IL191586A0 - Heterocycle-substituted 3-alkyl azetidine derivatives - Google Patents

Heterocycle-substituted 3-alkyl azetidine derivatives

Info

Publication number
IL191586A0
IL191586A0 IL191586A IL19158608A IL191586A0 IL 191586 A0 IL191586 A0 IL 191586A0 IL 191586 A IL191586 A IL 191586A IL 19158608 A IL19158608 A IL 19158608A IL 191586 A0 IL191586 A0 IL 191586A0
Authority
IL
Israel
Prior art keywords
heterocycle
substituted
azetidine derivatives
alkyl
alkyl azetidine
Prior art date
Application number
IL191586A
Other languages
English (en)
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Publication of IL191586A0 publication Critical patent/IL191586A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL191586A 2005-11-28 2008-05-20 Heterocycle-substituted 3-alkyl azetidine derivatives IL191586A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74018305P 2005-11-28 2005-11-28
PCT/US2006/045328 WO2007062193A1 (en) 2005-11-28 2006-11-22 Heterocycle-substituted 3-alkyl azetidine derivatives

Publications (1)

Publication Number Publication Date
IL191586A0 true IL191586A0 (en) 2008-12-29

Family

ID=37779312

Family Applications (1)

Application Number Title Priority Date Filing Date
IL191586A IL191586A0 (en) 2005-11-28 2008-05-20 Heterocycle-substituted 3-alkyl azetidine derivatives

Country Status (15)

Country Link
EP (1) EP1954692A1 (ko)
KR (1) KR20080073721A (ko)
AR (1) AR058199A1 (ko)
BR (1) BRPI0619018A2 (ko)
CR (1) CR10014A (ko)
DO (1) DOP2006000261A (ko)
EC (1) ECSP088477A (ko)
IL (1) IL191586A0 (ko)
MA (1) MA30086B1 (ko)
NO (1) NO20082919L (ko)
PE (1) PE20070647A1 (ko)
RU (1) RU2008126248A (ko)
SV (1) SV2009002917A (ko)
TW (1) TW200804317A (ko)
WO (1) WO2007062193A1 (ko)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7906652B2 (en) * 2005-11-28 2011-03-15 Merck Sharp & Dohme Corp. Heterocycle-substituted 3-alkyl azetidine derivatives
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
WO2009054923A2 (en) * 2007-10-24 2009-04-30 Merck & Co., Inc. Synthesis and crystalline forms of cb-1 antagonist/inverse agonist
US9440948B2 (en) 2010-09-03 2016-09-13 University Of Florida Research Foundation, Inc. Nicotine compounds and analogs thereof, synthetic methods of making compounds, and methods of use
EP2683699B1 (de) 2011-03-08 2015-06-24 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120056A1 (de) 2011-03-08 2012-09-13 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120054A1 (de) 2011-03-08 2012-09-13 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120052A1 (de) 2011-03-08 2012-09-13 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
US8828995B2 (en) 2011-03-08 2014-09-09 Sanofi Branched oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2805810B1 (fr) * 2000-03-03 2002-04-26 Aventis Pharma Sa Compositions pharmaceutiques contenant des derives de 3- amino-azetidine, les nouveaux derives et leur preparation
FR2805817B1 (fr) * 2000-03-03 2002-04-26 Aventis Pharma Sa Compositions pharmaceutiques contenant des derives d'azetidine, les nouveaux derives d'azetidine et leur preparation
FR2805818B1 (fr) * 2000-03-03 2002-04-26 Aventis Pharma Sa Derives d'azetidine, leur preparation et les compositions pharmaceutiques les contenant
US7485732B2 (en) * 2003-06-11 2009-02-03 Merck & Co., Inc. Substituted 3-alkyl and 3-alkenyl azetidine derivatives
CN101426500A (zh) * 2005-05-02 2009-05-06 默克公司 治疗糖尿病和肥胖症的二肽基肽酶iv抑制剂和cb1受体拮抗剂的药物组合物

Also Published As

Publication number Publication date
RU2008126248A (ru) 2010-01-10
MA30086B1 (fr) 2008-12-01
BRPI0619018A2 (pt) 2016-11-29
PE20070647A1 (es) 2007-08-11
EP1954692A1 (en) 2008-08-13
DOP2006000261A (es) 2007-07-15
ECSP088477A (es) 2008-06-30
CR10014A (es) 2008-07-29
TW200804317A (en) 2008-01-16
NO20082919L (no) 2008-08-27
WO2007062193A1 (en) 2007-05-31
KR20080073721A (ko) 2008-08-11
SV2009002917A (es) 2009-02-19
AR058199A1 (es) 2008-01-23

Similar Documents

Publication Publication Date Title
HUS2000022I1 (hu) Tiglien-3-on származékok
HK1129305A1 (zh) 取代的 -氨基-吡咯並三嗪衍生物
GB0505941D0 (en) Human-to-mobile interfaces
EP1905769A4 (en) BENZIMIDAZOLE DERIVATIVE WITH HETEROCYCLE SUBSTITUTION
IL192092A0 (en) Aryl-isoxazolo-4-yl-oxadiazole derivatives
ZA200707358B (en) 1-benzylindole-2-carboxamide derivatives
PL1954674T3 (pl) Nowe pochodne N-fenetylokarboksyamidu
IL191586A0 (en) Heterocycle-substituted 3-alkyl azetidine derivatives
EP1871741A4 (en) SUBSTITUTED AZETIDINONE
ZA200802421B (en) 1-Acyldihydropyrazol derivatives
ZA200802088B (en) 4-Phenyl-6-substitued-pyrimidine-2-carbonitrile derivatives
HK1128022A1 (en) Triazole derivatives
ZA200804257B (en) Azaindole-2-carboxamide derivatives
IL184841A0 (en) Substituted aminoalkyl-and amidoalkyl-benzopyran derivatives
ZA200805353B (en) Aryl-isoxazol-4-yl-imidazole derivatives
IL184559A0 (en) Imidazole derivatives
IL191138A0 (en) Pyrazoloisoquinoline derivatives
EP1870412A4 (en) 2-THIOETHENYLCARBAPENEM DERIVATIVE
GB0511410D0 (en) Benzotrizepinone derivatives
AU2005100526A4 (en) Windows Hydrogenerator
ZA200706577B (en) Dihydroimidazothiazole derivatives
GB2424924B (en) Hinges
AU2005902628A0 (en) Auger
AU2005902963A0 (en) Auger
AU2005907278A0 (en) Tiglien-3-one derivatives