IL64621A - Chemical methods and intermediates for preparing substituted pyrimidinones - Google Patents
Chemical methods and intermediates for preparing substituted pyrimidinonesInfo
- Publication number
- IL64621A IL64621A IL64621A IL6462181A IL64621A IL 64621 A IL64621 A IL 64621A IL 64621 A IL64621 A IL 64621A IL 6462181 A IL6462181 A IL 6462181A IL 64621 A IL64621 A IL 64621A
- Authority
- IL
- Israel
- Prior art keywords
- intermediates
- chemical methods
- preparing substituted
- substituted pyrimidinones
- pyrimidine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/56—One oxygen atom and one sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Priority Applications (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IL7332681A IL73326A (en) | 1981-02-06 | 1981-12-22 | 4-hydroxy-pyrimidine derivatives and their preparation |
IL73325A IL73325A (en) | 1981-02-06 | 1981-12-22 | Pyrimidine derivatives |
IL73325A IL73325A0 (en) | 1981-02-06 | 1984-10-26 | Pyrimidine derivatives and their preparation |
IL73326A IL73326A0 (en) | 1981-02-06 | 1984-10-26 | Pyrimidine derivatives |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/232,105 US4352933A (en) | 1981-02-06 | 1981-02-06 | Chemical methods and intermediates for preparing substituted pyrimidinones |
Publications (2)
Publication Number | Publication Date |
---|---|
IL64621A0 IL64621A0 (en) | 1982-03-31 |
IL64621A true IL64621A (en) | 1985-10-31 |
Family
ID=22871897
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL64621A IL64621A (en) | 1981-02-06 | 1981-12-22 | Chemical methods and intermediates for preparing substituted pyrimidinones |
Country Status (12)
Country | Link |
---|---|
US (1) | US4352933A (fr) |
EP (2) | EP0058055B1 (fr) |
JP (1) | JPS57163378A (fr) |
KR (1) | KR880001473B1 (fr) |
AT (1) | ATE29882T1 (fr) |
DE (1) | DE3277373D1 (fr) |
DK (1) | DK49782A (fr) |
ES (1) | ES509274A0 (fr) |
GR (1) | GR75406B (fr) |
IE (1) | IE53005B1 (fr) |
IL (1) | IL64621A (fr) |
PT (1) | PT74293B (fr) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4477663A (en) * | 1981-02-06 | 1984-10-16 | Smithkline Beckman Corporation | Intermediates for preparing substituted pyrimidinones |
US4620001A (en) * | 1981-02-06 | 1986-10-28 | Smithkline Beckman Corporation | Chemical methods and intermediates for preparing substituted pyrimidinones |
US4675406A (en) * | 1981-02-06 | 1987-06-23 | Smithkline Beckman Corporation | Substituted pyrimidinones |
DK230482A (da) * | 1981-05-30 | 1982-12-01 | Smith Kline French Lab | Pyrimidonsalt og fremstilling heraf |
ATE21901T1 (de) * | 1982-07-30 | 1986-09-15 | Smith Kline French Lab | Aminopyrimidinone und ihre herstellung. |
US4772704A (en) * | 1983-09-21 | 1988-09-20 | Bristol-Myers Company | 2,5-disubstituted-4(3H)-pyrimidones having histamine H2 -receptor antagonist activity |
JP2807577B2 (ja) * | 1990-06-15 | 1998-10-08 | エーザイ株式会社 | 環状アミド誘導体 |
CA2309177A1 (fr) * | 1997-11-06 | 1999-05-20 | Stephen Allan Smith | Composes de pyrimidinone et compositions pharmaceutiques les renfermant |
EP2382865A1 (fr) | 2010-04-28 | 2011-11-02 | Bayer CropScience AG | Combinaisons d'agents actifs synergiques |
US9241486B2 (en) | 2012-08-31 | 2016-01-26 | Bayer Cropscience Lp | Combination and methods for controlling turfgrass pests |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1419994A (en) * | 1973-05-03 | 1976-01-07 | Smith Kline French Lab | Heterocyclicalkylaminotheterocyclic compounds methods for their preparation and compositions comprising them |
US4153793A (en) * | 1973-05-03 | 1979-05-08 | Smith Kline & French Laboratories Limited | Imidazo alkylamino pyrimidones |
US4145546A (en) * | 1975-10-02 | 1979-03-20 | Smith Kline & French Laboratories Limited | 4-Pyrimidone compounds |
US4216318A (en) * | 1975-12-29 | 1980-08-05 | Smith Kline & French Laboratories Limited | Heterocyclic alkyl 4-pyrimidones |
US4154834A (en) * | 1975-12-29 | 1979-05-15 | Smith Kline & French Laboratories Limited | Substituted isocytosines having histamine H2 -antagonist activity |
GB1582528A (en) * | 1977-03-25 | 1981-01-07 | Smith Kline French Lab | Amino pyrimidone derivatives |
IN151188B (fr) * | 1978-02-13 | 1983-03-05 | Smith Kline French Lab | |
AU527202B2 (en) * | 1978-04-11 | 1983-02-24 | Smith Kline & French Laboratories Limited | 2-aminopyrimidones |
ZA793443B (en) * | 1978-07-26 | 1980-12-31 | Glaxo Group Ltd | Heterocyclic derivatives |
US4374836A (en) * | 1978-10-16 | 1983-02-22 | Imperial Chemical Industries Ltd. | Antisecretory heterocyclic derivatives, process for their manufacture and pharmaceutical compositions containing them |
DE2962609D1 (en) * | 1979-04-11 | 1982-06-09 | Estel Hoogovens Bv | Expandable coiler mandrel |
CA1140129A (fr) * | 1979-08-21 | 1983-01-25 | Ronald J. King | Derives de la 4-pyrimidone |
-
1981
- 1981-02-06 US US06/232,105 patent/US4352933A/en not_active Expired - Fee Related
- 1981-12-22 IL IL64621A patent/IL64621A/xx unknown
-
1982
- 1982-01-15 PT PT74293A patent/PT74293B/pt unknown
- 1982-02-03 ES ES509274A patent/ES509274A0/es active Granted
- 1982-02-04 DE DE8282300562T patent/DE3277373D1/de not_active Expired
- 1982-02-04 EP EP82300562A patent/EP0058055B1/fr not_active Expired
- 1982-02-04 AT AT82300562T patent/ATE29882T1/de not_active IP Right Cessation
- 1982-02-04 EP EP84111114A patent/EP0141973A3/fr not_active Ceased
- 1982-02-05 DK DK49782A patent/DK49782A/da not_active Application Discontinuation
- 1982-02-05 GR GR67224A patent/GR75406B/el unknown
- 1982-02-05 JP JP57018094A patent/JPS57163378A/ja active Pending
- 1982-02-06 KR KR8200509A patent/KR880001473B1/ko not_active IP Right Cessation
- 1982-02-08 IE IE270/82A patent/IE53005B1/en unknown
Also Published As
Publication number | Publication date |
---|---|
KR880001473B1 (ko) | 1988-08-13 |
KR830009088A (ko) | 1983-12-17 |
EP0141973A2 (fr) | 1985-05-22 |
JPS57163378A (en) | 1982-10-07 |
US4352933A (en) | 1982-10-05 |
DK49782A (da) | 1982-08-07 |
IE53005B1 (en) | 1988-05-11 |
EP0058055A3 (en) | 1982-10-27 |
IL64621A0 (en) | 1982-03-31 |
GR75406B (fr) | 1984-07-13 |
EP0141973A3 (fr) | 1986-02-26 |
PT74293A (en) | 1982-02-01 |
PT74293B (pt) | 1983-06-28 |
ES8302723A1 (es) | 1983-01-16 |
ATE29882T1 (de) | 1987-10-15 |
EP0058055B1 (fr) | 1987-09-23 |
DE3277373D1 (en) | 1987-10-29 |
ES509274A0 (es) | 1983-01-16 |
EP0058055A2 (fr) | 1982-08-18 |
IE820270L (en) | 1982-08-06 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AU3811689A (en) | Alpha-arylacrylates substituted by a heterocyclic radical, and fungicides which contain these compounds | |
GB1447108A (en) | Pyrimidone compounds | |
IL64621A (en) | Chemical methods and intermediates for preparing substituted pyrimidinones | |
KR830005216A (ko) | 이미다조[4,5-b] 피리딘 유도체의 제조방법 | |
IE32035L (en) | Preparation of substituted vinyl pyrimidines and¹imidazolines | |
KR870006033A (ko) | 피리디닐 피리미딘 유도체의 제조 방법 | |
ES472182A1 (es) | Un procedimiento para la preparacion de nuevas 5-alquiltio- pirimidinas | |
HU9503825D0 (en) | Process for the preparation of fluoroathenylthio heterocyclic derivatives | |
EP0191298A3 (fr) | 1,6-Naphtyridine-2(1H)-ones utiles comme cardiotoniques et leur préparation | |
AU553927B2 (en) | Oxazolo- thiazolo- imidazolo (5,4-b) pyridines | |
YU46444B (sh) | Postupak za izradu derivata imidazola | |
UA8032A1 (uk) | Спосіб одержання 2-(4-метоксіфенілпропіоніл)аміно-6-н-пропіламіно-4,5,6,7-тетрагідробензотіазола у вигляді рацемата або (-)-енантіомера або його кислотно-аддітивної солі | |
AU6653190A (en) | Fungicides | |
GB583815A (en) | New pyrimidine compounds | |
GB1340160A (en) | 7-ureidocephalosporins | |
GB1418298A (en) | Process for the manufacture of amino-derivatives of n-heterocyclic compounds | |
GB1185039A (en) | Pyrimidine Derivatives and Compositions containing them | |
ATE17943T1 (de) | Als schaedlingsbekaempfungsmittel wirksame pyrimidin derivate. | |
JPS57176981A (en) | Dihydropyrimidine compound and its salts | |
ES8304094A1 (es) | Procedimiento para preparar una sal de pirimidona. | |
SU1496220A1 (ru) | Трис(2-гидроксиэтил)аммониевые соли гетерилтиоуксусных кислот, обладающие гиполипидемическим действием | |
ES8205410A1 (es) | Un procedimiento para preparar una pirazolo-piridinona | |
GB1467763A (en) | 2-substituted thio-1,4-benzodiazepine derivatives | |
ES8500913A1 (es) | "procedimiento para la obtencion de un compuesto derivado de la 2,4-dioxopirimidina" | |
SE7702797L (sv) | Forfarande for framstellning av 5-fluorouracilderivat |