HUP0600304A2 - Compounds active at the glucocorticoid receptor ii - Google Patents

Compounds active at the glucocorticoid receptor ii

Info

Publication number
HUP0600304A2
HUP0600304A2 HU0600304A HUP0600304A HUP0600304A2 HU P0600304 A2 HUP0600304 A2 HU P0600304A2 HU 0600304 A HU0600304 A HU 0600304A HU P0600304 A HUP0600304 A HU P0600304A HU P0600304 A2 HUP0600304 A2 HU P0600304A2
Authority
HU
Hungary
Prior art keywords
glucocorticoid receptor
compounds active
compounds
active
glucocorticoid
Prior art date
Application number
HU0600304A
Other languages
English (en)
Inventor
Benjamin Pelcman
Annika Gustafsson
Philip R Kym
Original Assignee
Karobio Ab
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Karobio Ab, Abbott Lab filed Critical Karobio Ab
Publication of HUP0600304A2 publication Critical patent/HUP0600304A2/hu

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    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/185Saturated compounds having only one carboxyl group and containing keto groups
    • C07C59/215Saturated compounds having only one carboxyl group and containing keto groups containing singly bound oxygen containing groups
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
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  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • General Chemical & Material Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • General Health & Medical Sciences (AREA)
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  • Veterinary Medicine (AREA)
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  • Diabetes (AREA)
  • Neurology (AREA)
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  • Obesity (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
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  • Cardiology (AREA)
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  • Virology (AREA)
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  • Addiction (AREA)
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HU0600304A 2000-11-29 2001-11-28 Compounds active at the glucocorticoid receptor ii HUP0600304A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0029102.1A GB0029102D0 (en) 2000-11-29 2000-11-29 Compounds active at the glucocorticoid receptor
PCT/IB2001/002302 WO2002043648A2 (en) 2000-11-29 2001-11-28 Compounds active at the glucocorticoid receptor ii

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HUP0600304A2 true HUP0600304A2 (en) 2006-08-28

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HU0600304A HUP0600304A2 (en) 2000-11-29 2001-11-28 Compounds active at the glucocorticoid receptor ii

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US (1) US7220752B2 (hu)
EP (1) EP1509188A4 (hu)
JP (1) JP2004536025A (hu)
KR (1) KR20030076583A (hu)
CN (1) CN1630515A (hu)
AU (1) AU2002223105A1 (hu)
BG (1) BG107871A (hu)
CA (1) CA2430311A1 (hu)
CZ (1) CZ20031310A3 (hu)
GB (1) GB0029102D0 (hu)
HU (1) HUP0600304A2 (hu)
MX (1) MXPA03004658A (hu)
NO (1) NO20032415D0 (hu)
PL (1) PL366056A1 (hu)
SK (1) SK6492003A3 (hu)
TR (1) TR200300763T2 (hu)
WO (1) WO2002043648A2 (hu)
ZA (1) ZA200303453B (hu)

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Publication number Priority date Publication date Assignee Title
US8097606B2 (en) 2003-07-23 2012-01-17 Corcept Therapeutics, Inc. Antiglucocorticoids for the treatment of catatonia
WO2005012221A1 (ja) * 2003-08-04 2005-02-10 Ono Pharmaceutical Co., Ltd. ジフェニルエーテル化合物、その製造方法および用途
US8795693B2 (en) * 2003-08-04 2014-08-05 Foamix Ltd. Compositions with modulating agents
US8986677B2 (en) * 2012-07-30 2015-03-24 Pop Test Cortisol Llc Therapeutic compositions and methods
US11723888B2 (en) 2021-12-09 2023-08-15 Nanopharmaceuticals Llc Polymer conjugated thyrointegrin antagonists

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1143948A3 (en) 1998-06-08 2002-09-11 Karo Bio Ab Liver-selective glucocorticoid antagonist for treating diabetes
GB9816935D0 (en) 1998-08-05 1998-09-30 Karobio Ab Novel glucocortoid and thyroid receptor ligands for the treatment of metabolic disorders

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Publication number Publication date
NO20032415L (no) 2003-05-27
JP2004536025A (ja) 2004-12-02
EP1509188A2 (en) 2005-03-02
GB0029102D0 (en) 2001-01-10
WO2002043648A3 (en) 2004-12-29
EP1509188A4 (en) 2005-11-23
WO2002043648A2 (en) 2002-06-06
CN1630515A (zh) 2005-06-22
WO2002043648A8 (en) 2002-09-06
PL366056A1 (en) 2005-01-24
SK6492003A3 (en) 2003-11-04
CA2430311A1 (en) 2002-06-06
US7220752B2 (en) 2007-05-22
ZA200303453B (en) 2005-05-26
US20040063781A1 (en) 2004-04-01
AU2002223105A1 (en) 2002-06-11
NO20032415D0 (no) 2003-05-27
KR20030076583A (ko) 2003-09-26
CZ20031310A3 (cs) 2003-10-15
TR200300763T2 (tr) 2004-09-21
BG107871A (bg) 2004-02-27
MXPA03004658A (es) 2003-09-04

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