he) | 1995-03-30 |
Family
ID=6386820
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL9527990A IL95279A (he) | 1989-08-04 | 1990-08-03 | 4-]ציקלואלקילן-1- )אימידאזוליל או טריאזוליל( מתיל[- בנזוניטרילים ותולדותיהם, תהליכים להכנתם ותכשירי רוקחות המכילים אותם |
Country Status (19)
| Country | Link |
|---|---|
| US (3) | US5135937A (he) |
| EP (1) | EP0411735B1 (he) |
| JP (1) | JP3207417B2 (he) |
| CN (1) | CN1024345C (he) |
| AT (1) | ATE122662T1 (he) |
| AU (1) | AU634266B2 (he) |
| CA (1) | CA2022682C (he) |
| DD (1) | DD296917A5 (he) |
| DE (2) | DE3926365A1 (he) |
| DK (1) | DK0411735T3 (he) |
| ES (1) | ES2074530T3 (he) |
| FI (1) | FI920425A0 (he) |
| HU (2) | HU217126B (he) |
| IE (1) | IE902843A1 (he) |
| IL (1) | IL95279A (he) |
| NO (1) | NO301115B1 (he) |
| PT (1) | PT94884B (he) |
| WO (1) | WO1991001975A1 (he) |
| ZA (1) | ZA906150B (he) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5352795A (en) * | 1986-03-07 | 1994-10-04 | Ciba-Geigy Corporation | Alpha-heterocycle substituted tolunitriles |
| US5112845A (en) * | 1986-03-07 | 1992-05-12 | Ciba-Geigy Corporation | Alpha-heterocycle substituted tolunitriles |
| TW224461B (he) * | 1990-09-18 | 1994-06-01 | Ciba Geigy Ag | |
| DE4107038A1 (de) * | 1991-03-01 | 1992-09-03 | Schering Ag | Triheteroarylmethane, verfahren zu deren herstellung, pharmazeutische praeparate die diese enthalten sowie ihre verwendung zur herstellung von arzneimitteln |
| DE4120107A1 (de) * | 1991-06-14 | 1992-12-17 | Schering Ag | Bicyclisch substituierte vinylimidazole, -triazole und -tetrazole |
| DE4435368A1 (de) * | 1994-09-22 | 1996-03-28 | Schering Ag | Verwendung von Aromatasehemmern zur Herstellung eines Arzneimittels zur Behandlung eines relativen Androgenmangels beim Mann |
| ZA9510926B (en) | 1994-12-23 | 1996-07-03 | Schering Ag | Compounds with progesterone-antagonistic and antiestrogenic action to be used together for female contraception |
| CA2380940C (en) * | 1999-08-13 | 2013-06-25 | Heinrich Wieland | Substances and agents for positively influencing collagen |
| CN101253160A (zh) * | 2005-07-06 | 2008-08-27 | 西科尔公司 | 制备来曲唑的改进方法 |
| CN100425621C (zh) * | 2006-07-06 | 2008-10-15 | 云南大学 | 甾体咪唑盐类化合物及其制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4609666A (en) * | 1984-06-18 | 1986-09-02 | Eli Lilly And Company | Aromatase inhibiting derivatives of α,α-bis(4-halophenyl)methyltetrazoles and triazoles |
| JPS62149666A (ja) * | 1985-12-25 | 1987-07-03 | Shionogi & Co Ltd | Ｎ−ビニルアゾ−ル類 |
| US4749713A (en) * | 1986-03-07 | 1988-06-07 | Ciba-Geigy Corporation | Alpha-heterocycle substituted tolunitriles |
-
1989
- 1989-08-04 DE DE3926365A patent/DE3926365A1/de not_active Withdrawn
-
1990
- 1990-08-02 DD DD90343215A patent/DD296917A5/de not_active IP Right Cessation
- 1990-08-02 PT PT94884A patent/PT94884B/pt unknown
- 1990-08-03 AU AU60194/90A patent/AU634266B2/en not_active Ceased
- 1990-08-03 US US07/563,114 patent/US5135937A/en not_active Expired - Fee Related
- 1990-08-03 CA CA002022682A patent/CA2022682C/en not_active Expired - Fee Related
- 1990-08-03 ZA ZA906150A patent/ZA906150B/xx unknown
- 1990-08-03 IL IL9527990A patent/IL95279A/he not_active IP Right Cessation
- 1990-08-04 CN CN90106813A patent/CN1024345C/zh not_active Expired - Fee Related
- 1990-08-06 AT AT90250201T patent/ATE122662T1/de not_active IP Right Cessation
- 1990-08-06 JP JP51080790A patent/JP3207417B2/ja not_active Expired - Fee Related
- 1990-08-06 HU HU9200324A patent/HU217126B/hu not_active IP Right Cessation
- 1990-08-06 HU HU9200324A patent/HUT59911A/hu unknown
- 1990-08-06 DK DK90250201.2T patent/DK0411735T3/da active
- 1990-08-06 ES ES90250201T patent/ES2074530T3/es not_active Expired - Lifetime
- 1990-08-06 DE DE59009084T patent/DE59009084D1/de not_active Expired - Lifetime
- 1990-08-06 EP EP90250201A patent/EP0411735B1/de not_active Expired - Lifetime
- 1990-08-06 WO PCT/DE1990/000611 patent/WO1991001975A1/de active Application Filing
- 1990-08-07 IE IE284390A patent/IE902843A1/en not_active IP Right Cessation
-
1992
- 1992-01-30 FI FI920425A patent/FI920425A0/fi unknown
- 1992-02-03 NO NO920432A patent/NO301115B1/no not_active IP Right Cessation
- 1992-05-28 US US07/889,331 patent/US5280035A/en not_active Expired - Fee Related
-
1993
- 1993-11-16 US US08/153,326 patent/US5411982A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP0411735B1 (de) | 1995-05-17 |
| US5135937A (en) | 1992-08-04 |
| IE902843A1 (en) | 1991-02-27 |
| DE59009084D1 (de) | 1995-06-22 |
| CN1049157A (zh) | 1991-02-13 |
| AU6019490A (en) | 1991-02-07 |
| WO1991001975A1 (de) | 1991-02-21 |
| JP3207417B2 (ja) | 2001-09-10 |
| NO301115B1 (no) | 1997-09-15 |
| HUT59911A (en) | 1992-07-28 |
| DE3926365A1 (de) | 1991-02-07 |
| CN1024345C (zh) | 1994-04-27 |
| CA2022682C (en) | 1997-01-21 |
| PT94884B (pt) | 1997-04-30 |
| NO920432D0 (no) | 1992-02-03 |
| HU9200324D0 (en) | 1992-04-28 |
| IL95279A0 (en) | 1991-06-30 |
| ES2074530T3 (es) | 1995-09-16 |
| ATE122662T1 (de) | 1995-06-15 |
| ZA906150B (en) | 1991-05-29 |
| EP0411735A1 (de) | 1991-02-06 |
| FI920425A0 (fi) | 1992-01-30 |
| US5411982A (en) | 1995-05-02 |
| US5280035A (en) | 1994-01-18 |
| NO920432L (no) | 1992-02-03 |
| DK0411735T3 (da) | 1995-10-16 |
| CA2022682A1 (en) | 1991-02-05 |
| AU634266B2 (en) | 1993-02-18 |
| PT94884A (pt) | 1991-04-18 |
| DD296917A5 (de) | 1991-12-19 |
| HU217126B (hu) | 1999-11-29 |
| JPH05501104A (ja) | 1993-03-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| MM9K | Patent not in force due to non-payment of renewal fees |