IL60743A - 4-substituted piperidinobutyrophenones,their preparation and antipsychotic compositions comprising them - Google Patents
4-substituted piperidinobutyrophenones,their preparation and antipsychotic compositions comprising themInfo
- Publication number
- IL60743A IL60743A IL60743A IL6074380A IL60743A IL 60743 A IL60743 A IL 60743A IL 60743 A IL60743 A IL 60743A IL 6074380 A IL6074380 A IL 6074380A IL 60743 A IL60743 A IL 60743A
- Authority
- IL
- Israel
- Prior art keywords
- piperidinobutyrophenones
- substituted
- preparation
- antipsychotic
- compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/30—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
- C07D211/32—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Anesthesiology (AREA)
- Psychiatry (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/072,499 US4283404A (en) | 1979-09-04 | 1979-09-04 | Aroylethenylpiperidinobutyrophenone antipsychotic agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL60743A0 IL60743A0 (en) | 1980-10-26 |
| IL60743A true IL60743A (en) | 1984-07-31 |
Family
ID=22107983
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL60743A IL60743A (en) | 1979-09-04 | 1980-08-01 | 4-substituted piperidinobutyrophenones,their preparation and antipsychotic compositions comprising them |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US4283404A (fr) |
| JP (1) | JPS5640666A (fr) |
| AU (1) | AU538603B2 (fr) |
| BE (1) | BE885018A (fr) |
| CA (1) | CA1147735A (fr) |
| CH (1) | CH646951A5 (fr) |
| DE (1) | DE3031929A1 (fr) |
| ES (1) | ES8106144A1 (fr) |
| FR (1) | FR2464252A1 (fr) |
| GB (3) | GB2057444B (fr) |
| IL (1) | IL60743A (fr) |
| IT (1) | IT1145386B (fr) |
| NL (1) | NL8004836A (fr) |
| ZA (1) | ZA804664B (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0661266A1 (fr) * | 1993-12-27 | 1995-07-05 | Toa Eiyo Ltd. | Composés cycliques aminés substitués comme 5HT2 antagonistes |
| CA2651732C (fr) | 2006-05-18 | 2014-10-14 | Mannkind Corporation | Inhibiteurs de kinases intracellulaires |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3080372A (en) * | 1960-03-25 | 1963-03-05 | Res Lab Dr C Janssen | 1-aroylalkyl-4-arylpiperidine derivatives |
| GB979555A (en) * | 1962-01-17 | 1965-01-06 | Bellon Labor Sa Roger | New benzyl piperidyl ketones |
| US3689492A (en) * | 1965-09-10 | 1972-09-05 | Hans Detlef Schroeder | 1-{8 4{40 -OXO-4-(p-FLUOROPHENYL)-n-BUTYL-1{40 {9 -4-ACETYL-4-(m-HYDROXY-PHENYL-PIPERIDINE |
| US3646014A (en) * | 1966-05-09 | 1972-02-29 | Aldrich Chem Co Inc | Chemical compounds |
| US3484446A (en) * | 1967-01-16 | 1969-12-16 | Aldrich Chem Co Inc | 1-(3-(4-fluorobenzoyl)propyl) - and 1 - (1,1-ethylenedioxy - 1 - (4 - fluorophenyl)-4-butyl)-4-piperidyl carbamates |
| NL130760C (fr) * | 1967-01-25 | |||
| CH516557A (de) * | 1967-12-01 | 1971-12-15 | Thomae Gmbh Dr K | Verfahren zur Herstellung neuer Zimtsäureamide |
| CH532048A (de) * | 1967-12-01 | 1973-02-15 | Thomae Gmbh Dr K | Verfahren zur Herstellung von neuen Zimtsäureamiden |
| US3576810A (en) * | 1968-06-20 | 1971-04-27 | Robins Co Inc A H | 1-substituted-3-(-4)-aroylpiperidines |
| US3637712A (en) * | 1970-01-26 | 1972-01-25 | Bristol Myers Co | Piperidylpropanol compounds |
| US3852455A (en) * | 1970-11-27 | 1974-12-03 | Richardson Merrell Inc | 4-{8 4({60 hydroxybenzyl)piperidino{9 -4-fluorobutyrophenone derivatives as tranquilizers |
| ZA717147B (en) * | 1970-11-27 | 1972-07-26 | Richardson Merrell Inc | 4-(4-(alpha-hydroxybenzyl)piperidino)-4'-fluorobutyrophenone derivatives |
| US3816443A (en) * | 1972-02-17 | 1974-06-11 | Merck & Co Inc | 4-(benzothiazol-2-yl)fluoro phenyl-acetic acids |
| US3797932A (en) * | 1972-10-31 | 1974-03-19 | Eastman Kodak Co | Vibration isolation arrangement for aperture card photographic copying machine |
| US4101662A (en) * | 1973-05-03 | 1978-07-18 | A. H. Robins Company, Incorporated | Method for inhibiting emesis and compositions therefor |
| SE7409245L (fr) * | 1973-07-19 | 1975-01-20 | Robins Co Inc A H | |
| GB1535791A (en) * | 1975-05-07 | 1978-12-13 | Ferrosan Ab | Derivatives of 4-piperidinol |
| CH602642A5 (fr) * | 1975-11-14 | 1978-07-31 | Orgamol Sa |
-
1979
- 1979-09-04 US US06/072,499 patent/US4283404A/en not_active Expired - Lifetime
-
1980
- 1980-07-31 ZA ZA00804664A patent/ZA804664B/xx unknown
- 1980-08-01 IL IL60743A patent/IL60743A/xx unknown
- 1980-08-07 CA CA000357813A patent/CA1147735A/fr not_active Expired
- 1980-08-13 ES ES494223A patent/ES8106144A1/es not_active Expired
- 1980-08-15 AU AU61489/80A patent/AU538603B2/en not_active Ceased
- 1980-08-23 DE DE19803031929 patent/DE3031929A1/de not_active Withdrawn
- 1980-08-26 JP JP11652680A patent/JPS5640666A/ja active Granted
- 1980-08-27 NL NL8004836A patent/NL8004836A/nl not_active Application Discontinuation
- 1980-08-28 CH CH649280A patent/CH646951A5/de not_active IP Right Cessation
- 1980-09-01 BE BE0/201939A patent/BE885018A/fr not_active IP Right Cessation
- 1980-09-02 IT IT49598/80A patent/IT1145386B/it active
- 1980-09-02 GB GB8028273A patent/GB2057444B/en not_active Expired
- 1980-09-04 FR FR8019136A patent/FR2464252A1/fr active Granted
-
1983
- 1983-02-01 GB GB08302742A patent/GB2121032B/en not_active Expired
- 1983-02-08 GB GB08303500A patent/GB2121033B/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| GB2057444B (en) | 1983-11-30 |
| NL8004836A (nl) | 1981-03-06 |
| FR2464252B1 (fr) | 1983-05-27 |
| GB2121032A (en) | 1983-12-14 |
| BE885018A (fr) | 1980-12-31 |
| ES494223A0 (es) | 1981-08-01 |
| GB2121033B (en) | 1984-05-16 |
| IT8049598A0 (it) | 1980-09-02 |
| JPS6341389B2 (fr) | 1988-08-17 |
| GB2121032B (en) | 1984-06-06 |
| IT1145386B (it) | 1986-11-05 |
| CA1147735A (fr) | 1983-06-07 |
| CH646951A5 (de) | 1984-12-28 |
| GB2057444A (en) | 1981-04-01 |
| IL60743A0 (en) | 1980-10-26 |
| ES8106144A1 (es) | 1981-08-01 |
| ZA804664B (en) | 1981-07-29 |
| AU538603B2 (en) | 1984-08-23 |
| JPS5640666A (en) | 1981-04-16 |
| FR2464252A1 (fr) | 1981-03-06 |
| GB8302742D0 (en) | 1983-03-02 |
| DE3031929A1 (de) | 1981-03-26 |
| AU6148980A (en) | 1981-03-12 |
| GB2121033A (en) | 1983-12-14 |
| GB8303500D0 (en) | 1983-03-16 |
| US4283404A (en) | 1981-08-11 |
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