IL74215A - Derivatives of 5-phenyltetrazolo(1,5-a)(1,2,4)triazolo(1,5-c)pyrimidine-6-alkanols and pharmaceutical compositions containing them - Google Patents

Derivatives of 5-phenyltetrazolo(1,5-a)(1,2,4)triazolo(1,5-c)pyrimidine-6-alkanols and pharmaceutical compositions containing them

Info

Publication number
IL74215A
IL74215A IL74215A IL7421585A IL74215A IL 74215 A IL74215 A IL 74215A IL 74215 A IL74215 A IL 74215A IL 7421585 A IL7421585 A IL 7421585A IL 74215 A IL74215 A IL 74215A
Authority
IL
Israel
Prior art keywords
pharmaceutical compositions
compositions containing
phenyltetrazolo
triazolo
alkanols
Prior art date
Application number
IL74215A
Other languages
English (en)
Other versions
IL74215A0 (en
Original Assignee
Searle & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Searle & Co filed Critical Searle & Co
Publication of IL74215A0 publication Critical patent/IL74215A0/xx
Publication of IL74215A publication Critical patent/IL74215A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL74215A 1984-02-03 1985-02-01 Derivatives of 5-phenyltetrazolo(1,5-a)(1,2,4)triazolo(1,5-c)pyrimidine-6-alkanols and pharmaceutical compositions containing them IL74215A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/576,700 US4562192A (en) 1984-02-03 1984-02-03 6-Substituted-5-phenyltetrazolo[1,5-a][1,2,4]triazole[1,5-c]pyrimidines, and pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
IL74215A0 IL74215A0 (en) 1985-05-31
IL74215A true IL74215A (en) 1988-09-30

Family

ID=24305604

Family Applications (1)

Application Number Title Priority Date Filing Date
IL74215A IL74215A (en) 1984-02-03 1985-02-01 Derivatives of 5-phenyltetrazolo(1,5-a)(1,2,4)triazolo(1,5-c)pyrimidine-6-alkanols and pharmaceutical compositions containing them

Country Status (16)

Country Link
US (1) US4562192A (es)
EP (1) EP0152841B1 (es)
JP (1) JPS60237087A (es)
AT (1) ATE35990T1 (es)
AU (1) AU571923B2 (es)
CA (1) CA1218061A (es)
DE (1) DE3563965D1 (es)
DK (1) DK44385A (es)
ES (4) ES8606354A1 (es)
FI (1) FI80699C (es)
GR (1) GR850297B (es)
IL (1) IL74215A (es)
NZ (1) NZ211025A (es)
PH (1) PH23945A (es)
PT (1) PT79909B (es)
ZA (1) ZA85802B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5071643A (en) * 1986-10-17 1991-12-10 R. P. Scherer Corporation Solvent system enhancing the solubility of pharmaceuticals for encapsulation
FR2678618B1 (fr) * 1991-07-05 1993-11-05 Upsa Laboratoires Nouveaux derives de triazolo pyrimidine antagonistes des recepteurs a l'angiotensine ii; leurs procedes de preparation, compositions pharmaceutiques les contenant.
US5358950A (en) * 1991-07-05 1994-10-25 Laboratoires Upsa Triazolopyrimidine derivatives which are angiotensin II receptor antagonists
JP5231829B2 (ja) 2007-02-15 2013-07-10 石原産業株式会社 ピリジル−トリアゾロピリミジン誘導体又はその塩、それらを含有する有害生物防除剤並びにそれらの製造方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3412094A (en) * 1967-06-21 1968-11-19 Searle & Co 5-alkyl-2-amino-4-azido-6-phenylpyrimidines and congeners
US4405780A (en) * 1979-08-08 1983-09-20 G. D. Searle & Co. 8-Substituted 7-phenyl-1,2,4,-triazolo[4,3-c]/[2,3-c]pyrimidines-5-amines and amides
US4483987A (en) * 1983-06-20 1984-11-20 G. D. Searle & Co. 8-Substituted 7-phenyl-1,2,4-triazolo[2,3-c]pyrimidines-5-amines and amides

Also Published As

Publication number Publication date
PT79909B (en) 1986-11-10
CA1218061A (en) 1987-02-17
PT79909A (en) 1985-03-01
ES540065A0 (es) 1986-04-01
ES549983A0 (es) 1986-12-16
FI850443A0 (fi) 1985-02-01
ZA85802B (en) 1986-03-26
NZ211025A (en) 1988-09-29
ATE35990T1 (de) 1988-08-15
DK44385A (da) 1985-08-04
ES8702411A1 (es) 1986-12-16
ES8702412A1 (es) 1987-01-01
ES8606354A1 (es) 1986-04-01
DE3563965D1 (de) 1988-09-01
ES8702410A1 (es) 1987-01-01
JPS60237087A (ja) 1985-11-25
US4562192A (en) 1985-12-31
AU3826085A (en) 1985-08-08
FI80699B (fi) 1990-03-30
DK44385D0 (da) 1985-01-31
FI80699C (fi) 1990-07-10
ES549982A0 (es) 1987-01-01
FI850443L (fi) 1985-08-04
IL74215A0 (en) 1985-05-31
GR850297B (es) 1985-05-29
PH23945A (en) 1990-01-23
EP0152841B1 (en) 1988-07-27
EP0152841A1 (en) 1985-08-28
ES549984A0 (es) 1987-01-01
AU571923B2 (en) 1988-04-28

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