MXPA03004658A - Compuestos activos en el receptor glucocorticoide ii. - Google Patents
Compuestos activos en el receptor glucocorticoide ii.Info
- Publication number
- MXPA03004658A MXPA03004658A MXPA03004658A MXPA03004658A MXPA03004658A MX PA03004658 A MXPA03004658 A MX PA03004658A MX PA03004658 A MXPA03004658 A MX PA03004658A MX PA03004658 A MXPA03004658 A MX PA03004658A MX PA03004658 A MXPA03004658 A MX PA03004658A
- Authority
- MX
- Mexico
- Prior art keywords
- glucocorticoid receptor
- compounds active
- compounds
- active
- glucocorticoid
- Prior art date
Links
Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/30—Oxygen atoms
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- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/185—Saturated compounds having only one carboxyl group and containing keto groups
- C07C59/215—Saturated compounds having only one carboxyl group and containing keto groups containing singly bound oxygen containing groups
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- C07C205/35—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
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- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
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- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Endocrinology (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Psychiatry (AREA)
- Pulmonology (AREA)
- Reproductive Health (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Urology & Nephrology (AREA)
- Oncology (AREA)
- Dermatology (AREA)
- Emergency Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Cardiology (AREA)
- Addiction (AREA)
- Virology (AREA)
- Ophthalmology & Optometry (AREA)
- Heart & Thoracic Surgery (AREA)
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0029102.1A GB0029102D0 (en) | 2000-11-29 | 2000-11-29 | Compounds active at the glucocorticoid receptor |
PCT/IB2001/002302 WO2002043648A2 (en) | 2000-11-29 | 2001-11-28 | Compounds active at the glucocorticoid receptor ii |
Publications (1)
Publication Number | Publication Date |
---|---|
MXPA03004658A true MXPA03004658A (es) | 2003-09-04 |
Family
ID=9904103
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MXPA03004658A MXPA03004658A (es) | 2000-11-29 | 2001-11-28 | Compuestos activos en el receptor glucocorticoide ii. |
Country Status (18)
Country | Link |
---|---|
US (1) | US7220752B2 (es) |
EP (1) | EP1509188A4 (es) |
JP (1) | JP2004536025A (es) |
KR (1) | KR20030076583A (es) |
CN (1) | CN1630515A (es) |
AU (1) | AU2002223105A1 (es) |
BG (1) | BG107871A (es) |
CA (1) | CA2430311A1 (es) |
CZ (1) | CZ20031310A3 (es) |
GB (1) | GB0029102D0 (es) |
HU (1) | HUP0600304A2 (es) |
MX (1) | MXPA03004658A (es) |
NO (1) | NO20032415D0 (es) |
PL (1) | PL366056A1 (es) |
SK (1) | SK6492003A3 (es) |
TR (1) | TR200300763T2 (es) |
WO (1) | WO2002043648A2 (es) |
ZA (1) | ZA200303453B (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8097606B2 (en) | 2003-07-23 | 2012-01-17 | Corcept Therapeutics, Inc. | Antiglucocorticoids for the treatment of catatonia |
EP1661879A4 (en) * | 2003-08-04 | 2006-11-29 | Ono Pharmaceutical Co | A DIPHENYL ETHER COMPOUND, PROCESS FOR THE PRODUCTION AND USE THEREOF |
US8795693B2 (en) * | 2003-08-04 | 2014-08-05 | Foamix Ltd. | Compositions with modulating agents |
US8986677B2 (en) * | 2012-07-30 | 2015-03-24 | Pop Test Cortisol Llc | Therapeutic compositions and methods |
US11723888B2 (en) | 2021-12-09 | 2023-08-15 | Nanopharmaceuticals Llc | Polymer conjugated thyrointegrin antagonists |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1999063976A2 (en) | 1998-06-08 | 1999-12-16 | Karo Bio Ab | Liver-selective glucocorticoid antagonist for treating diabetes |
GB9816935D0 (en) * | 1998-08-05 | 1998-09-30 | Karobio Ab | Novel glucocortoid and thyroid receptor ligands for the treatment of metabolic disorders |
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2000
- 2000-11-29 GB GBGB0029102.1A patent/GB0029102D0/en not_active Ceased
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2001
- 2001-11-28 HU HU0600304A patent/HUP0600304A2/hu unknown
- 2001-11-28 US US10/433,015 patent/US7220752B2/en not_active Expired - Fee Related
- 2001-11-28 WO PCT/IB2001/002302 patent/WO2002043648A2/en not_active Application Discontinuation
- 2001-11-28 CZ CZ20031310A patent/CZ20031310A3/cs unknown
- 2001-11-28 CN CNA018195679A patent/CN1630515A/zh active Pending
- 2001-11-28 AU AU2002223105A patent/AU2002223105A1/en not_active Abandoned
- 2001-11-28 MX MXPA03004658A patent/MXPA03004658A/es unknown
- 2001-11-28 JP JP2002545627A patent/JP2004536025A/ja active Pending
- 2001-11-28 TR TR2003/00763T patent/TR200300763T2/xx unknown
- 2001-11-28 CA CA002430311A patent/CA2430311A1/en not_active Abandoned
- 2001-11-28 PL PL01366056A patent/PL366056A1/xx not_active Application Discontinuation
- 2001-11-28 KR KR10-2003-7007215A patent/KR20030076583A/ko not_active Application Discontinuation
- 2001-11-28 EP EP01998301A patent/EP1509188A4/en not_active Withdrawn
- 2001-11-28 SK SK649-2003A patent/SK6492003A3/sk unknown
-
2003
- 2003-05-06 ZA ZA200303453A patent/ZA200303453B/en unknown
- 2003-05-27 NO NO20032415A patent/NO20032415D0/no not_active Application Discontinuation
- 2003-06-02 BG BG107871A patent/BG107871A/bg unknown
Also Published As
Publication number | Publication date |
---|---|
WO2002043648A2 (en) | 2002-06-06 |
WO2002043648A8 (en) | 2002-09-06 |
SK6492003A3 (en) | 2003-11-04 |
TR200300763T2 (tr) | 2004-09-21 |
HUP0600304A2 (en) | 2006-08-28 |
NO20032415L (no) | 2003-05-27 |
KR20030076583A (ko) | 2003-09-26 |
US7220752B2 (en) | 2007-05-22 |
CA2430311A1 (en) | 2002-06-06 |
GB0029102D0 (en) | 2001-01-10 |
EP1509188A2 (en) | 2005-03-02 |
CZ20031310A3 (cs) | 2003-10-15 |
ZA200303453B (en) | 2005-05-26 |
EP1509188A4 (en) | 2005-11-23 |
US20040063781A1 (en) | 2004-04-01 |
NO20032415D0 (no) | 2003-05-27 |
WO2002043648A3 (en) | 2004-12-29 |
CN1630515A (zh) | 2005-06-22 |
JP2004536025A (ja) | 2004-12-02 |
BG107871A (bg) | 2004-02-27 |
PL366056A1 (en) | 2005-01-24 |
AU2002223105A1 (en) | 2002-06-11 |
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