IL39341A - Thieno(3,2-d)pyrimidines,their preparation and pharmaceutical compositions containing them - Google Patents

Thieno(3,2-d)pyrimidines,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL39341A
IL39341A IL39341A IL3934172A IL39341A IL 39341 A IL39341 A IL 39341A IL 39341 A IL39341 A IL 39341A IL 3934172 A IL3934172 A IL 3934172A IL 39341 A IL39341 A IL 39341A
Authority
IL
Israel
Prior art keywords
thieno
pyrimidines
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
IL39341A
Other languages
English (en)
Other versions
IL39341A0 (en
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19712121950 external-priority patent/DE2121950A1/de
Priority claimed from DE19712137341 external-priority patent/DE2137341A1/de
Priority claimed from DE19722215299 external-priority patent/DE2215299A1/de
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of IL39341A0 publication Critical patent/IL39341A0/xx
Publication of IL39341A publication Critical patent/IL39341A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
IL39341A 1971-05-04 1972-05-03 Thieno(3,2-d)pyrimidines,their preparation and pharmaceutical compositions containing them IL39341A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19712121950 DE2121950A1 (en) 1971-05-04 1971-05-04 Thieno(3,2-d)pyrimidine derivs - with thrombocyte aggregation inhibiting activity
DE19712137341 DE2137341A1 (de) 1971-07-26 1971-07-26 Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine
DE19722215299 DE2215299A1 (de) 1972-03-29 1972-03-29 Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine

Publications (2)

Publication Number Publication Date
IL39341A0 IL39341A0 (en) 1972-07-26
IL39341A true IL39341A (en) 1975-08-31

Family

ID=27183398

Family Applications (1)

Application Number Title Priority Date Filing Date
IL39341A IL39341A (en) 1971-05-04 1972-05-03 Thieno(3,2-d)pyrimidines,their preparation and pharmaceutical compositions containing them

Country Status (15)

Country Link
US (1) US3888851A (de)
AT (1) AT318619B (de)
AU (1) AU4181572A (de)
BE (1) BE783044A (de)
BG (1) BG20593A3 (de)
DD (1) DD97656A5 (de)
DK (1) DK129844B (de)
ES (1) ES402302A1 (de)
FR (1) FR2135294B1 (de)
GB (1) GB1393161A (de)
HU (1) HU163960B (de)
IL (1) IL39341A (de)
NL (1) NL7206041A (de)
PL (1) PL82381B1 (de)
RO (1) RO62428A (de)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4054656A (en) * 1975-09-10 1977-10-18 Mead Johnson & Company Thieno[2,3-d]pyrimidine antiallergic agents
US5098902A (en) * 1991-03-18 1992-03-24 Warner-Lambert Company Method of treating neurodegenerative diseases
CA2129337A1 (en) * 1992-02-19 1993-09-02 Jotham W. Coe Heterocyclic compounds for enhancing antitumor activity
PL340412A1 (en) 1997-10-20 2001-01-29 Hoffmann La Roche Bicyclic kinase inhibitors
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
GB0423653D0 (en) 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
CN101163706A (zh) * 2005-04-21 2008-04-16 贝林格尔·英格海姆国际有限公司 用于治疗炎性疾病的二氢噻吩并嘧啶
KR101402474B1 (ko) 2006-04-26 2014-06-19 제넨테크, 인크. 포스포이노시티드 3-키나제 억제제 화합물 및 이를 포함하는 약학적 조성물
BRPI0710874A2 (pt) 2006-04-26 2012-02-14 Hoffmann La Roche compostos de tienopirimidina, processos de produção dos referidos compostos, composições farmacêuticas contendo os mesmos, kit, produto, e usos dos compostos
EP2041139B1 (de) 2006-04-26 2011-11-09 F. Hoffmann-La Roche AG Pharmazeutische verbindungen
TWI499420B (zh) 2006-12-07 2015-09-11 Hoffmann La Roche 肌醇磷脂3-激酶抑制劑化合物及使用方法
KR101507182B1 (ko) * 2006-12-07 2015-03-30 제넨테크, 인크. 포스포이노시타이드 3-키나제 억제제 화합물 및 그의 사용 방법
CA2704711C (en) 2007-09-24 2016-07-05 Genentech, Inc. Thiazolopyrimidine p13k inhibitor compounds and methods of use
BRPI0817781A2 (pt) * 2007-10-19 2019-09-24 Boehringer Ingelheim Int piperazino-diidroteinopirimidinas substituídas com heterociclo
US8354528B2 (en) 2007-10-25 2013-01-15 Genentech, Inc. Process for making thienopyrimidine compounds
GB0721095D0 (en) 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
AU2010224125B2 (en) 2009-03-12 2015-05-14 Genentech, Inc. Combinations of phosphoinositide 3-kinase inhibitor compounds and chemotherapeutic agents for the treatment of hematopoietic malignancies
SG175708A1 (en) * 2009-05-27 2011-12-29 Genentech Inc Bicyclic pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
SG182247A1 (en) * 2009-05-27 2012-08-30 Hoffmann La Roche Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
JP2013528787A (ja) 2010-04-16 2013-07-11 ジェネンテック, インコーポレイテッド Pi3k/aktキナーゼ経路インヒビターの効果の予測バイオマーカーとしてのfox03a
US20140004209A1 (en) 2010-12-22 2014-01-02 Genentech, Inc. Autophagy inducer and inhibitor combination therapy for the treatment of neoplasms
KR102182488B1 (ko) 2013-02-25 2020-11-24 제넨테크, 인크. 약물 내성 akt 돌연변이체의 검출 및 치료를 위한 방법 및 조성물
GB201410816D0 (en) * 2014-06-17 2014-07-30 Ucb Biopharma Sprl And Katholieke Universiteit Leuven Therapeutic agents

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3259623A (en) * 1963-06-14 1966-07-05 Olin Mathieson Process for preparing 2-(secondary amino)-halogenopyrimidines
DE1470356A1 (de) * 1964-01-15 1970-04-30 Thomae Gmbh Dr K Neue Thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
US3210368A (en) * 1964-09-29 1965-10-05 Ciba Geigy Corp Certain 2-amino-4-aryl-5-n, n-disubstituted amino-lower alkyl-thiazole compounds

Also Published As

Publication number Publication date
FR2135294A1 (de) 1972-12-15
GB1393161A (en) 1975-05-07
HU163960B (de) 1973-11-28
DK129844B (da) 1974-11-25
FR2135294B1 (de) 1975-10-17
DK129844C (de) 1975-05-12
NL7206041A (de) 1972-11-07
ES402302A1 (es) 1975-04-01
AT318619B (de) 1974-11-11
AU4181572A (en) 1973-11-08
DD97656A5 (de) 1973-05-12
US3888851A (en) 1975-06-10
BG20593A3 (bg) 1975-12-05
IL39341A0 (en) 1972-07-26
BE783044A (fr) 1972-11-06
RO62428A (fr) 1978-01-15
PL82381B1 (de) 1975-10-31

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