IL204520A - Oxadiazole diaryl compounds, their preparations and pharmaceutical preparations containing them - Google Patents

Oxadiazole diaryl compounds, their preparations and pharmaceutical preparations containing them

Info

Publication number
IL204520A
IL204520A IL204520A IL20452010A IL204520A IL 204520 A IL204520 A IL 204520A IL 204520 A IL204520 A IL 204520A IL 20452010 A IL20452010 A IL 20452010A IL 204520 A IL204520 A IL 204520A
Authority
IL
Israel
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
diaryl compounds
oxadiazole
Prior art date
Application number
IL204520A
Other languages
English (en)
Hebrew (he)
Other versions
IL204520A0 (en
Inventor
Agnes Bombrun
Anna Quattropani
Cyril Montagne
Wolfgang Sauer
Original Assignee
Agnes Bombrun
Merck Serono Sa
Anna Quattropani
Cyril Montagne
Wolfgang Sauer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agnes Bombrun, Merck Serono Sa, Anna Quattropani, Cyril Montagne, Wolfgang Sauer filed Critical Agnes Bombrun
Publication of IL204520A0 publication Critical patent/IL204520A0/en
Publication of IL204520A publication Critical patent/IL204520A/en

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • C—CHEMISTRY; METALLURGY
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    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/07—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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IL204520A 2007-10-04 2010-03-16 Oxadiazole diaryl compounds, their preparations and pharmaceutical preparations containing them IL204520A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07117925 2007-10-04
US99813607P 2007-10-09 2007-10-09
PCT/EP2008/063185 WO2009043890A1 (en) 2007-10-04 2008-10-01 Oxadiazole diaryl compounds

Publications (2)

Publication Number Publication Date
IL204520A0 IL204520A0 (en) 2010-11-30
IL204520A true IL204520A (en) 2016-04-21

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Family Applications (1)

Application Number Title Priority Date Filing Date
IL204520A IL204520A (en) 2007-10-04 2010-03-16 Oxadiazole diaryl compounds, their preparations and pharmaceutical preparations containing them

Country Status (15)

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US (2) US8404676B2 (OSRAM)
EP (1) EP2193126B1 (OSRAM)
JP (3) JP5727223B2 (OSRAM)
KR (1) KR20100083814A (OSRAM)
CN (2) CN101815707B (OSRAM)
AR (1) AR068730A1 (OSRAM)
AU (1) AU2008306886B2 (OSRAM)
BR (1) BRPI0817597A2 (OSRAM)
CA (1) CA2696829C (OSRAM)
EA (1) EA201070423A1 (OSRAM)
ES (1) ES2547877T3 (OSRAM)
IL (1) IL204520A (OSRAM)
MX (1) MX2010003614A (OSRAM)
WO (1) WO2009043890A1 (OSRAM)
ZA (1) ZA201001217B (OSRAM)

Families Citing this family (20)

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CN101815707A (zh) 2010-08-25
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JP2015025001A (ja) 2015-02-05
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BRPI0817597A2 (pt) 2015-04-07
CA2696829A1 (en) 2009-04-09
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US8404676B2 (en) 2013-03-26
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EA201070423A1 (ru) 2010-10-29
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