IL140020A - Dosage form to achieve a plasma concentration profile increases after administration for a long period of time - Google Patents
Dosage form to achieve a plasma concentration profile increases after administration for a long period of timeInfo
- Publication number
- IL140020A IL140020A IL140020A IL14002000A IL140020A IL 140020 A IL140020 A IL 140020A IL 140020 A IL140020 A IL 140020A IL 14002000 A IL14002000 A IL 14002000A IL 140020 A IL140020 A IL 140020A
- Authority
- IL
- Israel
- Prior art keywords
- drug
- dosage form
- layer
- release
- form according
- Prior art date
Links
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- 229940044519 poloxamer 188 Drugs 0.000 description 1
- 229910000160 potassium phosphate Inorganic materials 0.000 description 1
- 235000011009 potassium phosphates Nutrition 0.000 description 1
- 102000004196 processed proteins & peptides Human genes 0.000 description 1
- 108090000765 processed proteins & peptides Proteins 0.000 description 1
- 238000012545 processing Methods 0.000 description 1
- 150000003180 prostaglandins Chemical class 0.000 description 1
- 235000018102 proteins Nutrition 0.000 description 1
- 108090000623 proteins and genes Proteins 0.000 description 1
- 102000004169 proteins and genes Human genes 0.000 description 1
- 238000012552 review Methods 0.000 description 1
- 229940125723 sedative agent Drugs 0.000 description 1
- 239000000932 sedative agent Substances 0.000 description 1
- 239000001488 sodium phosphate Substances 0.000 description 1
- 229910000162 sodium phosphate Inorganic materials 0.000 description 1
- 235000011008 sodium phosphates Nutrition 0.000 description 1
- 239000000126 substance Substances 0.000 description 1
- 230000009747 swallowing Effects 0.000 description 1
- 230000008961 swelling Effects 0.000 description 1
- 230000001975 sympathomimetic effect Effects 0.000 description 1
- 229940064707 sympathomimetics Drugs 0.000 description 1
- 239000011975 tartaric acid Substances 0.000 description 1
- 235000002906 tartaric acid Nutrition 0.000 description 1
- 238000012360 testing method Methods 0.000 description 1
- 239000003204 tranquilizing agent Substances 0.000 description 1
- 230000002936 tranquilizing effect Effects 0.000 description 1
- VZCYOOQTPOCHFL-UHFFFAOYSA-N trans-butenedioic acid Natural products OC(=O)C=CC(O)=O VZCYOOQTPOCHFL-UHFFFAOYSA-N 0.000 description 1
- 230000007723 transport mechanism Effects 0.000 description 1
- RYFMWSXOAZQYPI-UHFFFAOYSA-K trisodium phosphate Chemical compound [Na+].[Na+].[Na+].[O-]P([O-])([O-])=O RYFMWSXOAZQYPI-UHFFFAOYSA-K 0.000 description 1
- 229940124549 vasodilator Drugs 0.000 description 1
- 239000003071 vasodilator agent Substances 0.000 description 1
- 239000001993 wax Substances 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N21/00—Investigating or analysing materials by the use of optical means, i.e. using sub-millimetre waves, infrared, visible or ultraviolet light
- G01N21/84—Systems specially adapted for particular applications
- G01N21/88—Investigating the presence of flaws or contamination
- G01N21/95—Investigating the presence of flaws or contamination characterised by the material or shape of the object to be examined
- G01N21/9508—Capsules; Tablets
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Biochemistry (AREA)
- Physics & Mathematics (AREA)
- Pathology (AREA)
- Immunology (AREA)
- General Physics & Mathematics (AREA)
- Analytical Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8778798P | 1998-06-03 | 1998-06-03 | |
| US09/253,317 US6919373B1 (en) | 1996-11-12 | 1999-02-19 | Methods and devices for providing prolonged drug therapy |
| PCT/US1999/011920 WO1999062496A1 (en) | 1998-06-03 | 1999-05-27 | Methods and devices for providing prolonged drug therapy |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL140020A true IL140020A (en) | 2012-10-31 |
Family
ID=27733446
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL140020A IL140020A (en) | 1998-06-03 | 2000-11-30 | Dosage form to achieve a plasma concentration profile increases after administration for a long period of time |
| IL211081A IL211081A0 (en) | 1998-06-03 | 2011-02-06 | Methods and devices for providing prolonged drug therapy |
| IL222437A IL222437A (en) | 1998-06-03 | 2012-10-15 | Multi-layer and osmotic dosage form |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL211081A IL211081A0 (en) | 1998-06-03 | 2011-02-06 | Methods and devices for providing prolonged drug therapy |
| IL222437A IL222437A (en) | 1998-06-03 | 2012-10-15 | Multi-layer and osmotic dosage form |
Country Status (6)
| Country | Link |
|---|---|
| US (3) | US7521067B1 (enExample) |
| JP (2) | JP2012082195A (enExample) |
| KR (1) | KR100827254B1 (enExample) |
| IL (3) | IL140020A (enExample) |
| NO (2) | NO333360B1 (enExample) |
| ZA (1) | ZA200007111B (enExample) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100827254B1 (ko) | 1998-06-03 | 2008-05-07 | 알자 코포레이션 | 연장된 약물 치료를 제공하기 위한 방법 및 장치 |
| US20050232995A1 (en) | 2002-07-29 | 2005-10-20 | Yam Nyomi V | Methods and dosage forms for controlled delivery of paliperidone and risperidone |
| WO2019173384A1 (en) | 2018-03-05 | 2019-09-12 | Kashiv Pharma Llc | Programmable pharmaceutical compositions for chrono drug release |
| JP7332093B2 (ja) * | 2018-04-16 | 2023-08-23 | エスアンドアール ファーマチェウティチ エス．ピー．エー． | 女性の生殖能力の改善のための異なる薬物動態プロファイルを有するレスベラトロルの混合物に基づく製剤の使用 |
| CA3065695C (en) | 2018-06-27 | 2021-06-01 | Kashiv Biosciences, Llc | Self-regulating osmotic gastroretentive drug delivery systems |
| CN113891713A (zh) * | 2019-01-25 | 2022-01-04 | 艾伦索尔医药发展股份有限公司 | 用于治疗注意力缺陷多动障碍的哌甲酯组合物 |
| EP3934622A1 (en) | 2019-03-05 | 2022-01-12 | Amneal Complex Products Research LLC | Delayed release methylphenidate compositions |
| US20220241184A1 (en) * | 2019-06-21 | 2022-08-04 | Kashiv Biosciences, Llc | Gastroretentive dosage forms of levodopa and carbidopa |
| US11964048B2 (en) | 2020-12-18 | 2024-04-23 | Amneal Complex Products Research Llc | Sustained release compositions comprising liothyronine |
Family Cites Families (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB952006A (en) | 1962-02-21 | 1964-03-11 | John Holroyd & Company Ltd | Multi-layer tablet making machines |
| US3634584A (en) | 1969-02-13 | 1972-01-11 | American Home Prod | Sustained action dosage form |
| US4096238A (en) | 1974-12-23 | 1978-06-20 | Alza Corporation | Method for administering drug to the gastrointestinal tract |
| US4327725A (en) | 1980-11-25 | 1982-05-04 | Alza Corporation | Osmotic device with hydrogel driving member |
| US4591500A (en) | 1983-04-25 | 1986-05-27 | Microencapsulation S.A. | Tablet having the shape of a capsule, process and device for its preparation |
| US4612008A (en) | 1983-05-11 | 1986-09-16 | Alza Corporation | Osmotic device with dual thermodynamic activity |
| US4783337A (en) | 1983-05-11 | 1988-11-08 | Alza Corporation | Osmotic system comprising plurality of members for dispensing drug |
| US4765989A (en) | 1983-05-11 | 1988-08-23 | Alza Corporation | Osmotic device for administering certain drugs |
| US4847093A (en) | 1986-06-19 | 1989-07-11 | Alza Corporation | Dosage form with means for governing rate of gas formation |
| US5236689A (en) | 1987-06-25 | 1993-08-17 | Alza Corporation | Multi-unit delivery system |
| US5391381A (en) | 1987-06-25 | 1995-02-21 | Alza Corporation | Dispenser capable of delivering plurality of drug units |
| US4874388A (en) | 1987-06-25 | 1989-10-17 | Alza Corporation | Multi-layer delivery system |
| US4915953A (en) | 1987-09-03 | 1990-04-10 | Alza Corporation | Dosage form for delivering acetaminophen or phenylpropanolamine |
| JP2770243B2 (ja) | 1989-09-21 | 1998-06-25 | ライオンエンジニアリング株式会社 | 錠剤成分量検査方法およびその装置 |
| US5089270A (en) | 1990-05-15 | 1992-02-18 | L. Perrigo Company | Capsule-shaped tablet |
| US5213738A (en) | 1990-05-15 | 1993-05-25 | L. Perrigo Company | Method for making a capsule-shaped tablet |
| US5464631A (en) | 1990-06-27 | 1995-11-07 | Warner-Lambert Company | Encapsulated dosage forms |
| US5156850A (en) * | 1990-08-31 | 1992-10-20 | Alza Corporation | Dosage form for time-varying patterns of drug delivery |
| US5160744A (en) | 1991-06-27 | 1992-11-03 | Alza Corporation | Verapmil therapy |
| US5190765A (en) | 1991-06-27 | 1993-03-02 | Alza Corporation | Therapy delayed |
| US5294770A (en) | 1992-01-14 | 1994-03-15 | Alza Corporation | Laser tablet treatment system with dual access to tablet |
| US5248310A (en) * | 1992-03-27 | 1993-09-28 | Alza Corporation | Oral osmotic device with hydrogel driving member |
| US5422831A (en) | 1992-08-03 | 1995-06-06 | Iowa State University Research Foundation, Inc. | Acoustic and video imaging system for quality determination of pharmaceutical products |
| DE4417015A1 (de) | 1994-05-14 | 1995-11-16 | Maschimpex Gmbh | Sortierautomat zur Sortierung bzw. Klassifikation von Kleinprodukten der pharmazeutischen und der Süßwarenindustrie nach Form und Farbe |
| US5582838A (en) * | 1994-12-22 | 1996-12-10 | Merck & Co., Inc. | Controlled release drug suspension delivery device |
| US5558879A (en) * | 1995-04-28 | 1996-09-24 | Andrx Pharmaceuticals, Inc. | Controlled release formulation for water soluble drugs in which a passageway is formed in situ |
| ZA97976B (en) * | 1996-04-05 | 1997-08-18 | Alza Corp | Uniform drug delivery theraphy. |
| WO1998006380A2 (en) * | 1996-08-16 | 1998-02-19 | Alza Corporation | Dosage form for providing ascending dose of drug |
| US5824338A (en) | 1996-08-19 | 1998-10-20 | L. Perrigo Company | Caplet and gelatin covering therefor |
| ES2262174T3 (es) * | 1996-09-30 | 2006-11-16 | Alza Corporation | Forma de dosificacion y procedimiento de administracion de medicamentos. |
| EP0946151B1 (en) | 1996-11-25 | 2006-05-10 | Alza Corporation | Ascending-dose dosage form |
| ES2203963T3 (es) * | 1997-05-30 | 2004-04-16 | Osmotica Corp. | Dispositivo osmotico multicapa. |
| KR100827254B1 (ko) | 1998-06-03 | 2008-05-07 | 알자 코포레이션 | 연장된 약물 치료를 제공하기 위한 방법 및 장치 |
-
1999
- 1999-05-27 KR KR1020007013610A patent/KR100827254B1/ko not_active Expired - Lifetime
- 1999-06-02 US US09/324,343 patent/US7521067B1/en not_active Expired - Fee Related
-
2000
- 2000-11-30 IL IL140020A patent/IL140020A/en not_active IP Right Cessation
- 2000-12-01 ZA ZA200007111A patent/ZA200007111B/xx unknown
-
2009
- 2009-03-11 US US12/402,075 patent/US8323691B2/en not_active Expired - Fee Related
-
2010
- 2010-07-27 NO NO20101070A patent/NO333360B1/no not_active IP Right Cessation
-
2011
- 2011-02-06 IL IL211081A patent/IL211081A0/en unknown
- 2011-10-06 JP JP2011222079A patent/JP2012082195A/ja not_active Withdrawn
-
2012
- 2012-10-15 IL IL222437A patent/IL222437A/en not_active IP Right Cessation
- 2012-10-18 US US13/654,958 patent/US8936810B2/en not_active Expired - Fee Related
-
2013
- 2013-03-06 NO NO20130342A patent/NO334409B1/no not_active IP Right Cessation
-
2014
- 2014-11-14 JP JP2014232011A patent/JP2015028095A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| KR100827254B1 (ko) | 2008-05-07 |
| US8936810B2 (en) | 2015-01-20 |
| IL211081A0 (en) | 2011-04-28 |
| NO333360B1 (no) | 2013-05-13 |
| ZA200007111B (en) | 2001-06-05 |
| US20130043612A1 (en) | 2013-02-21 |
| NO20101070L (no) | 2001-02-05 |
| IL222437A (en) | 2015-10-29 |
| US8323691B2 (en) | 2012-12-04 |
| NO334409B1 (no) | 2014-02-24 |
| US20090186085A1 (en) | 2009-07-23 |
| US7521067B1 (en) | 2009-04-21 |
| NO20130342L (no) | 2001-02-05 |
| JP2015028095A (ja) | 2015-02-12 |
| KR20010043980A (ko) | 2001-05-25 |
| JP2012082195A (ja) | 2012-04-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| EXP | Patent expired |