HUP9802795A2 - Elhízás kezelésére alkalmas, béta-adrenerg ágenst és étvágycsökkentő hatású vegyületet tartalmazó gyógyászati készítmények - Google Patents

Elhízás kezelésére alkalmas, béta-adrenerg ágenst és étvágycsökkentő hatású vegyületet tartalmazó gyógyászati készítmények

Info

Publication number
HUP9802795A2
HUP9802795A2 HU9802795A HUP9802795A HUP9802795A2 HU P9802795 A2 HUP9802795 A2 HU P9802795A2 HU 9802795 A HU9802795 A HU 9802795A HU P9802795 A HUP9802795 A HU P9802795A HU P9802795 A2 HUP9802795 A2 HU P9802795A2
Authority
HU
Hungary
Prior art keywords
agent
corpulence
treatment
pharmaceutical compositions
compositions containing
Prior art date
Application number
HU9802795A
Other languages
English (en)
Inventor
Robert Lee Dow
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of HU9802795D0 publication Critical patent/HU9802795D0/hu
Publication of HUP9802795A2 publication Critical patent/HUP9802795A2/hu
Publication of HUP9802795A3 publication Critical patent/HUP9802795A3/hu

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/2264—Obesity-gene products, e.g. leptin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Genetics & Genomics (AREA)
  • Child & Adolescent Psychology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

A találmány őlyan gyógyászati készítményekre vőnatkőzik, amelyekegyrészt egy, az étkezési magatartást módősító vegyületet, ennekprődrűgját vagy ennek gyógyászatilag elfőgadható sóját vagy az űtóbbiprődrűgját, másrészt (4-(2-(2-(6-aminő-piridin-3-il)-2(R)-hidrőxi-etil-aminő)-etőxi)-fenil)-ecetsavat, ennek prődrűgját vagy az említett(4-(2-(2-(6-aminő-piridin-3-il)-2(R)-hidrőxi-etil-aminő)-etőxi)-fenil)-ecet- sav gyógyászatilag elfőgadható sóját vagy az űtóbbiprődrűgját tartalmazzák. A találmány szerinti gyógyászati készítményekelhízás és diabétesz kezelésére hasznősíthatók. ŕ
HU9802795A 1997-12-03 1998-12-02 Pharmaceutical compositions containing beta-adrenergic agent and anorectic agent for the treatment of corpulence HUP9802795A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6726897P 1997-12-03 1997-12-03

Publications (3)

Publication Number Publication Date
HU9802795D0 HU9802795D0 (en) 1999-01-28
HUP9802795A2 true HUP9802795A2 (hu) 1999-08-30
HUP9802795A3 HUP9802795A3 (en) 2000-01-28

Family

ID=22074866

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9802795A HUP9802795A3 (en) 1997-12-03 1998-12-02 Pharmaceutical compositions containing beta-adrenergic agent and anorectic agent for the treatment of corpulence

Country Status (7)

Country Link
EP (1) EP0920864A1 (hu)
JP (1) JPH11228447A (hu)
KR (1) KR19990062718A (hu)
AU (1) AU9605598A (hu)
CA (1) CA2255318A1 (hu)
HU (1) HUP9802795A3 (hu)
IL (1) IL127306A0 (hu)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH11515027A (ja) * 1995-11-01 1999-12-21 メルク エンド カンパニー インコーポレーテッド 糖尿病と肥満の治療のための組合せ療法
US6246876B1 (en) 1997-11-13 2001-06-12 Telefonaktiebolaget L M Ericsson (Publ) Synchronization messages for hand-off operations
US6090942A (en) * 1998-10-15 2000-07-18 Pfizer Inc. Process and intermediates for a β3 -adrenergic receptor agonist
KR20010102198A (ko) * 1999-02-16 2001-11-15 후루타 타케시 치환 아세틸피리딘 유도체 및 그를 이용하는 광학활성 β3작용제 중간체의 제조 방법
US6344481B1 (en) * 1999-03-01 2002-02-05 Pfizer Inc. Thyromimetic antiobesity agents
US7115750B1 (en) 1999-09-20 2006-10-03 Takeda Pharmaceutical Company Limited Melanin concentrating hormone antagonist
FR2814678B1 (fr) † 2000-10-04 2002-12-20 Aventis Pharma Sa Association d'un antagoniste du recepteur cb1 et de sibutramine, les compositions pharmaceutiques les contenant et leur utilisation pour la traitement de l'obesite
IL160983A0 (en) 2001-09-24 2004-08-31 Imp College Innovations Ltd Use of pyy for preparation of a medicament for modification of feeding behavior
US8058233B2 (en) 2002-01-10 2011-11-15 Oregon Health And Science University Modification of feeding behavior using PYY and GLP-1
EP1474163A2 (en) * 2002-01-10 2004-11-10 Imperial College Innovations Limited Modification of feeding behavior
EP1496838B1 (en) 2002-03-12 2010-11-03 Merck Sharp & Dohme Corp. Substituted amides
GB0300571D0 (en) * 2003-01-10 2003-02-12 Imp College Innovations Ltd Modification of feeding behaviour
PE20071162A1 (es) * 2005-12-21 2007-11-30 Schering Corp Combinacion de un antagonista/agonista inverso de h3 y un supresor del apetito
WO2007139062A1 (ja) * 2006-05-30 2007-12-06 Kyorin Pharmaceutical Co., Ltd. 肥満治療剤並びに肥満の治療及び予防方法
TWI428346B (zh) 2006-12-13 2014-03-01 Imp Innovations Ltd 新穎化合物及其等對進食行為影響
JP6253451B2 (ja) 2014-02-05 2017-12-27 学校法人自治医科大学 満腹感持続剤および満足感を維持する方法
EP3393470B1 (en) 2015-12-22 2021-01-20 Zogenix International Limited Metabolism resistant fenfluramine analogs and methods of using the same
KR20180091924A (ko) 2015-12-22 2018-08-16 조게닉스 인터내셔널 리미티드 펜플루라민 조성물 및 그 제조 방법
CN109689103A (zh) 2016-08-24 2019-04-26 周格尼克斯国际有限公司 用于抑制5-ht2b激动剂的形成的制剂及其使用方法
US10682317B2 (en) 2017-09-26 2020-06-16 Zogenix International Limited Ketogenic diet compatible fenfluramine formulation
WO2019216919A1 (en) 2018-05-11 2019-11-14 Zogenix International Limited Compositions and methods for treating seizure-induced sudden death
US11612574B2 (en) 2020-07-17 2023-03-28 Zogenix International Limited Method of treating patients infected with severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH11504648A (ja) * 1995-05-10 1999-04-27 ファイザー・インコーポレーテッド β−アドレナリン作動性アゴニスト
WO1996035671A1 (en) * 1995-05-10 1996-11-14 Pfizer Inc. β-ADRENERGIC AGONISTS
JPH11515027A (ja) * 1995-11-01 1999-12-21 メルク エンド カンパニー インコーポレーテッド 糖尿病と肥満の治療のための組合せ療法

Also Published As

Publication number Publication date
HU9802795D0 (en) 1999-01-28
JPH11228447A (ja) 1999-08-24
IL127306A0 (en) 1999-09-22
KR19990062718A (ko) 1999-07-26
HUP9802795A3 (en) 2000-01-28
EP0920864A1 (en) 1999-06-09
AU9605598A (en) 1999-06-24
CA2255318A1 (en) 1999-06-03

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