IL67925A0 - Laevorotatory isomer of mequitazine,its preparation and pharmaceutical compositions containing it - Google Patents

Laevorotatory isomer of mequitazine,its preparation and pharmaceutical compositions containing it

Info

Publication number
IL67925A0
IL67925A0 IL67925A IL6792583A IL67925A0 IL 67925 A0 IL67925 A0 IL 67925A0 IL 67925 A IL67925 A IL 67925A IL 6792583 A IL6792583 A IL 6792583A IL 67925 A0 IL67925 A0 IL 67925A0
Authority
IL
Israel
Prior art keywords
mequitazine
preparation
pharmaceutical compositions
compositions containing
laevorotatory isomer
Prior art date
Application number
IL67925A
Other languages
English (en)
Original Assignee
Pharmuka Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmuka Lab filed Critical Pharmuka Lab
Publication of IL67925A0 publication Critical patent/IL67925A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL67925A 1982-03-05 1983-02-16 Laevorotatory isomer of mequitazine,its preparation and pharmaceutical compositions containing it IL67925A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8203667A FR2522660A1 (fr) 1982-03-05 1982-03-05 Isomere levogyre de la mequitazine, son procede de preparation et medicaments le contenant

Publications (1)

Publication Number Publication Date
IL67925A0 true IL67925A0 (en) 1983-06-15

Family

ID=9271621

Family Applications (1)

Application Number Title Priority Date Filing Date
IL67925A IL67925A0 (en) 1982-03-05 1983-02-16 Laevorotatory isomer of mequitazine,its preparation and pharmaceutical compositions containing it

Country Status (13)

Country Link
EP (1) EP0089860A1 (xx)
JP (1) JPS58162588A (xx)
AU (1) AU1213283A (xx)
DK (1) DK57883A (xx)
ES (1) ES520339A0 (xx)
FI (1) FI830739L (xx)
FR (1) FR2522660A1 (xx)
GR (1) GR78102B (xx)
IL (1) IL67925A0 (xx)
MA (1) MA19731A1 (xx)
NO (1) NO830745L (xx)
PT (1) PT76348A (xx)
ZA (1) ZA831441B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1251161B (it) * 1991-08-07 1995-05-04 Derivati ammonio quaternari di (-) e (+)-3-(10 h-fenotiazin-10-ilmetil)-l-azabiciclo (2.2.2.)ottano e composizioni farmaceutiche che li contengono
FR2772029B1 (fr) * 1997-12-08 2000-02-25 Pf Medicament Procede de preparation de la mequitazine et nouvel intermediaire de synthese
FR2777278B1 (fr) * 1998-04-09 2000-06-30 Pf Medicament Nouveau procede de preparation de la 3-hydroxymethyl quinuclidine, intermediaire de synthese de la mequitazine
FR2876910B1 (fr) * 2004-10-21 2007-04-13 Pierre Fabre Medicament Sa Complexe comprenant la mequitazine, une cyclodextrine et un agent d'interaction
FR2896690B1 (fr) * 2006-01-30 2008-05-02 Pierre Fabre Medicament Sa Utilisation de l'enantiomere(s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique
FR2911606B1 (fr) * 2007-01-18 2009-04-17 Pierre Fabre Medicament Sa Nouveau derive de la quinuclidine utile dans la preparation de la mequitazine
FR2916142A1 (fr) * 2007-05-15 2008-11-21 Pierre Fabre Medicament Sa Forme pharmaceutique comprenant du (10-[(3s)-1-azabicyclo [2.2.2]oct-3-ylmethyl]-10h-phenothiazine se presentant sous une forme appropriee pour l'administration d'unde dose journaliere comprise entre 1 et 3 mg
FR2924344B1 (fr) * 2007-12-04 2010-04-16 Pf Medicament Utilisation de la mequitazine sous la forme de racemate ou d'enantiomeres pour la preparation d'un medicament destine au traitement ou a la prevention de pathologies impliquant les recepteurs histaminiques h4.
FR2970255B1 (fr) * 2011-01-10 2013-09-06 Pf Medicament Vinyl quinuclidine utile en tant qu'intermediaire de synthese dans la preparation de la (r)-mequitazine.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1250534A (xx) * 1969-03-03 1971-10-20

Also Published As

Publication number Publication date
JPS58162588A (ja) 1983-09-27
NO830745L (no) 1983-09-06
GR78102B (xx) 1984-09-26
FR2522660B1 (xx) 1984-09-21
DK57883A (da) 1983-09-06
DK57883D0 (da) 1983-02-10
AU1213283A (en) 1983-09-08
FI830739L (fi) 1983-09-06
PT76348A (fr) 1983-04-01
MA19731A1 (fr) 1983-02-25
FI830739A0 (fi) 1983-03-04
EP0089860A1 (fr) 1983-09-28
FR2522660A1 (fr) 1983-09-09
ES8403896A1 (es) 1984-04-01
ZA831441B (en) 1983-11-30
ES520339A0 (es) 1984-04-01

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