IL140039A0 - Ureas and carbamates of n-heterocyclic carboxylic acids and carboxylic acid isosteres - Google Patents
Ureas and carbamates of n-heterocyclic carboxylic acids and carboxylic acid isosteresInfo
- Publication number
- IL140039A0 IL140039A0 IL14003998A IL14003998A IL140039A0 IL 140039 A0 IL140039 A0 IL 140039A0 IL 14003998 A IL14003998 A IL 14003998A IL 14003998 A IL14003998 A IL 14003998A IL 140039 A0 IL140039 A0 IL 140039A0
- Authority
- IL
- Israel
- Prior art keywords
- ureas
- carbamates
- carboxylic acid
- acid isosteres
- heterocyclic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/401—Proline; Derivatives thereof, e.g. captopril
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
- A61K8/4913—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
- A61K8/4946—Imidazoles or their condensed derivatives, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
- A61K8/496—Triazoles or their condensed derivatives, e.g. benzotriazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q7/00—Preparations for affecting hair growth
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Epidemiology (AREA)
- Birds (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Dermatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8784498P | 1998-06-03 | 1998-06-03 | |
PCT/US1998/025570 WO1999062879A1 (en) | 1998-06-03 | 1998-12-03 | Ureas and carbamates of n-heterocyclic carboxylic acids and carboxylic acid isosteres |
Publications (1)
Publication Number | Publication Date |
---|---|
IL140039A0 true IL140039A0 (en) | 2002-02-10 |
Family
ID=22207585
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL14003998A IL140039A0 (en) | 1998-06-03 | 1998-12-03 | Ureas and carbamates of n-heterocyclic carboxylic acids and carboxylic acid isosteres |
Country Status (17)
Country | Link |
---|---|
US (2) | US20020007075A1 (xx) |
EP (1) | EP1082301A1 (xx) |
JP (1) | JP2002516903A (xx) |
KR (1) | KR20010052502A (xx) |
CN (1) | CN1299346A (xx) |
AU (1) | AU1620499A (xx) |
BG (1) | BG105014A (xx) |
BR (1) | BR9815881A (xx) |
CA (1) | CA2333960A1 (xx) |
EA (1) | EA200001246A1 (xx) |
HU (1) | HUP0102847A2 (xx) |
IL (1) | IL140039A0 (xx) |
NO (1) | NO20006111L (xx) |
PL (1) | PL348671A1 (xx) |
SK (1) | SK18292000A3 (xx) |
WO (1) | WO1999062879A1 (xx) |
ZA (1) | ZA9811061B (xx) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2000302757A (ja) * | 1999-04-16 | 2000-10-31 | Shiseido Co Ltd | N−置換ピペリジン誘導体 |
CN1382140A (zh) | 1999-07-09 | 2002-11-27 | 奥索-麦克尼尔药品公司 | 具有神经营养活性的吡咯烷和哌啶、以及含有它们的相关组合物 |
EE200300168A (et) | 2000-10-30 | 2003-06-16 | Janssen Pharmaceutica N.V. | Tripeptidüülpeptidaasi inhibiitorid, nende valmistamine ja kasutamine ravimina ning neid sisaldav farmatseutiline kompositsioon |
ES2647664T3 (es) | 2011-01-04 | 2017-12-26 | Novartis Ag | Compuestos de indol o análogos de los mismos útiles para el tratamiento de la degeneración macular relacionada con la edad (AMD) |
JP6209605B2 (ja) | 2012-06-28 | 2017-10-04 | ノバルティス アーゲー | ピロリジン誘導体、および補体経路調節因子としてのその使用 |
ES2712190T3 (es) | 2012-06-28 | 2019-05-09 | Novartis Ag | Moduladores de la vía del complemento y sus usos |
US9468661B2 (en) | 2012-06-28 | 2016-10-18 | Novartis Ag | Pyrrolidine derivatives and their use as complement pathway modulators |
JP6273274B2 (ja) | 2012-06-28 | 2018-01-31 | ノバルティス アーゲー | 補体経路モジュレーターおよびその使用 |
JP6154897B2 (ja) | 2012-06-28 | 2017-06-28 | ノバルティス アーゲー | ピロリジン誘導体、および補体経路調節因子としてのその使用 |
KR20150036481A (ko) | 2012-07-12 | 2015-04-07 | 노파르티스 아게 | 보체 경로 조절제 및 그의 용도 |
WO2023090853A1 (ko) * | 2021-11-19 | 2023-05-25 | 고려대학교 세종산학협력단 | 신규 우레아계 또는 카바메이트계 p2x7 수용체 길항제 및 이를 유효성분으로 포함하는 주요 우울 장애의 예방 또는 치료용 약학 조성물 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS55151555A (en) * | 1979-05-14 | 1980-11-26 | Tanabe Seiyaku Co Ltd | Proline derivatives and their production |
US4402969A (en) * | 1981-03-23 | 1983-09-06 | Merck & Co., Inc. | Antihypertensive proline derivatives |
DE3134933A1 (de) * | 1981-09-03 | 1983-03-31 | Hoechst Ag, 6230 Frankfurt | "harnstoffderivate, verfahren zu ihrer herstellung und diese enthaltende medikamente sowie deren verwendung" |
JPS58170752A (ja) * | 1982-03-30 | 1983-10-07 | Kureha Chem Ind Co Ltd | N−カルバモイルアミノ酸誘導体 |
DE4228455A1 (de) * | 1992-08-26 | 1994-09-15 | Beiersdorf Ag | Kosmetische und dermatologische Lichtschutzformulierungen mit einem Gehalt an Thiolen und/oder Thiolderivaten |
US5411991A (en) * | 1992-12-22 | 1995-05-02 | Shander; Douglas | Method of reducing hair growth employing sulfhydryl active compounds |
US5264619B1 (en) * | 1993-01-15 | 1996-05-14 | Cosmos Pharm Corp | Anti-androgenic cyclo and bicyclo alkenes |
US5744485A (en) * | 1994-03-25 | 1998-04-28 | Vertex Pharmaceuticals Incorporated | Carbamates and ureas as modifiers of multi-drug resistance |
US5780484A (en) * | 1996-11-13 | 1998-07-14 | Vertex Pharmaceuticals Incorporated | Methods for stimulating neurite growth with piperidine compounds |
US5935989A (en) * | 1996-12-31 | 1999-08-10 | Gpi Nil Holdings Inc. | N-linked ureas and carbamates of heterocyclic thioesters |
-
1998
- 1998-12-03 EA EA200001246A patent/EA200001246A1/ru unknown
- 1998-12-03 PL PL98348671A patent/PL348671A1/xx unknown
- 1998-12-03 SK SK1829-2000A patent/SK18292000A3/sk unknown
- 1998-12-03 JP JP2000552091A patent/JP2002516903A/ja active Pending
- 1998-12-03 ZA ZA9811061A patent/ZA9811061B/xx unknown
- 1998-12-03 KR KR1020007013636A patent/KR20010052502A/ko not_active Application Discontinuation
- 1998-12-03 CA CA002333960A patent/CA2333960A1/en not_active Abandoned
- 1998-12-03 HU HU0102847A patent/HUP0102847A2/hu unknown
- 1998-12-03 AU AU16204/99A patent/AU1620499A/en not_active Abandoned
- 1998-12-03 CN CN98814098A patent/CN1299346A/zh active Pending
- 1998-12-03 WO PCT/US1998/025570 patent/WO1999062879A1/en not_active Application Discontinuation
- 1998-12-03 IL IL14003998A patent/IL140039A0/xx unknown
- 1998-12-03 EP EP98960656A patent/EP1082301A1/en not_active Withdrawn
- 1998-12-03 BR BR9815881-3A patent/BR9815881A/pt not_active Application Discontinuation
-
2000
- 2000-12-01 NO NO20006111A patent/NO20006111L/no not_active Application Discontinuation
- 2000-12-01 BG BG105014A patent/BG105014A/xx unknown
-
2001
- 2001-01-30 US US09/771,686 patent/US20020007075A1/en not_active Abandoned
- 2001-05-03 US US09/847,432 patent/US20020042442A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
PL348671A1 (en) | 2002-06-03 |
WO1999062879A1 (en) | 1999-12-09 |
BG105014A (en) | 2001-08-31 |
NO20006111D0 (no) | 2000-12-01 |
ZA9811061B (en) | 1999-12-03 |
US20020007075A1 (en) | 2002-01-17 |
JP2002516903A (ja) | 2002-06-11 |
CA2333960A1 (en) | 1999-12-09 |
AU1620499A (en) | 1999-12-20 |
EA200001246A1 (ru) | 2001-08-27 |
BR9815881A (pt) | 2002-07-23 |
KR20010052502A (ko) | 2001-06-25 |
HUP0102847A2 (hu) | 2001-12-28 |
WO1999062879A8 (en) | 2000-05-04 |
NO20006111L (no) | 2001-02-01 |
US20020042442A1 (en) | 2002-04-11 |
SK18292000A3 (sk) | 2001-07-10 |
CN1299346A (zh) | 2001-06-13 |
EP1082301A1 (en) | 2001-03-14 |
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