IL40533A - The preparation of 2,4-diamino-5-benzylpyrimidines and certain novel such compounds - Google Patents

The preparation of 2,4-diamino-5-benzylpyrimidines and certain novel such compounds

Info

Publication number
IL40533A
IL40533A IL40533A IL4053372A IL40533A IL 40533 A IL40533 A IL 40533A IL 40533 A IL40533 A IL 40533A IL 4053372 A IL4053372 A IL 4053372A IL 40533 A IL40533 A IL 40533A
Authority
IL
Israel
Prior art keywords
acid
formula
carbon
phenol
group
Prior art date
Application number
IL40533A
Other languages
English (en)
Other versions
IL40533A0 (en
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of IL40533A0 publication Critical patent/IL40533A0/xx
Publication of IL40533A publication Critical patent/IL40533A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Liquid Crystal Substances (AREA)
IL40533A 1971-10-12 1972-10-10 The preparation of 2,4-diamino-5-benzylpyrimidines and certain novel such compounds IL40533A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB4749271A GB1413471A (en) 1971-10-12 1971-10-12 2,4-diamino-5-benzylpyrimidines and a process for their preparation
GB5751271 1971-12-10

Publications (2)

Publication Number Publication Date
IL40533A0 IL40533A0 (en) 1972-12-29
IL40533A true IL40533A (en) 1976-03-31

Family

ID=26266064

Family Applications (2)

Application Number Title Priority Date Filing Date
IL40533A IL40533A (en) 1971-10-12 1972-10-10 The preparation of 2,4-diamino-5-benzylpyrimidines and certain novel such compounds
IL47450A IL47450A (en) 1971-10-12 1972-10-10 2,4-diamino-pyrimidine derivatives and their preparation

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL47450A IL47450A (en) 1971-10-12 1972-10-10 2,4-diamino-pyrimidine derivatives and their preparation

Country Status (21)

Country Link
US (1) US4116958A (da)
JP (1) JPS5328434B2 (da)
AR (1) AR197006A1 (da)
AU (1) AU474788B2 (da)
BE (1) BE789904A (da)
CA (1) CA997763A (da)
CH (1) CH593267A5 (da)
DD (1) DD102696A5 (da)
DE (2) DE2249532A1 (da)
DK (1) DK132795C (da)
ES (1) ES407479A1 (da)
FI (1) FI56176C (da)
FR (1) FR2157843B1 (da)
GB (1) GB1413471A (da)
IE (1) IE37072B1 (da)
IL (2) IL40533A (da)
NL (1) NL7213685A (da)
NO (1) NO137093C (da)
PL (1) PL78480B1 (da)
SE (2) SE405119B (da)
ZM (1) ZM16472A1 (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH592066A5 (da) * 1973-02-26 1977-10-14 Hoffmann La Roche
US4255574A (en) * 1973-02-26 1981-03-10 Hoffmann-La Roche Inc. Process for preparing 2,4-diamino-pyrimidines
NO791699L (no) * 1978-05-24 1979-11-27 Wellcome Found Benzylpyrimidinforbindelser og fremgangsmaate til deres fremstilling
IT1138146B (it) * 1981-08-11 1986-09-17 Proter Spa Processo per la produzione della 2,4-diammino-(3,5-dimetossi-4-metos sietossi-benzil)-pirimidina
JPS6175513A (ja) * 1985-07-01 1986-04-17 Hitachi Ltd シリコン結晶膜の製造方法
UA111630C2 (uk) 2011-10-06 2016-05-25 Сіс Рісорсез Лтд. Система для паління

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB920412A (en) * 1958-04-18 1963-03-06 Wellcome Found Pyrimidine derivatives and the manufacture thereof
DE1204678B (de) * 1958-04-18 1965-11-11 Wellcome Found Verfahren zur Herstellung von in 5'-oder 6'-Stellung bromsubstituierten 2, 4-Diamino-5-benzylpyrimidinen
DE1303727B (de) * 1959-09-03 1976-02-05 Ausscheidung aus: 14 45 176 The Wellcome Foundation Ltd., London Alpha-Arylidensubstituierte Propioni-Irile
GB1142654A (en) * 1965-10-28 1969-02-12 Wellcome Found Cyano-acetals and their use in benzylpyrimidine synthesis
GB1128234A (en) * 1966-02-19 1968-09-25 Wellcome Found 5-benzylpyrimidine derivatives and process for the preparation thereof
BE710100A (da) * 1967-02-02 1968-07-30
GB1247347A (en) * 1968-01-19 1971-09-22 Burroughs Wellcome Co Pyrimidine derivatives, the preparation thereof and compositions containing the same
DK120706B (da) * 1969-01-27 1971-07-05 Egyt Gyogyszervegyeszeti Gyar Fremgangsmåde til fremstilling af 2,4-diamino-5-(3',4',5'-trimethoxybenzyl)-pyrimidin.
US3819629A (en) * 1970-02-10 1974-06-25 Burroughs Wellcome Co Method for preparing 2,4-diamino-5-(3,4,5-trimethoxybenzyl)pyrimidine

Also Published As

Publication number Publication date
BE789904A (fr) 1973-04-10
DK132795B (da) 1976-02-09
DK132795C (da) 1976-07-12
SE7506083L (sv) 1975-05-28
AR197006A1 (es) 1974-03-08
DE2249532C2 (da) 1987-06-19
JPS5328434B2 (da) 1978-08-15
JPS4844270A (da) 1973-06-26
IL47450A (en) 1976-03-31
DD102696A5 (da) 1973-12-20
IL40533A0 (en) 1972-12-29
NO137093B (no) 1977-09-19
FR2157843A1 (da) 1973-06-08
FI56176B (fi) 1979-08-31
DE2249532A1 (de) 1973-04-26
AU474788B2 (en) 1976-08-05
GB1413471A (en) 1975-11-12
AU4766772A (en) 1974-04-26
DE2264413A1 (de) 1974-04-18
NL7213685A (da) 1973-04-16
PL78480B1 (en) 1975-06-30
CA997763A (en) 1976-09-28
IE37072B1 (en) 1977-04-27
FR2157843B1 (da) 1977-01-14
ZM16472A1 (en) 1974-04-22
US4116958A (en) 1978-09-26
SE413506B (sv) 1980-06-02
CH593267A5 (da) 1977-11-30
FI56176C (fi) 1979-12-10
NO137093C (no) 1977-12-28
IE37072L (en) 1973-04-12
ES407479A1 (es) 1976-02-01
SE405119B (sv) 1978-11-20
DE2264413C2 (da) 1987-05-21

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