IL35823A - Beating Process in 61 - Methyl - A9 - Fluoro - B11, A71, 12 Trihydroxy 1, 4 - Preganadian - 3, 02 - Dion and its 12 - Acylates - Google Patents

Beating Process in 61 - Methyl - A9 - Fluoro - B11, A71, 12 Trihydroxy 1, 4 - Preganadian - 3, 02 - Dion and its 12 - Acylates

Info

Publication number
IL35823A
IL35823A IL35823A IL3582370A IL35823A IL 35823 A IL35823 A IL 35823A IL 35823 A IL35823 A IL 35823A IL 3582370 A IL3582370 A IL 3582370A IL 35823 A IL35823 A IL 35823A
Authority
IL
Israel
Prior art keywords
acid
compound
new process
process according
yielding
Prior art date
Application number
IL35823A
Other languages
English (en)
Hebrew (he)
Other versions
IL35823A0 (en
Original Assignee
Villax I
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Villax I filed Critical Villax I
Publication of IL35823A0 publication Critical patent/IL35823A0/xx
Publication of IL35823A publication Critical patent/IL35823A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C07J5/0046Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
    • C07J5/0061Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16
    • C07J5/0069Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group
    • C07J5/0076Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group by an alkyl group

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Table Devices Or Equipment (AREA)
IL35823A 1969-12-13 1970-12-10 Beating Process in 61 - Methyl - A9 - Fluoro - B11, A71, 12 Trihydroxy 1, 4 - Preganadian - 3, 02 - Dion and its 12 - Acylates IL35823A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PT5292369 1969-12-13

Publications (2)

Publication Number Publication Date
IL35823A0 IL35823A0 (en) 1971-02-25
IL35823A true IL35823A (en) 1977-08-31

Family

ID=20081704

Family Applications (3)

Application Number Title Priority Date Filing Date
IL49763A IL49763A (en) 1969-12-13 1970-12-10 B 61 - Methyl - 9, 11 - Epoxy - A 71 - Hydroxy - 1, 4 - Pragadian - 3, 02 - Discussion and preparation
IL35823A IL35823A (en) 1969-12-13 1970-12-10 Beating Process in 61 - Methyl - A9 - Fluoro - B11, A71, 12 Trihydroxy 1, 4 - Preganadian - 3, 02 - Dion and its 12 - Acylates
IL49763A IL49763A0 (en) 1969-12-13 1976-06-10 Novel 9,11-epoxy-pregnadienes and their preparation

Family Applications Before (1)

Application Number Title Priority Date Filing Date
IL49763A IL49763A (en) 1969-12-13 1970-12-10 B 61 - Methyl - 9, 11 - Epoxy - A 71 - Hydroxy - 1, 4 - Pragadian - 3, 02 - Discussion and preparation

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL49763A IL49763A0 (en) 1969-12-13 1976-06-10 Novel 9,11-epoxy-pregnadienes and their preparation

Country Status (15)

Country Link
US (1) US3792046A (US20020128544A1-20020912-P00008.png)
JP (3) JPS508080B1 (US20020128544A1-20020912-P00008.png)
AT (1) AT304774B (US20020128544A1-20020912-P00008.png)
BE (1) BE760236A (US20020128544A1-20020912-P00008.png)
CA (1) CA932321A (US20020128544A1-20020912-P00008.png)
CH (1) CH551395A (US20020128544A1-20020912-P00008.png)
DE (1) DE2059050A1 (US20020128544A1-20020912-P00008.png)
DK (1) DK130991B (US20020128544A1-20020912-P00008.png)
ES (1) ES386385A1 (US20020128544A1-20020912-P00008.png)
FR (1) FR2081356B1 (US20020128544A1-20020912-P00008.png)
GB (1) GB1328998A (US20020128544A1-20020912-P00008.png)
IL (3) IL49763A (US20020128544A1-20020912-P00008.png)
NL (1) NL166694C (US20020128544A1-20020912-P00008.png)
NO (1) NO136049C (US20020128544A1-20020912-P00008.png)
ZA (1) ZA708393B (US20020128544A1-20020912-P00008.png)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58212359A (ja) * 1982-05-25 1983-12-10 マグネツト・モ−トル・ゲゼルシヤフト・フユア・マグネツトモ−トリツシエ・テクニ−ク・ミツト・ベシユレンクテル・ハフツンク 回転電気機械
JPS6261175U (US20020128544A1-20020912-P00008.png) * 1985-10-02 1987-04-16
JPS62135570U (US20020128544A1-20020912-P00008.png) * 1986-02-19 1987-08-26
EP1399464A1 (en) * 2001-06-18 2004-03-24 PHARMACIA & UPJOHN COMPANY Process to prepare 11beta, 17alpha, 21-trihydroxy-6alpha-methylpregna-1,4-diene-3,20-dione 21-acetate
US20040006240A1 (en) * 2001-06-18 2004-01-08 Pearlman Bruce Allen Process to prepare 11beta,17alpha ,21-trihydroxy-6alpha-methylpregna-1,4-diene-3,20-dione 21-acetate
CN101555268B (zh) * 2009-05-21 2011-11-30 广西万德药业股份有限公司 一种糖皮质激素类9,11环氧物中间体制备方法
CN102304163A (zh) * 2011-07-11 2012-01-04 浙江仙居仙乐药业有限公司 一种倍他米松上氟合成方法
CN104945464B (zh) * 2015-04-17 2016-10-26 浙江仙居仙乐药业有限公司 一种倍他米松环氧水解物的合成方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1274397A (fr) * 1958-12-16 1961-10-27 Chimiotherapie Lab Franc Procédé de préparation de dérivés 9alpha-fluoro 16alpha-méthyl delta1, 4-pregnadiènes
FR1243528A (fr) * 1959-08-05 1960-10-14 Chimiotherapie Lab Franc Procédé d'acétoxylation de stéroïdes en 21 par l'intermédiaire de dérivés diiodés

Also Published As

Publication number Publication date
DK130991B (da) 1975-05-12
NL166694C (nl) 1981-09-15
IL35823A0 (en) 1971-02-25
IL49763A0 (en) 1976-08-31
AT304774B (de) 1973-01-25
NL166694B (nl) 1981-04-15
JPS5721279B1 (US20020128544A1-20020912-P00008.png) 1982-05-06
GB1328998A (en) 1973-09-05
ZA708393B (en) 1972-07-26
NO136049B (US20020128544A1-20020912-P00008.png) 1977-04-04
FR2081356B1 (US20020128544A1-20020912-P00008.png) 1976-09-17
CA932321A (en) 1973-08-21
NO136049C (no) 1977-07-13
JPS5721280B1 (US20020128544A1-20020912-P00008.png) 1982-05-06
IL49763A (en) 1977-08-31
US3792046A (en) 1974-02-12
DK130991C (US20020128544A1-20020912-P00008.png) 1975-12-08
NL7017904A (US20020128544A1-20020912-P00008.png) 1971-06-15
JPS508080B1 (US20020128544A1-20020912-P00008.png) 1975-04-01
FR2081356A1 (US20020128544A1-20020912-P00008.png) 1971-12-03
ES386385A1 (es) 1973-03-16
CH551395A (de) 1974-07-15
DE2059050A1 (de) 1972-04-06
BE760236A (fr) 1971-05-17

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