ES549984A0 - Procedimiento para preparar 6-sustituido-5-feniltetrazol (1,5-a)-(1,2,4)triazol-(1,5-c)pirimidinas - Google Patents

Procedimiento para preparar 6-sustituido-5-feniltetrazol (1,5-a)-(1,2,4)triazol-(1,5-c)pirimidinas

Info

Publication number
ES549984A0
ES549984A0 ES549984A ES549984A ES549984A0 ES 549984 A0 ES549984 A0 ES 549984A0 ES 549984 A ES549984 A ES 549984A ES 549984 A ES549984 A ES 549984A ES 549984 A0 ES549984 A0 ES 549984A0
Authority
ES
Spain
Prior art keywords
substituted
phenyltetrazole
pyrimidines
triazol
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES549984A
Other languages
English (en)
Other versions
ES8702412A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GD Searle LLC
Original Assignee
GD Searle LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by GD Searle LLC filed Critical GD Searle LLC
Publication of ES549984A0 publication Critical patent/ES549984A0/es
Publication of ES8702412A1 publication Critical patent/ES8702412A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ES549984A 1984-02-03 1985-12-16 Procedimiento para preparar 6-sustituido-5-feniltetrazol (1,5-a)-(1,2,4)triazol-(1,5-c)pirimidinas Expired ES8702412A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/576,700 US4562192A (en) 1984-02-03 1984-02-03 6-Substituted-5-phenyltetrazolo[1,5-a][1,2,4]triazole[1,5-c]pyrimidines, and pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
ES549984A0 true ES549984A0 (es) 1987-01-01
ES8702412A1 ES8702412A1 (es) 1987-01-01

Family

ID=24305604

Family Applications (4)

Application Number Title Priority Date Filing Date
ES540065A Expired ES8606354A1 (es) 1984-02-03 1985-02-01 6-sustituido-5-feniltetrazol 1,5-a-1,2,4 triazol 1,5-c piri-midinas
ES549984A Expired ES8702412A1 (es) 1984-02-03 1985-12-16 Procedimiento para preparar 6-sustituido-5-feniltetrazol (1,5-a)-(1,2,4)triazol-(1,5-c)pirimidinas
ES549983A Expired ES8702411A1 (es) 1984-02-03 1985-12-16 Procedimiento para preparar 6-sustituido-5-feniltetrazol (1,5-a)-(1,2,4)triazol-(1,5-c)pirimidinas
ES549982A Expired ES8702410A1 (es) 1984-02-03 1985-12-16 Procedimiento para preparar 6-sustituido-5-feniltetrazol (1,5-a)-(1,2,4)triazol-(1,5-c)pirimidinas

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES540065A Expired ES8606354A1 (es) 1984-02-03 1985-02-01 6-sustituido-5-feniltetrazol 1,5-a-1,2,4 triazol 1,5-c piri-midinas

Family Applications After (2)

Application Number Title Priority Date Filing Date
ES549983A Expired ES8702411A1 (es) 1984-02-03 1985-12-16 Procedimiento para preparar 6-sustituido-5-feniltetrazol (1,5-a)-(1,2,4)triazol-(1,5-c)pirimidinas
ES549982A Expired ES8702410A1 (es) 1984-02-03 1985-12-16 Procedimiento para preparar 6-sustituido-5-feniltetrazol (1,5-a)-(1,2,4)triazol-(1,5-c)pirimidinas

Country Status (16)

Country Link
US (1) US4562192A (es)
EP (1) EP0152841B1 (es)
JP (1) JPS60237087A (es)
AT (1) ATE35990T1 (es)
AU (1) AU571923B2 (es)
CA (1) CA1218061A (es)
DE (1) DE3563965D1 (es)
DK (1) DK44385A (es)
ES (4) ES8606354A1 (es)
FI (1) FI80699C (es)
GR (1) GR850297B (es)
IL (1) IL74215A (es)
NZ (1) NZ211025A (es)
PH (1) PH23945A (es)
PT (1) PT79909B (es)
ZA (1) ZA85802B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5071643A (en) * 1986-10-17 1991-12-10 R. P. Scherer Corporation Solvent system enhancing the solubility of pharmaceuticals for encapsulation
US5358950A (en) * 1991-07-05 1994-10-25 Laboratoires Upsa Triazolopyrimidine derivatives which are angiotensin II receptor antagonists
FR2678618B1 (fr) * 1991-07-05 1993-11-05 Upsa Laboratoires Nouveaux derives de triazolo pyrimidine antagonistes des recepteurs a l'angiotensine ii; leurs procedes de preparation, compositions pharmaceutiques les contenant.
JP5231829B2 (ja) 2007-02-15 2013-07-10 石原産業株式会社 ピリジル−トリアゾロピリミジン誘導体又はその塩、それらを含有する有害生物防除剤並びにそれらの製造方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3412094A (en) * 1967-06-21 1968-11-19 Searle & Co 5-alkyl-2-amino-4-azido-6-phenylpyrimidines and congeners
US4405780A (en) * 1979-08-08 1983-09-20 G. D. Searle & Co. 8-Substituted 7-phenyl-1,2,4,-triazolo[4,3-c]/[2,3-c]pyrimidines-5-amines and amides
US4483987A (en) * 1983-06-20 1984-11-20 G. D. Searle & Co. 8-Substituted 7-phenyl-1,2,4-triazolo[2,3-c]pyrimidines-5-amines and amides

Also Published As

Publication number Publication date
IL74215A0 (en) 1985-05-31
DE3563965D1 (de) 1988-09-01
DK44385A (da) 1985-08-04
ES8702410A1 (es) 1987-01-01
GR850297B (es) 1985-05-29
NZ211025A (en) 1988-09-29
ES540065A0 (es) 1986-04-01
FI80699B (fi) 1990-03-30
AU3826085A (en) 1985-08-08
DK44385D0 (da) 1985-01-31
EP0152841B1 (en) 1988-07-27
ZA85802B (en) 1986-03-26
PT79909B (en) 1986-11-10
PT79909A (en) 1985-03-01
ES8606354A1 (es) 1986-04-01
US4562192A (en) 1985-12-31
FI80699C (fi) 1990-07-10
ES8702411A1 (es) 1986-12-16
CA1218061A (en) 1987-02-17
FI850443L (fi) 1985-08-04
ES549983A0 (es) 1986-12-16
FI850443A0 (fi) 1985-02-01
JPS60237087A (ja) 1985-11-25
PH23945A (en) 1990-01-23
ES8702412A1 (es) 1987-01-01
IL74215A (en) 1988-09-30
EP0152841A1 (en) 1985-08-28
AU571923B2 (en) 1988-04-28
ES549982A0 (es) 1987-01-01
ATE35990T1 (de) 1988-08-15

Similar Documents

Publication Publication Date Title
ES514664A0 (es) "un procedimiento para la preparacion de derivados de aminoacidos utiles como agentes antihipertensores".
HUT49592A (en) Process for producing bis/hydroxymethyl/-cyclobutyl-purines and pyrimidines, as well as pharmaceutical compositions comprising same
ES8603477A1 (es) Procedimiento para preparar una 1h-imidazo (4, 5-c) quinolin-4-amina
ES547169A0 (es) Procedimiento para la preparacion de 4,5-dihidro-3 (2h)-pi- ridazinonas sustituidas
ES542322A0 (es) Un procedimiento para la preparacion de derivados de la 2 pirimidinil-1-piperazina
ZA839693B (en) Substituted 4-aminomethylene-chromans and-chromens,processes for their preparation and their use in medicaments
HUT44128A (en) Process for producing substituted pyrimidines and pesticide compositions containing them as active components
PT86362A (en) Process for the preparation of anxiolytic compositions containing n-(1-azabicyclo ]2,2.2."-oct-3-yl) benzamides and thiobenzamides
JO1406B1 (en) Chemical compounds
EP0153152A3 (en) (2-oxo-1,2,3,5-tetrahydroimidazo-/2,1-b/quinnazolinyl)-oxyalkylamides, their preparation, compositions containing them and their use in making medicaments
PT78081A (en) Process for the preparation of n-piperazinylalkanoylanilydes useful as anti-hypertensive agents
FI915254A7 (fi) Tetrahydrofoolihaposta johdettuja diastereoisomeerisiä yhdisteitä, men etelmä niiden valmistamiseksi ja käyttö pelkistettyjen fosfaattien 6S- ja 6R-diastereoisomeerien synteesissä
EP0249248A3 (en) Purine derivatives
ES549984A0 (es) Procedimiento para preparar 6-sustituido-5-feniltetrazol (1,5-a)-(1,2,4)triazol-(1,5-c)pirimidinas
ATE41662T1 (de) Derivate von dihydro-1h-pyrrolo(1,2-c>imidazol3,5-dion zur aktivierung des wahrnehmungsvermoegens.
FR2520742B1 (fr) 1,3,4-thiadiazolo(3,2-a)pyrimidines substituees utiles comme medicaments et procede de leur preparation
DK478485A (da) 4-oxo-pyrido(2,3-d)pyrimidin-derivater, deres fremstilling og anvendelse
ES8507530A1 (es) Un procedimiento para la preparacion de aricoxicicloalcanolaminolaminoalquilen-aril-cetonas.
PT83141A (en) Process for the preparation of 3,7-disubstituted-3-cephem compounds useful as antimicrobial agents
DE3462495D1 (en) Process for the preparation of 2,2-dialkylpropyl isocyanates substituted in position 3 by heterocycles or by the dialkylamino group
ZA8683B (en) Antihypertensive agents,pharmaceutical compositions containing them and process for the preparation of the agents and compositions
FI850401L (fi) Maettade tricykliska kvaevehaltiga dioner saosom medel foer aktivering av fattningsfoeremaogan.