IL60758A0 - Carbapenem derivatives,their preparation and pharmaceutical compositions containing them - Google Patents

Carbapenem derivatives,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL60758A0
IL60758A0 IL60758A IL6075880A IL60758A0 IL 60758 A0 IL60758 A0 IL 60758A0 IL 60758 A IL60758 A IL 60758A IL 6075880 A IL6075880 A IL 6075880A IL 60758 A0 IL60758 A0 IL 60758A0
Authority
IL
Israel
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
carbapenem derivatives
carbapenem
Prior art date
Application number
IL60758A
Other languages
English (en)
Original Assignee
Beecham Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group Ltd filed Critical Beecham Group Ltd
Publication of IL60758A0 publication Critical patent/IL60758A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D477/00Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • C07D477/10Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D477/12Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
    • C07D477/16Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 3
    • C07D477/20Sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL60758A 1979-08-10 1980-08-05 Carbapenem derivatives,their preparation and pharmaceutical compositions containing them IL60758A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7927901 1979-08-10
GB8012724 1980-04-17

Publications (1)

Publication Number Publication Date
IL60758A0 true IL60758A0 (en) 1980-10-26

Family

ID=26272503

Family Applications (1)

Application Number Title Priority Date Filing Date
IL60758A IL60758A0 (en) 1979-08-10 1980-08-05 Carbapenem derivatives,their preparation and pharmaceutical compositions containing them

Country Status (12)

Country Link
US (1) US4473578A (fr)
EP (2) EP0055990B1 (fr)
AU (1) AU6119680A (fr)
CA (1) CA1175841A (fr)
DE (1) DE3070269D1 (fr)
DK (1) DK344080A (fr)
ES (2) ES494136A0 (fr)
FI (1) FI802446A (fr)
GR (1) GR69935B (fr)
IL (1) IL60758A0 (fr)
NO (1) NO802377L (fr)
NZ (1) NZ194584A (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0072121A1 (fr) * 1981-08-08 1983-02-16 Beecham Group Plc Antibiotiques béta-lactamiques
US4552873A (en) * 1981-08-19 1985-11-12 Sankyo Company Limited Carbapenem compounds, and compositions containing them
EP0079167A1 (fr) * 1981-11-09 1983-05-18 Beecham Group Plc Un dérivé de carbapénème, préparation et application
EP0079244B1 (fr) * 1981-11-10 1986-12-30 Shionogi & Co., Ltd. Pluracidomycine du type B,C et D et leurs analogues, leurs production et un microorganisme utilisé à cette fin
US4556517A (en) * 1981-12-29 1985-12-03 Shionogi & Co., Ltd. Carbapenem derivatives
EP0091576B1 (fr) * 1982-03-26 1987-07-29 Hoechst Uk Limited Dérivés du 7-oxo-4-thia-1-azabicyclo(3,2,0)heptane
US4683301A (en) * 1982-04-08 1987-07-28 Bristol-Myers Company Carbapenem antibiotics
US4710568A (en) * 1982-04-09 1987-12-01 Bristol-Myers Company Carbapenem antibiotics
US4642341A (en) * 1982-04-09 1987-02-10 Bristol-Myers Company Carbapenem antibiotics
US4665170A (en) * 1982-06-18 1987-05-12 Bristol-Myers Company Carbapenem antibiotics
US4640799A (en) * 1982-06-18 1987-02-03 Bristol-Myers Company Carbapenem antibiotics
US4536335A (en) * 1982-06-18 1985-08-20 Bristol-Myers Company Carbapenem antibiotics
US4746736A (en) * 1982-09-28 1988-05-24 Bristol-Myers Company Carbapenem antibiotics
US4732977A (en) * 1982-09-28 1988-03-22 Bristol Myers Company Carbapenem antibiotics
EP0110280B1 (fr) * 1982-11-29 1994-10-12 Schering Corporation Procédé de préparation de dérivés de pénème
EP0137403A3 (fr) * 1983-09-28 1987-04-15 Takeda Chemical Industries, Ltd. Carbapénèmes, leur préparation et leur utilisation
US4698339A (en) * 1983-09-28 1987-10-06 Takeda Chemical Industries, Ltd. Carbapenems, their production and use
ZA848416B (en) * 1983-11-10 1986-06-25 Dow Chemical Co Fluorophenoxy compounds,herbicidal compositions and methods
US4717728A (en) * 1983-11-21 1988-01-05 Merck & Co., Inc. Cyclic amidinyl and cyclic guanidinyl thio carbapenems

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1531141A (en) * 1976-08-17 1978-11-01 Beecham Group Ltd Beta-lactam antibiotics
NL7802826A (nl) * 1977-04-08 1978-10-10 Merck & Co Inc Thienamycinederivaat, werkwijze voor het bereiden daarvan, alsmede farmaceutische preparaten.
US4235917A (en) * 1977-05-05 1980-11-25 Merck & Co., Inc. N-Alkyl-N-acyl derivatives of thienamycin
EP0001567B1 (fr) * 1977-10-13 1981-12-02 Sanraku-Ocean Co., Ltd. Antibiotiques PS-6 et PS-7 apparentés à la thiénamycine, procédé pour leur préparation et compositions les contenant
US4347368A (en) * 1977-10-19 1982-08-31 Merck & Co., Inc. 3-Substituted-6-substituted-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid
AU4061378A (en) * 1977-10-19 1980-04-17 Merck & Co., Inc. 1-azabicyclo (3.2.0) hept-2-enes
US4347367A (en) * 1977-10-19 1982-08-31 Merck & Co., Inc. 3-Substituted-6-(1'-hydroxyethyl)-7-oxo-1-azabicyclo[3.2.0]-hept-2-ene-2-carboxylic acid
EP0003740B1 (fr) * 1978-01-19 1982-01-27 Beecham Group Plc Antibiotiques dérivés de bêta-lactame, un procédé pour leur préparation et compositions pharmaceutiques les contenant
EP0004132A1 (fr) * 1978-03-04 1979-09-19 Beecham Group Plc Esters d'antibiotiques dérivés de béta-lactame, procédé de préparation et compositions pharmaceutiques les contenant et les composés utilisables comme agents antibactériens
US4203902A (en) * 1978-04-21 1980-05-20 Merck & Co., Inc. Process for preparing 6- and 2-substituted-1-carbadethiapen-2-em-3-carboxylic acids
EP0005348B1 (fr) * 1978-05-06 1982-09-22 Beecham Group Plc Dérivés de carbapénème, procédé pour leur préparation et compositions pharmaceutiques les contenant
EP0005349A1 (fr) * 1978-05-06 1979-11-14 Beecham Group Plc Alkylcarbapénèmes, leur préparation, compositions pharmaceutiques les contenant et les intermédiaires
EP0007753B1 (fr) * 1978-08-02 1982-08-25 Beecham Group Plc Agents antibactériens de bêta-lactame, un procédé pour leur préparation et compositions pharmaceutiques les contenant
DE2966187D1 (en) * 1978-08-23 1983-10-27 Beecham Group Plc Beta-lactam antibacterial compounds, their preparation and pharmaceutical compositions containing them
DE2961882D1 (en) * 1978-08-25 1982-03-04 Beecham Group Plc Beta-lactam anti-bacterials, compositions containing them and a process for their preparation
EP0008885B1 (fr) * 1978-09-09 1983-11-30 Beecham Group Plc Composés de bêta-lactame, leur préparation et application
EP0011173B1 (fr) * 1978-11-01 1983-05-11 Sanraku-Ocean Co., Ltd. Procédé pour la production de composés antibiotiques bêta-lactame
EP0017992A1 (fr) * 1979-04-19 1980-10-29 Merck & Co. Inc. Acides 1-carbadéthiapén-2-èm-carboxyliques substitués en position 2 et 6, procédés pour les préparer, compositions pharmaceutiques antibiotiques les contenant et procédé pour préparer des intermédiaires
US4376774A (en) * 1979-05-29 1983-03-15 Merck & Co., Inc. Antibiotic N-heterocyclyl thienamycin

Also Published As

Publication number Publication date
DE3070269D1 (en) 1985-04-18
EP0055990B1 (fr) 1986-06-11
ES499856A0 (es) 1982-01-16
EP0024832A1 (fr) 1981-03-11
ES8106308A1 (es) 1981-08-01
US4473578A (en) 1984-09-25
EP0024832B1 (fr) 1985-03-13
DK344080A (da) 1981-02-11
ES494136A0 (es) 1981-08-01
AU6119680A (en) 1981-02-12
GR69935B (fr) 1982-07-21
NZ194584A (en) 1983-05-31
ES8202010A1 (es) 1982-01-16
NO802377L (no) 1981-02-11
FI802446A (fi) 1981-02-11
EP0055990A1 (fr) 1982-07-14
CA1175841A (fr) 1984-10-09

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