ID27127A - SENYAWA-SENYAWA TRIAZOLO (4,5-d) PIRIMIDINA YANG BARU - Google Patents

SENYAWA-SENYAWA TRIAZOLO (4,5-d) PIRIMIDINA YANG BARU

Info

Publication number
ID27127A
ID27127A IDW20001348A ID20001348A ID27127A ID 27127 A ID27127 A ID 27127A ID W20001348 A IDW20001348 A ID W20001348A ID 20001348 A ID20001348 A ID 20001348A ID 27127 A ID27127 A ID 27127A
Authority
ID
Indonesia
Prior art keywords
new pyrimidine
triazolo compounds
triazolo
compounds
pyrimidine
Prior art date
Application number
IDW20001348A
Other languages
English (en)
Inventor
Brian Springthope
Paul Willis
Roger Brown
Garry Pairaudeau
Stephen Thom
Original Assignee
Astrazeneca Uk Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE9800458A external-priority patent/SE9800458D0/xx
Priority claimed from SE9803669A external-priority patent/SE9803669D0/xx
Application filed by Astrazeneca Uk Ltd filed Critical Astrazeneca Uk Ltd
Publication of ID27127A publication Critical patent/ID27127A/id

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
IDW20001348A 1998-02-17 1999-02-05 SENYAWA-SENYAWA TRIAZOLO (4,5-d) PIRIMIDINA YANG BARU ID27127A (id)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9800458A SE9800458D0 (sv) 1998-02-17 1998-02-17 Novel compounds
SE9803669A SE9803669D0 (sv) 1998-10-26 1998-10-26 Novel compounds

Publications (1)

Publication Number Publication Date
ID27127A true ID27127A (id) 2001-03-01

Family

ID=26663214

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW20001348A ID27127A (id) 1998-02-17 1999-02-05 SENYAWA-SENYAWA TRIAZOLO (4,5-d) PIRIMIDINA YANG BARU

Country Status (21)

Country Link
US (1) US6369064B1 (id)
EP (1) EP1056749B1 (id)
JP (1) JP2002503663A (id)
KR (1) KR20010078696A (id)
CN (1) CN1291193A (id)
AR (1) AR015515A1 (id)
AT (1) ATE232866T1 (id)
AU (1) AU2650099A (id)
BR (1) BR9907934A (id)
CA (1) CA2316264A1 (id)
DE (1) DE69905451T2 (id)
HU (1) HUP0100328A3 (id)
ID (1) ID27127A (id)
IL (1) IL137812A0 (id)
MX (1) MXPA00007634A (id)
NO (1) NO20004089L (id)
NZ (1) NZ505250A (id)
PL (1) PL342430A1 (id)
SK (1) SK12242000A3 (id)
TR (1) TR200002380T2 (id)
WO (1) WO1999041254A1 (id)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9702773D0 (sv) * 1997-07-22 1997-07-22 Astra Pharma Prod Novel compounds
SE9904129D0 (sv) 1999-11-15 1999-11-15 Astra Pharma Prod Novel compounds
GB0013488D0 (en) * 2000-06-02 2000-07-26 Astrazeneca Ab Chemical compound
TWI290549B (en) * 2000-06-02 2007-12-01 Astrazeneca Ab Process for the preparation of cyclopropyl carboxylic acid ester and derivatives
US7086397B2 (en) * 2002-02-16 2006-08-08 Graham Lindley Spruiell Patient usable emergency medical kit
GB0219746D0 (en) * 2002-08-23 2002-10-02 Inst Of Ex Botany Ascr Azapurine derivatives
US7335648B2 (en) 2003-10-21 2008-02-26 Inspire Pharmaceuticals, Inc. Non-nucleotide composition and method for inhibiting platelet aggregation
US7504497B2 (en) 2003-10-21 2009-03-17 Inspire Pharmaceuticals, Inc. Orally bioavailable compounds and methods for inhibiting platelet aggregation
US7749981B2 (en) 2003-10-21 2010-07-06 Inspire Pharmaceuticals, Inc. Drug-eluting stents coated with non-nucleotide P2Y12 receptor antagonist compound
WO2005040174A1 (en) 2003-10-21 2005-05-06 Inspire Pharmaceuticals, Inc. Tetrahydro-furo`3,4-d!dioxole compounds and compositions and method for inhibiting platelet aggregation
US7932376B2 (en) 2005-05-05 2011-04-26 Inspire Pharmaceuticals, Inc. Pyrimidine-based non-nucleotide composition and method for inhibiting platelet aggregation
JPWO2007020935A1 (ja) * 2005-08-17 2009-02-26 小野薬品工業株式会社 Ｐ２ｙ１２受容体および／またはｐ２ｙ１４受容体ブロッカーを含有してなる疼痛治療剤
JP2010508350A (ja) * 2006-10-31 2010-03-18 ヤンセン ファーマシューティカ エヌ．ベー． Ａｄｐｐ２ｙ１２レセプターアンタゴニストとしてのトリアゾロピリミジン誘導体
EP2340252B1 (en) * 2008-09-09 2015-11-11 AstraZeneca AB A process for preparing [1s- ]1-alpha, 2-alpha, 3-beta (1s*, 2r*) 5-beta] ]-3- [7- [2- (3, 4-dif luorophenyl) -cyclopropylamino]- 5- (propylthio) -3h-1, 2, 3-triazolo [4, 5-d]pyrimidin-3-yl]-5- (2- hydroxyethoxy) cyclopentane-1, 2-diol and to its intermediates
WO2015027431A1 (en) * 2013-08-29 2015-03-05 Merck Sharp & Dohme Corp. 2,2-difluorodioxolo a2a receptor antagonists
WO2015162630A1 (en) * 2014-04-25 2015-10-29 Anlon Chemical Research Organization Novel processes for preparing triazolo [4,5-d]- pyrimidines, including ticagrelor, vianew intermediates and new route of synthesis.
MX2018011453A (es) 2016-03-22 2019-01-10 Merck Sharp & Dohme Moduladores alostericos de receptores de acetilcolina nicotinicos.
CN111116592A (zh) * 2019-11-27 2020-05-08 杭州沧海帆医药科技有限公司 嘧啶并三氮唑类化合物及其医药用途
CN112876485A (zh) * 2021-01-25 2021-06-01 郭丽伟 一种用于治疗子宫平滑肌高频率强直性收缩相关疾病的化合物
EP4436566A1 (en) * 2021-11-22 2024-10-02 Purdue Research Foundation Cell-potent bisubstrate inhibitors for nicotinamide n-methyltransferase (nnmt) and uses thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4742064A (en) 1985-09-10 1988-05-03 Regents Of The University Of Minnesota Antiviral carbocyclic analogs of xylofuranosylpurines
GB8826205D0 (en) 1988-11-09 1988-12-14 Wellcome Found Heterocyclic compounds
US5747496A (en) * 1995-07-11 1998-05-05 Astra Pharmaceuticals Limited Inhibitors of platelet aggregation
EP0946561B1 (en) 1996-12-20 2002-02-13 AstraZeneca AB Triazolo(4,5-d)pyrimidinyl derivatives and their use as medicaments
SE9702774D0 (sv) * 1997-07-22 1997-07-22 Astra Pharma Prod Novel compounds
SE9702772D0 (sv) * 1997-07-22 1997-07-22 Astra Pharma Prod Novel compounds

Also Published As

Publication number Publication date
TR200002380T2 (tr) 2001-03-21
JP2002503663A (ja) 2002-02-05
DE69905451T2 (de) 2003-11-20
HUP0100328A3 (en) 2003-04-28
DE69905451D1 (de) 2003-03-27
ATE232866T1 (de) 2003-03-15
HUP0100328A2 (hu) 2001-09-28
WO1999041254A1 (en) 1999-08-19
NO20004089D0 (no) 2000-08-16
NZ505250A (en) 2002-10-25
EP1056749B1 (en) 2003-02-19
KR20010078696A (ko) 2001-08-21
US6369064B1 (en) 2002-04-09
EP1056749A1 (en) 2000-12-06
AU2650099A (en) 1999-08-30
NO20004089L (no) 2000-10-16
MXPA00007634A (es) 2003-09-10
IL137812A0 (en) 2001-10-31
CA2316264A1 (en) 1999-08-19
BR9907934A (pt) 2000-10-24
CN1291193A (zh) 2001-04-11
SK12242000A3 (sk) 2001-03-12
AR015515A1 (es) 2001-05-02
PL342430A1 (en) 2001-06-04

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