HUP0300569A2 - Pirano[2,3-c]imidazo[1,2-a]piridin-származékok, gasztrointesztinális rendellenességek kezelésére és a vegyületeket tartalmazó gyógyszerkészítmények - Google Patents

Pirano[2,3-c]imidazo[1,2-a]piridin-származékok, gasztrointesztinális rendellenességek kezelésére és a vegyületeket tartalmazó gyógyszerkészítmények

Info

Publication number
HUP0300569A2
HUP0300569A2 HU0300569A HUP0300569A HUP0300569A2 HU P0300569 A2 HUP0300569 A2 HU P0300569A2 HU 0300569 A HU0300569 A HU 0300569A HU P0300569 A HUP0300569 A HU P0300569A HU P0300569 A2 HUP0300569 A2 HU P0300569A2
Authority
HU
Hungary
Prior art keywords
compounds
treatment
pyrano
imidazo
pharmaceutical compositions
Prior art date
Application number
HU0300569A
Other languages
English (en)
Inventor
Wilm Buhr
Wolfgang Kromer
Stefan Postius
Jörg Senn-Bilfinger
Wolfgang-Alexander Simon
Original Assignee
Altana Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Publication of HUP0300569A2 publication Critical patent/HUP0300569A2/hu
Publication of HUP0300569A3 publication Critical patent/HUP0300569A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Az (1) általános képletű vegyületek (mely képletben Rl jelentésemetil- vagy hidroxi-metil-csoport; R2a és R2b közül az egyikhidrogénatomot és a másik hidroxi-, metoxi-, etoxi-, propoxi-,izopropoxi-, butoxi-, metoxi-etoxi- vagy metoxi-propoxi-csoportotképvisel; Ra3 és R3b közül az egyik hidrogénatomot és a másikhidroxi-, metoxi-, etoxi-, propoxi-, izopropoxi-, butoxi-, metoxi-etoxi- vagy metoxi-propoxi-csoportot képvisel; mimellett R2a vagy R2begyrészről és R3a vagy R3b másrészről nem lehet egyidejűleghidroxilcsoport) és sóik a gyomor-bélrendszer betegségei megelőzéséreés kezelésére alkalmazhatók. A találmány kiterjed a vegyületekettartalmazó gyógyszerkészítményekre is. Ó
HU0300569A 2000-03-29 2001-03-28 Pyrano[2,3-c]imidazo[-1,2-a]pyridine derivatives for the treatment of gastrointestinal disorders and pharmaceutical compositions containing the compounds HUP0300569A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00106690 2000-03-29
PCT/EP2001/003510 WO2001072755A1 (en) 2000-03-29 2001-03-28 Pyrano[2,3-c]imidazo[-1,2-a]pyridine derivatives for the treatment of gastrointestinal disorders

Publications (2)

Publication Number Publication Date
HUP0300569A2 true HUP0300569A2 (hu) 2003-07-28
HUP0300569A3 HUP0300569A3 (en) 2004-10-28

Family

ID=8168269

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0300569A HUP0300569A3 (en) 2000-03-29 2001-03-28 Pyrano[2,3-c]imidazo[-1,2-a]pyridine derivatives for the treatment of gastrointestinal disorders and pharmaceutical compositions containing the compounds

Country Status (23)

Country Link
US (2) US20030100578A1 (hu)
EP (1) EP1286999B1 (hu)
JP (1) JP2003528877A (hu)
KR (1) KR20020082494A (hu)
CN (1) CN1221554C (hu)
AT (1) ATE381568T1 (hu)
AU (1) AU784611B2 (hu)
BR (1) BR0109589A (hu)
CA (1) CA2404466A1 (hu)
CZ (1) CZ20023210A3 (hu)
DE (1) DE60131968T2 (hu)
EA (1) EA006095B1 (hu)
ES (1) ES2298233T3 (hu)
HK (1) HK1053838A1 (hu)
HR (1) HRP20020855A2 (hu)
HU (1) HUP0300569A3 (hu)
MX (1) MXPA02009550A (hu)
NO (1) NO20024572D0 (hu)
NZ (1) NZ520836A (hu)
PL (1) PL365824A1 (hu)
SK (1) SK13862002A3 (hu)
WO (1) WO2001072755A1 (hu)
ZA (1) ZA200207635B (hu)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2404460A1 (en) * 2000-03-29 2001-10-04 Altana Pharma Ag Alkylated imidazopyridine derivatives
CN1692113A (zh) 2000-10-25 2005-11-02 奥坦纳医药公司 作为胃分泌抑制剂的多取代咪唑并吡啶
NZ540504A (en) 2002-11-19 2007-12-21 Altana Pharma Ag 8-Substituted imidazopyridines for the treatment of gastrointestinal disorders
CA2515676A1 (en) * 2003-02-17 2004-08-26 Altana Pharma Ag Imidazopyridines containing combinations and their use in treating gastrointestinal inflammatory disorders
AR044129A1 (es) 2003-05-06 2005-08-24 Altana Pharma Ag Compuestos intermedios de imidazopiridina. proceso de preparacion.
MXPA05012463A (es) * 2003-05-27 2006-01-30 Altana Pharma Ag Combinaciones farmaceuticas de un inhibidor de bomba protonica y un compuesto que modifica la motilidad gastrointestinal.
EP1682133A1 (en) 2003-11-03 2006-07-26 AstraZeneca AB Imidazo 1,2-a pyridine derivatives for the treatment of silent gastro-esophageal reflux
CA2549860A1 (en) 2003-12-19 2005-06-30 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives
AR048869A1 (es) * 2004-04-26 2006-06-07 Altana Pharma Ag Bencimidazoles triciclicos
DE102006001335B4 (de) * 2006-01-09 2016-08-04 Rogers Germany Gmbh Verwendung eines wärmetransportierenden Mediums

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9401197D0 (sv) * 1994-04-11 1994-04-11 Astra Ab Active compounds
WO1998042707A1 (en) * 1997-03-24 1998-10-01 Byk Gulden Lomberg Chemische Fabrik Gmbh Tetrahydropyrido compounds
CN1257505A (zh) * 1997-05-28 2000-06-21 比克·古尔顿·劳姆贝尔格化学公司 稠合的二氢吡喃类化合物
CA2404460A1 (en) * 2000-03-29 2001-10-04 Altana Pharma Ag Alkylated imidazopyridine derivatives

Also Published As

Publication number Publication date
HK1053838A1 (en) 2003-11-07
MXPA02009550A (es) 2004-05-14
DE60131968D1 (de) 2008-01-31
PL365824A1 (en) 2005-01-10
NO20024572L (no) 2002-09-24
CA2404466A1 (en) 2001-10-04
EA200200883A1 (ru) 2003-04-24
AU5622801A (en) 2001-10-08
ZA200207635B (en) 2003-10-20
HRP20020855A2 (en) 2004-12-31
BR0109589A (pt) 2003-02-04
EP1286999B1 (en) 2007-12-19
CZ20023210A3 (cs) 2003-01-15
CN1419556A (zh) 2003-05-21
EA006095B1 (ru) 2005-08-25
ES2298233T3 (es) 2008-05-16
DE60131968T2 (de) 2008-12-11
JP2003528877A (ja) 2003-09-30
KR20020082494A (ko) 2002-10-31
ATE381568T1 (de) 2008-01-15
CN1221554C (zh) 2005-10-05
NO20024572D0 (no) 2002-09-24
US6936623B2 (en) 2005-08-30
HUP0300569A3 (en) 2004-10-28
NZ520836A (en) 2005-01-28
WO2001072755A1 (en) 2001-10-04
AU784611B2 (en) 2006-05-11
US20030100578A1 (en) 2003-05-29
US20040180920A1 (en) 2004-09-16
SK13862002A3 (sk) 2003-03-04
EP1286999A1 (en) 2003-03-05

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Legal Events

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FD9A Lapse of provisional protection due to non-payment of fees