IL100642A - Process for the preparation of (2-) diethylamino (rifmacin P) AED / P (and its new intermediate - Google Patents

Process for the preparation of (2-) diethylamino (rifmacin P) AED / P (and its new intermediate

Info

Publication number
IL100642A
IL100642A IL10064292A IL10064292A IL100642A IL 100642 A IL100642 A IL 100642A IL 10064292 A IL10064292 A IL 10064292A IL 10064292 A IL10064292 A IL 10064292A IL 100642 A IL100642 A IL 100642A
Authority
IL
Israel
Prior art keywords
dea
iii
process according
bromorifamycin
quinonimine
Prior art date
Application number
IL10064292A
Other languages
English (en)
Hebrew (he)
Other versions
IL100642A0 (en
Inventor
Gianbattista Panzone
Anacleto Gianantonio
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of IL100642A0 publication Critical patent/IL100642A0/xx
Publication of IL100642A publication Critical patent/IL100642A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Virology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL10064292A 1991-01-28 1992-01-13 Process for the preparation of (2-) diethylamino (rifmacin P) AED / P (and its new intermediate IL100642A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP91101037 1991-01-28

Publications (2)

Publication Number Publication Date
IL100642A0 IL100642A0 (en) 1992-09-06
IL100642A true IL100642A (en) 1995-11-27

Family

ID=8206332

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10064292A IL100642A (en) 1991-01-28 1992-01-13 Process for the preparation of (2-) diethylamino (rifmacin P) AED / P (and its new intermediate

Country Status (14)

Country Link
US (1) US5378837A (de)
EP (1) EP0497125B1 (de)
JP (1) JP3154783B2 (de)
KR (1) KR920014819A (de)
AT (1) ATE174336T1 (de)
CA (1) CA2059999C (de)
DE (1) DE69227790T2 (de)
DK (1) DK0497125T3 (de)
ES (1) ES2124708T3 (de)
GR (1) GR3029624T3 (de)
HU (1) HU208697B (de)
IE (1) IE920235A1 (de)
IL (1) IL100642A (de)
ZA (1) ZA92537B (de)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1470426A (en) * 1974-08-30 1977-04-14 Lepetit Spa Rifamycins
IT1053787B (it) * 1974-10-29 1981-10-10 Pastori A Macrolidi azotati e loro preparazione
GB1523199A (en) * 1976-05-28 1978-08-31 Lepetit Spa Rifamycin sv derivatives
GB1523198A (en) * 1976-05-28 1978-08-31 Lepetit Spa Thiazolo-rifamycin derivatives
CH629212A5 (it) * 1976-10-18 1982-04-15 Erba Farmitalia Procedimento per la preparazione di composti di rifamicina.
IT1090759B (it) * 1977-11-29 1985-06-26 Alfa Farmaceutici Spa Procedimento per la preparazione di 3 iodio e 3 bromo rifamicina s
GB8531887D0 (en) * 1985-12-30 1986-02-05 Lepetit Spa Rifamycin sv derivatives

Also Published As

Publication number Publication date
ATE174336T1 (de) 1998-12-15
GR3029624T3 (en) 1999-06-30
DE69227790T2 (de) 1999-06-10
CA2059999A1 (en) 1992-07-29
AU1033092A (en) 1992-07-30
EP0497125B1 (de) 1998-12-09
CA2059999C (en) 2001-09-25
IE920235A1 (en) 1992-07-29
KR920014819A (ko) 1992-08-25
HUT61315A (en) 1992-12-28
DK0497125T3 (da) 1999-08-16
AU650509B2 (en) 1994-06-23
JPH04346990A (ja) 1992-12-02
DE69227790D1 (de) 1999-01-21
IL100642A0 (en) 1992-09-06
JP3154783B2 (ja) 2001-04-09
ES2124708T3 (es) 1999-02-16
ZA92537B (en) 1992-12-30
HU208697B (en) 1993-12-28
EP0497125A1 (de) 1992-08-05
US5378837A (en) 1995-01-03
HU9200255D0 (en) 1992-05-28

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