IL117289A - Spectinomycin boron derivatives and stable high potency aqueous pharmaceutical compositions containing them - Google Patents
Spectinomycin boron derivatives and stable high potency aqueous pharmaceutical compositions containing themInfo
- Publication number
- IL117289A IL117289A IL11728996A IL11728996A IL117289A IL 117289 A IL117289 A IL 117289A IL 11728996 A IL11728996 A IL 11728996A IL 11728996 A IL11728996 A IL 11728996A IL 117289 A IL117289 A IL 117289A
- Authority
- IL
- Israel
- Prior art keywords
- spectinomycin
- pharmaceutical compositions
- compositions containing
- aqueous pharmaceutical
- stable high
- Prior art date
Links
- 229960000268 spectinomycin Drugs 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- -1 Spectinomycin boron derivatives Chemical class 0.000 title 1
- HEMHJVSKTPXQMS-UHFFFAOYSA-M Sodium hydroxide Chemical compound [OH-].[Na+] HEMHJVSKTPXQMS-UHFFFAOYSA-M 0.000 abstract 3
- UNFWWIHTNXNPBV-WXKVUWSESA-N spectinomycin Chemical compound O([C@@H]1[C@@H](NC)[C@@H](O)[C@H]([C@@H]([C@H]1O1)O)NC)[C@]2(O)[C@H]1O[C@H](C)CC2=O UNFWWIHTNXNPBV-WXKVUWSESA-N 0.000 abstract 2
- KGBXLFKZBHKPEV-UHFFFAOYSA-N boric acid Chemical compound OB(O)O KGBXLFKZBHKPEV-UHFFFAOYSA-N 0.000 abstract 1
- 239000004327 boric acid Substances 0.000 abstract 1
- 150000001639 boron compounds Chemical class 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000002576 ketones Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/396,629 US5556879A (en) | 1995-03-01 | 1995-03-01 | Aqueous spectinomycin borate solutions |
Publications (2)
Publication Number | Publication Date |
---|---|
IL117289A0 IL117289A0 (en) | 1996-06-18 |
IL117289A true IL117289A (en) | 1999-07-14 |
Family
ID=23568013
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL11728996A IL117289A (en) | 1995-03-01 | 1996-02-28 | Spectinomycin boron derivatives and stable high potency aqueous pharmaceutical compositions containing them |
Country Status (9)
Country | Link |
---|---|
US (1) | US5556879A (xx) |
EP (1) | EP0812324B1 (xx) |
AT (1) | ATE192749T1 (xx) |
AU (1) | AU4943196A (xx) |
DE (1) | DE69608260T2 (xx) |
ES (1) | ES2147369T3 (xx) |
IL (1) | IL117289A (xx) |
NZ (1) | NZ303194A (xx) |
WO (1) | WO1996026945A1 (xx) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6184244B1 (en) | 1996-12-16 | 2001-02-06 | Idun Pharmaceuticals, Inc. | C-terminal modified (N-substituted)-2-indolyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases |
EP2461805B1 (en) * | 2009-07-24 | 2017-11-01 | University of Tennessee Research Foundation | Spectinamides as anti-tuberculosis agents |
WO2014085599A1 (en) | 2012-11-30 | 2014-06-05 | Acura Pharmaceuticals, Inc. | Self-regulated release of active pharmaceutical ingredient |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3234092A (en) * | 1959-10-20 | 1966-02-08 | Upjohn Co | Actinospectacin and process for producing same |
-
1995
- 1995-03-01 US US08/396,629 patent/US5556879A/en not_active Expired - Lifetime
-
1996
- 1996-02-27 AU AU49431/96A patent/AU4943196A/en not_active Abandoned
- 1996-02-27 EP EP96905820A patent/EP0812324B1/en not_active Expired - Lifetime
- 1996-02-27 AT AT96905820T patent/ATE192749T1/de not_active IP Right Cessation
- 1996-02-27 WO PCT/EP1996/000816 patent/WO1996026945A1/en active IP Right Grant
- 1996-02-27 ES ES96905820T patent/ES2147369T3/es not_active Expired - Lifetime
- 1996-02-27 DE DE69608260T patent/DE69608260T2/de not_active Expired - Lifetime
- 1996-02-27 NZ NZ303194A patent/NZ303194A/en not_active IP Right Cessation
- 1996-02-28 IL IL11728996A patent/IL117289A/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
IL117289A0 (en) | 1996-06-18 |
ATE192749T1 (de) | 2000-05-15 |
EP0812324B1 (en) | 2000-05-10 |
WO1996026945A1 (en) | 1996-09-06 |
AU4943196A (en) | 1996-09-18 |
DE69608260T2 (de) | 2001-04-26 |
ES2147369T3 (es) | 2000-09-01 |
DE69608260D1 (en) | 2000-06-15 |
NZ303194A (en) | 1999-04-29 |
US5556879A (en) | 1996-09-17 |
EP0812324A1 (en) | 1997-12-17 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FF | Patent granted | ||
FF | Patent granted | ||
MM9K | Patent not in force due to non-payment of renewal fees |