HUP0300619A3 - Pharmaceutical compositions containing oxadiazole derivatives having anticancer effects - Google Patents

Pharmaceutical compositions containing oxadiazole derivatives having anticancer effects

Info

Publication number
HUP0300619A3
HUP0300619A3 HU0300619A HUP0300619A HUP0300619A3 HU P0300619 A3 HUP0300619 A3 HU P0300619A3 HU 0300619 A HU0300619 A HU 0300619A HU P0300619 A HUP0300619 A HU P0300619A HU P0300619 A3 HUP0300619 A3 HU P0300619A3
Authority
HU
Hungary
Prior art keywords
pharmaceutical compositions
compositions containing
oxadiazole derivatives
anticancer effects
containing oxadiazole
Prior art date
Application number
HU0300619A
Other languages
English (en)
Hungarian (hu)
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of HUP0300619A2 publication Critical patent/HUP0300619A2/hu
Publication of HUP0300619A3 publication Critical patent/HUP0300619A3/hu

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245Oxadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
HU0300619A 2000-04-21 2001-04-16 Pharmaceutical compositions containing oxadiazole derivatives having anticancer effects HUP0300619A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000120234 2000-04-21
PCT/JP2001/003214 WO2001083463A1 (fr) 2000-04-21 2001-04-16 Derives d'oxadiazole efficaces en matiere de traitement ou de prevention d'etats pathologiques glomerulaires

Publications (2)

Publication Number Publication Date
HUP0300619A2 HUP0300619A2 (hu) 2003-07-28
HUP0300619A3 true HUP0300619A3 (en) 2006-02-28

Family

ID=18631080

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0300619A HUP0300619A3 (en) 2000-04-21 2001-04-16 Pharmaceutical compositions containing oxadiazole derivatives having anticancer effects

Country Status (16)

Country Link
US (2) US6720343B2 (US07585860-20090908-C00150.png)
EP (1) EP1277744A4 (US07585860-20090908-C00150.png)
JP (1) JP3974781B2 (US07585860-20090908-C00150.png)
KR (1) KR100542780B1 (US07585860-20090908-C00150.png)
CN (1) CN1199956C (US07585860-20090908-C00150.png)
AU (2) AU2001246916B2 (US07585860-20090908-C00150.png)
BR (1) BR0110211A (US07585860-20090908-C00150.png)
CA (1) CA2406685C (US07585860-20090908-C00150.png)
HU (1) HUP0300619A3 (US07585860-20090908-C00150.png)
MX (1) MXPA02010325A (US07585860-20090908-C00150.png)
NO (1) NO324868B1 (US07585860-20090908-C00150.png)
PL (1) PL203161B1 (US07585860-20090908-C00150.png)
RU (1) RU2275371C2 (US07585860-20090908-C00150.png)
TW (1) TWI294877B (US07585860-20090908-C00150.png)
WO (1) WO2001083463A1 (US07585860-20090908-C00150.png)
ZA (1) ZA200208307B (US07585860-20090908-C00150.png)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030105144A1 (en) 2001-04-17 2003-06-05 Ping Gao Stabilized oral pharmaceutical composition
EP1650199A4 (en) * 2003-07-30 2008-11-19 Shionogi & Co SULPHONAMIDE DERIVATIVE WITH ISOXAZOL RING
US7659294B2 (en) * 2004-10-22 2010-02-09 Merck & Co., Inc. 2-(aryl)azacyclylmethyl carboxylates, sulfonates, phosphonates, phosphinates and heterocycles as S1P receptor agonists
US7576222B2 (en) 2004-12-28 2009-08-18 Wyeth Alkynyl-containing tryptophan derivative inhibitors of TACE/matrix metalloproteinase
GB0601744D0 (en) * 2006-01-27 2006-03-08 Novartis Ag Organic compounds
KR20090007792A (ko) * 2006-05-09 2009-01-20 화이자 프로덕츠 인크. 시클로알킬아미노산 유도체 및 이들의 제약 조성물
KR100783585B1 (ko) 2006-08-22 2007-12-07 한국생명공학연구원 스탯의 활성을 저해하는 옥사다이아졸 우레아 화합물을 유효성분으로 함유하는 암의 예방 또는 치료제
JP5718053B2 (ja) 2007-08-27 2015-05-13 ヘリコン・セラピューティクス・インコーポレーテッド 治療用イソオキサゾール化合物
CA2706834A1 (en) * 2007-12-10 2009-06-18 Actelion Pharmaceuticals Ltd Thiophene derivatives as agonists of s1p1/edg1
AR077969A1 (es) 2009-08-31 2011-10-05 Abbott Healthcare Products Bv Derivados de (tio)morfolina comomoduladores de s1p
TW201643169A (zh) 2010-07-09 2016-12-16 艾伯維股份有限公司 作為s1p調節劑的螺-哌啶衍生物
TWI522361B (zh) 2010-07-09 2016-02-21 艾伯維公司 作為s1p調節劑的稠合雜環衍生物
TW201206893A (en) 2010-07-09 2012-02-16 Abbott Healthcare Products Bv Bisaryl (thio) morpholine derivatives as S1P modulators
CN103450167A (zh) * 2012-05-28 2013-12-18 南京大学 一类含1,3,4-噁二唑和吡嗪环的酰腙类衍生物及其制备方法与用途
US10710994B2 (en) * 2018-03-19 2020-07-14 Genentech, Inc. Oxadiazole transient receptor potential channel inhibitors
EP4051683A1 (en) 2019-10-31 2022-09-07 Escape Bio, Inc. Solid forms of an s1p-receptor modulator
CN113264899B (zh) * 2021-04-09 2022-06-14 台州学院 一种1,3,5-噁二嗪类化合物及其制备和应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69836877D1 (de) 1997-07-22 2007-02-22 Shionogi & Co Verwendung von Matrix- Metalloproteinase Inhibitoren zur Behandlung oder Vorbeugung von Glomerulopathie
WO2000015213A1 (fr) * 1998-09-11 2000-03-23 Shionogi & Co., Ltd. Agent de prevention ou de traitement de l'insuffisance cardiaque congestive

Also Published As

Publication number Publication date
JP3974781B2 (ja) 2007-09-12
US20030203940A1 (en) 2003-10-30
CN1199956C (zh) 2005-05-04
MXPA02010325A (es) 2003-04-25
CA2406685C (en) 2006-10-31
TWI294877B (US07585860-20090908-C00150.png) 2008-03-21
AU4691601A (en) 2001-11-12
KR100542780B1 (ko) 2006-01-11
NO324868B1 (no) 2007-12-17
CA2406685A1 (en) 2002-10-17
KR20030019357A (ko) 2003-03-06
PL203161B1 (pl) 2009-08-31
BR0110211A (pt) 2003-06-03
NO20025035D0 (no) 2002-10-18
AU2001246916B2 (en) 2004-10-07
NO20025035L (no) 2002-12-19
CN1436179A (zh) 2003-08-13
PL359415A1 (en) 2004-08-23
RU2275371C2 (ru) 2006-04-27
EP1277744A1 (en) 2003-01-22
ZA200208307B (en) 2003-10-15
US20040122066A1 (en) 2004-06-24
EP1277744A4 (en) 2007-07-11
WO2001083463A1 (fr) 2001-11-08
HUP0300619A2 (hu) 2003-07-28
US6720343B2 (en) 2004-04-13

Similar Documents

Publication Publication Date Title
GB2358583B (en) Pharmaceutical compositions
HUP0300582A3 (en) Pharmaceutical compositions
IL150447A0 (en) Pharmaceutical compositions containing entecavir
HUP0200530A3 (en) Anticancer compositions containing hydroximatairesinol
HUP0300619A3 (en) Pharmaceutical compositions containing oxadiazole derivatives having anticancer effects
GB0009584D0 (en) Pharmaceutical compositions
HUP0400644A3 (en) Pharmaceutical compositions containing aspirin
AU8576801A (en) Pharmaceutical compositions
IL137363A0 (en) Pharmaceutical compositions containing mupirocin
HUP0400553A3 (en) Pharmaceutical compositions
AU2001246916A1 (en) Oxadiazole derivatives having anticancer effects
HUP0303184A3 (en) Substituted c-cyclohexylmethylamine derivatives and pharmaceutical compositions containing them
AU1390002A (en) Pharmaceutical compositions
HUP0303204A3 (en) 1-methylcarbapenem derivatives and pharmaceutical compositions containing them
GB0009613D0 (en) Pharmaceutical compositions
IL156372A0 (en) Carbazole derivatives and pharmaceutical compositions containing the same
AU4834101A (en) N-deacetylthiocolchicine derivatives and pharmaceutical compositions containing them
IL156174A (en) 1,2,4-oxadiazole derivatives and pharmaceutical compositions containing them
IL149470A0 (en) Pharmaceutical compositions containing carboxamidoadenosine derivatives
AU2001239349A1 (en) Oral pharmaceutical compositions containing n-sulphonylindoline derivatives
PT1326607E (pt) Composições farmacêuticas contendo ácidos oxapenemo-3- carboxílicos
GB0031288D0 (en) Pharmaceutical compositions
HU0700204D0 (en) Pharmaceutical compositions
GB0031282D0 (en) Pharmaceutical compositions
GB0018321D0 (en) Pharmaceutical compositions

Legal Events

Date Code Title Description
FH91 Appointment of a representative

Free format text: FORMER REPRESENTATIVE(S): BELICZAY LASZLO, S.B.G. & K. SZABADALMI UEGYVIVOEI IRODA, HU

Representative=s name: DR. LANG TIVADARNE, S.B.G. & K. SZABADALMI UEG, HU

FH92 Termination of representative

Representative=s name: BELICZAY LASZLO, S.B.G. & K. SZABADALMI UEGYVI, HU

FD9A Lapse of provisional protection due to non-payment of fees