IE44316B1 - Indazole derivatives - Google Patents

Indazole derivatives

Info

Publication number
IE44316B1
IE44316B1 IE2637/76A IE263776A IE44316B1 IE 44316 B1 IE44316 B1 IE 44316B1 IE 2637/76 A IE2637/76 A IE 2637/76A IE 263776 A IE263776 A IE 263776A IE 44316 B1 IE44316 B1 IE 44316B1
Authority
IE
Ireland
Prior art keywords
compound
chg
group
formula
hydrogen
Prior art date
Application number
IE2637/76A
Other languages
English (en)
Other versions
IE44316L (en
Original Assignee
Sandoz Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH1571675A external-priority patent/CH605934A5/de
Priority claimed from CH1664575A external-priority patent/CH605858A5/de
Application filed by Sandoz Ltd filed Critical Sandoz Ltd
Publication of IE44316L publication Critical patent/IE44316L/xx
Publication of IE44316B1 publication Critical patent/IE44316B1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IE2637/76A 1975-12-03 1976-12-01 Indazole derivatives IE44316B1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH1571675A CH605934A5 (en) 1975-12-03 1975-12-03 Myotonolytic oxazolinyl- and thiazolinyl-amino-indazole derivs.
CH1664575A CH605858A5 (en) 1975-12-22 1975-12-22 Myotonolytic oxazolinyl- and thiazolinyl-amino-indazole derivs.
CH927976 1976-07-20
CH931276 1976-07-21

Publications (2)

Publication Number Publication Date
IE44316L IE44316L (en) 1977-06-03
IE44316B1 true IE44316B1 (en) 1981-10-21

Family

ID=27429211

Family Applications (1)

Application Number Title Priority Date Filing Date
IE2637/76A IE44316B1 (en) 1975-12-03 1976-12-01 Indazole derivatives

Country Status (20)

Country Link
US (1) US4086353A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JPS5268177A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU510820B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BE (1) BE848962A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA1082714A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE2653005A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK528976A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES453861A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI763385A7 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2333504A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB1564327A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IE (1) IE44316B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL51028A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (1) NL7613317A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (1) NO764039L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NZ (1) NZ182779A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PH (1) PH12642A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PT (1) PT65918B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SE (1) SE424553B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
YU (1) YU293876A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1982000824A1 (en) * 1980-09-05 1982-03-18 Geissmann F 1h and 2h indazol derivatives and medicaments containing them
IL160744A0 (en) * 2001-09-26 2004-08-31 Pharmacia Italia Spa Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
SE0402763D0 (sv) * 2004-11-11 2004-11-11 Astrazeneca Ab Nitro indazole derivatives
SE0402762D0 (sv) * 2004-11-11 2004-11-11 Astrazeneca Ab Indazole sulphonamide derivatives
ATE507224T1 (de) * 2005-11-15 2011-05-15 Array Biopharma Inc Verfahren und zwischenverbindungen zur herstellung von n4-phenyl-quinazolin-4-amin derivaten
EP1966152A2 (en) * 2005-12-20 2008-09-10 Takeda Pharmaceutical Company Limited Glucokinase activators
RU2477282C2 (ru) * 2007-08-17 2013-03-10 Эл Джи Лайф Сайенсиз Лтд. Соединения индола в качестве ингибиторов клеточного некроза
US20100291533A1 (en) * 2008-01-04 2010-11-18 Soon Ha Kim Indole and indazole derivatives having a cell-, tissue- and organ-preserving effect
KR101404151B1 (ko) * 2011-11-25 2014-06-05 가톨릭대학교 산학협력단 안과 질환의 예방 및 치료용 약학 조성물
WO2016115272A1 (en) 2015-01-13 2016-07-21 Vanderbilt University Benzothiazole and benzisothiazole-substituted compounds as mglur4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
US9980945B2 (en) 2015-01-13 2018-05-29 Vanderbilt University Benzoisoxazole-substituted compounds as MGLUR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
US10526323B2 (en) 2015-01-30 2020-01-07 Vanderbilt University Indazole and azaindazole substituted compounds as mGluR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3759903A (en) * 1971-07-28 1973-09-18 Squibb & Sons Inc Thiazolinyl and thiazinyl derivatives of indazoles

Also Published As

Publication number Publication date
JPS5268177A (en) 1977-06-06
IL51028A (en) 1980-06-30
GB1564327A (en) 1980-04-10
PT65918B (fr) 1978-07-05
AU510820B2 (en) 1980-07-17
NL7613317A (nl) 1977-06-07
YU293876A (en) 1982-05-31
DE2653005A1 (de) 1977-06-08
PH12642A (en) 1979-07-11
AU2025276A (en) 1978-06-08
PT65918A (fr) 1977-01-01
CA1082714A (en) 1980-07-29
NO764039L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1977-06-06
BE848962A (fr) 1977-06-01
SE7613195L (sv) 1977-06-04
FR2333504B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1980-08-29
ES453861A1 (es) 1978-03-01
SE424553B (sv) 1982-07-26
IE44316L (en) 1977-06-03
IL51028A0 (en) 1977-02-28
DK528976A (da) 1977-06-04
FR2333504A1 (fr) 1977-07-01
NZ182779A (en) 1979-08-31
FI763385A7 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1977-06-04
US4086353A (en) 1978-04-25

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