IL295149A - Therapeutic combinations comprising ubiquitin-specific-processing protease 1 (usp1) inhibitors and poly (adp-ribose) polymerase (parp) inhibitors - Google Patents
Therapeutic combinations comprising ubiquitin-specific-processing protease 1 (usp1) inhibitors and poly (adp-ribose) polymerase (parp) inhibitorsInfo
- Publication number
- IL295149A IL295149A IL295149A IL29514922A IL295149A IL 295149 A IL295149 A IL 295149A IL 295149 A IL295149 A IL 295149A IL 29514922 A IL29514922 A IL 29514922A IL 295149 A IL295149 A IL 295149A
- Authority
- IL
- Israel
- Prior art keywords
- cancer
- inhibitor
- usp1
- parp
- pharmaceutically acceptable
- Prior art date
Links
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Landscapes
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| WO2018165615A1 (en) * | 2017-03-09 | 2018-09-13 | The Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College | Parp-1 and methods of use thereof |
| KR20190130625A (ko) * | 2017-03-27 | 2019-11-22 | 테사로, 인코포레이티드 | 니라파립 제제 |
| US11485736B2 (en) * | 2018-12-20 | 2022-11-01 | KSQ Therapeutics, Inc. | Substituted pyrazolopyrimidines and substituted purines and their use as ubiquitin-specific-processing protease 1 (USP1) inhibitors |
| US20230065636A1 (en) * | 2020-01-15 | 2023-03-02 | KSQ Therapeutics, Inc. | Compositions of substituted pyrazolopyrimidines and uses thereof |
| WO2021163530A1 (en) * | 2020-02-14 | 2021-08-19 | KSQ Therapeutics, Inc. | Therapeutic combinations comprising ubiquitin-specific-processing protease 1 (usp1) inhibitors and poly (adp-ribose) polymerase (parp) inhibitors |
| KR20230098186A (ko) * | 2020-10-30 | 2023-07-03 | 케이에스큐 세러퓨틱스 인코포레이티드 | 치환된 피라졸로피리미딘의 고체 상태 형태 및 이의 용도 |
-
2021
- 2021-02-12 WO PCT/US2021/017912 patent/WO2021163530A1/en not_active Ceased
- 2021-02-12 MX MX2022009818A patent/MX2022009818A/es unknown
- 2021-02-12 US US17/904,159 patent/US20230277533A1/en not_active Abandoned
- 2021-02-12 KR KR1020227027461A patent/KR20220140732A/ko active Pending
- 2021-02-12 CA CA3168009A patent/CA3168009A1/en active Pending
- 2021-02-12 JP JP2022548896A patent/JP2023514568A/ja active Pending
- 2021-02-12 AU AU2021218805A patent/AU2021218805A1/en active Pending
- 2021-02-12 IL IL295149A patent/IL295149A/en unknown
- 2021-02-12 EP EP21754160.6A patent/EP4103165A4/en not_active Withdrawn
- 2021-02-12 CN CN202180013564.7A patent/CN115066235A/zh active Pending
- 2021-02-17 TW TW110105371A patent/TW202140026A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20220140732A (ko) | 2022-10-18 |
| US20230277533A1 (en) | 2023-09-07 |
| MX2022009818A (es) | 2022-09-05 |
| EP4103165A4 (en) | 2024-02-28 |
| TW202140026A (zh) | 2021-11-01 |
| CN115066235A (zh) | 2022-09-16 |
| WO2021163530A1 (en) | 2021-08-19 |
| EP4103165A1 (en) | 2022-12-21 |
| AU2021218805A1 (en) | 2022-09-01 |
| JP2023514568A (ja) | 2023-04-06 |
| CA3168009A1 (en) | 2021-08-19 |
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