IL151496A0 - Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same - Google Patents

Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same

Info

Publication number
IL151496A0
IL151496A0 IL15149600A IL15149600A IL151496A0 IL 151496 A0 IL151496 A0 IL 151496A0 IL 15149600 A IL15149600 A IL 15149600A IL 15149600 A IL15149600 A IL 15149600A IL 151496 A0 IL151496 A0 IL 151496A0
Authority
IL
Israel
Prior art keywords
clarithromycin
processes
pharmaceutical composition
same
free
Prior art date
Application number
IL15149600A
Other languages
English (en)
Original Assignee
Teva Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Pharma filed Critical Teva Pharma
Publication of IL151496A0 publication Critical patent/IL151496A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C07F7/1872—Preparation; Treatments not provided for in C07F7/20
    • C07F7/1892—Preparation; Treatments not provided for in C07F7/20 by reactions not provided for in C07F7/1876 - C07F7/1888

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL15149600A 2000-02-29 2000-12-15 Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same IL151496A0 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US18588800P 2000-02-29 2000-02-29
US18912000P 2000-03-14 2000-03-14
US21323900P 2000-06-22 2000-06-22
PCT/US2000/033843 WO2001064224A1 (en) 2000-02-29 2000-12-15 Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same

Publications (1)

Publication Number Publication Date
IL151496A0 true IL151496A0 (en) 2003-04-10

Family

ID=27392028

Family Applications (1)

Application Number Title Priority Date Filing Date
IL15149600A IL151496A0 (en) 2000-02-29 2000-12-15 Processes for preparing clarithromycin and clarithromycin intermediate, essentially oxime-free clarithromycin, and pharmaceutical composition comprising the same

Country Status (15)

Country Link
US (3) US6617436B2 (sh)
EP (1) EP1313486A1 (sh)
JP (1) JP2004509062A (sh)
KR (1) KR20030047873A (sh)
AU (2) AU2578701A (sh)
CA (1) CA2401571A1 (sh)
CZ (1) CZ20023167A3 (sh)
HR (1) HRP20020709A2 (sh)
HU (1) HUP0302466A2 (sh)
IL (1) IL151496A0 (sh)
IS (1) IS6531A (sh)
PL (1) PL366021A1 (sh)
SK (1) SK13722002A3 (sh)
WO (1) WO2001064224A1 (sh)
YU (1) YU64202A (sh)

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CN102417532A (zh) * 2011-12-20 2012-04-18 浙江国邦药业有限公司 一种泰利霉素关键中间体5-德胺糖基-6-o-甲基红霉素的合成方法
CN102718821B (zh) * 2012-06-27 2014-12-03 浙江国邦药业有限公司 一种克拉霉素合成过程中甲基化反应以及甲基化试剂的回收套用方法
CN103880901A (zh) * 2012-12-23 2014-06-25 菏泽市方明制药有限公司 一种克拉霉素中间甲化物的制备方法
CN106905204B (zh) * 2017-02-24 2018-07-20 杭州新桂实业有限公司 一种克拉霉素合成过程中甲基化反应溶剂的回收套用方法
CN108117573A (zh) * 2017-12-26 2018-06-05 宁夏启元药业有限公司 4"-o-（三甲基硅）红霉素a 9-o-（1-乙氧基-1-甲基乙基）肟的合成方法

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Also Published As

Publication number Publication date
KR20030047873A (ko) 2003-06-18
EP1313486A1 (en) 2003-05-28
YU64202A (sh) 2005-03-15
SK13722002A3 (sk) 2003-08-05
PL366021A1 (en) 2005-01-24
US20060205683A1 (en) 2006-09-14
US6617436B2 (en) 2003-09-09
CZ20023167A3 (cs) 2003-10-15
AU2001225787C1 (en) 2006-09-21
CA2401571A1 (en) 2001-09-07
WO2001064224A1 (en) 2001-09-07
IS6531A (is) 2002-08-28
US7101858B2 (en) 2006-09-05
AU2578701A (en) 2001-09-12
US20010037015A1 (en) 2001-11-01
JP2004509062A (ja) 2004-03-25
US20030216556A1 (en) 2003-11-20
HRP20020709A2 (en) 2004-12-31
HUP0302466A2 (hu) 2003-11-28
AU2001225787B2 (en) 2005-12-08

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