HUP0103712A2 - Paroxetin sók, eljárás az előállításukra és gyógyászati alkalmazásuk - Google Patents

Paroxetin sók, eljárás az előállításukra és gyógyászati alkalmazásuk

Info

Publication number
HUP0103712A2
HUP0103712A2 HU0103712A HUP0103712A HUP0103712A2 HU P0103712 A2 HUP0103712 A2 HU P0103712A2 HU 0103712 A HU0103712 A HU 0103712A HU P0103712 A HUP0103712 A HU P0103712A HU P0103712 A2 HUP0103712 A2 HU P0103712A2
Authority
HU
Hungary
Prior art keywords
paroxetine
salts
preparation
pharmaceutical use
acids
Prior art date
Application number
HU0103712A
Other languages
English (en)
Inventor
Victor Witold Jacewicz
Original Assignee
Smithkline Beecham Plc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc. filed Critical Smithkline Beecham Plc.
Publication of HUP0103712A2 publication Critical patent/HUP0103712A2/hu
Publication of HUP0103712A3 publication Critical patent/HUP0103712A3/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

A találmány tárgya a savak csoportjából kiválasztott savak paroxetinsói. A találmány új vegyületekre, előállítási eljárásaikra éskülönféle rendellenességek kezelésében történő felhasználásukravonatkozik. Ó
HU0103712A 1998-07-02 1999-06-30 Salts of paroxetine, process for their preparation and their pharmaceutical use HUP0103712A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9814316.7A GB9814316D0 (en) 1998-07-02 1998-07-02 Novel compounds

Publications (2)

Publication Number Publication Date
HUP0103712A2 true HUP0103712A2 (hu) 2002-05-29
HUP0103712A3 HUP0103712A3 (en) 2002-09-30

Family

ID=10834803

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0103712A HUP0103712A3 (en) 1998-07-02 1999-06-30 Salts of paroxetine, process for their preparation and their pharmaceutical use

Country Status (21)

Country Link
EP (1) EP1091958A1 (hu)
JP (1) JP2002519421A (hu)
KR (1) KR20010053337A (hu)
CN (1) CN1314906A (hu)
AP (1) AP2000002017A0 (hu)
AU (2) AU4903999A (hu)
BG (1) BG105204A (hu)
BR (1) BR9911679A (hu)
CA (1) CA2336470A1 (hu)
CZ (1) CZ20004923A3 (hu)
EA (1) EA200100098A1 (hu)
GB (1) GB9814316D0 (hu)
HU (1) HUP0103712A3 (hu)
ID (1) ID27766A (hu)
IL (1) IL140385A0 (hu)
NO (1) NO20006547L (hu)
PL (1) PL345365A1 (hu)
SK (1) SK20242000A3 (hu)
TR (1) TR200100055T2 (hu)
WO (1) WO2000001692A1 (hu)
ZA (2) ZA992899B (hu)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2524610C (en) 2003-05-07 2014-03-25 Osteologix A/S Strontium combinations for prophylaxis/treatment of cartilage and/or bone conditions
AU2004237439B2 (en) 2003-05-07 2009-09-10 Osteologix A/S Treating cartilage/bone conditions with water-soluble strontium salts
AU2005216596B2 (en) 2004-02-26 2011-03-24 Osteologix A/S Strontium-containing compounds for use in the prevention or treatment of necrotic bone conditions
AU2005240257B2 (en) 2004-05-06 2011-11-24 Osteologix A/S High yield and rapid syntheses methods for producing metallo-organic salts
KR100672184B1 (ko) 2004-09-21 2007-01-19 주식회사종근당 파록세틴의 콜린산 또는 콜린산 유도체 염
US9873667B2 (en) 2006-07-27 2018-01-23 Emisphere Technologies Inc. Arylsulfanyl compounds and compositions for delivering active agents
CN109212055B (zh) * 2018-08-19 2021-05-07 丁立平 一种测定饮用水中四种痕量单卤代苯乙酸的气相色谱-质谱联用法
CN109342633B (zh) * 2018-11-27 2020-10-02 北京市化工职业病防治院 尿液中苯、甲苯和二甲苯代谢物的检测方法
CN111337460B (zh) * 2018-12-18 2021-09-17 中国科学院大连化学物理研究所 一种高稳定性Halo-tag探针及其合成和生物应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8430581D0 (en) * 1984-12-04 1985-01-09 Ferrosan As Treatment
ES2058061T3 (es) * 1985-10-25 1994-11-01 Beecham Group Plc Derivado de piperidina, su preparacion y su uso como medicamento.
CA2206592A1 (en) * 1996-05-30 1997-11-30 Shu-Zhong Wang Method of producing amorphous paroxetine hydrochloride
HU221921B1 (hu) * 1996-07-08 2003-02-28 Richter Gedeon Vegyészeti Gyár Rt. N-benzil-piperidin- és tetrahidropiridinszármazékok és eljárás azok előállítására
AU3108097A (en) * 1997-06-10 1998-12-30 Synthon B.V. 4-phenylpiperidine compounds
JP2002505254A (ja) * 1998-02-06 2002-02-19 スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー パロキセチン塩

Also Published As

Publication number Publication date
IL140385A0 (en) 2002-02-10
HUP0103712A3 (en) 2002-09-30
GB9814316D0 (en) 1998-09-02
NO20006547D0 (no) 2000-12-21
SK20242000A3 (sk) 2001-07-10
ZA992899B (en) 2000-03-29
KR20010053337A (ko) 2001-06-25
AU4903999A (en) 2000-01-24
JP2002519421A (ja) 2002-07-02
EP1091958A1 (en) 2001-04-18
WO2000001692A1 (en) 2000-01-13
TR200100055T2 (tr) 2001-07-23
ZA200100020B (en) 2002-03-25
ID27766A (id) 2001-04-26
CA2336470A1 (en) 2000-01-13
AU2002100370A4 (en) 2002-06-06
AP2000002017A0 (en) 2000-12-31
BG105204A (en) 2001-11-30
PL345365A1 (en) 2001-12-17
EA200100098A1 (ru) 2001-08-27
NO20006547L (no) 2001-02-12
BR9911679A (pt) 2002-01-29
CZ20004923A3 (cs) 2001-08-15
CN1314906A (zh) 2001-09-26

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