HUP0102808A2 - Ektoparaziticid készítmények - Google Patents
Ektoparaziticid készítményekInfo
- Publication number
- HUP0102808A2 HUP0102808A2 HU0102808A HUP0102808A HUP0102808A2 HU P0102808 A2 HUP0102808 A2 HU P0102808A2 HU 0102808 A HU0102808 A HU 0102808A HU P0102808 A HUP0102808 A HU P0102808A HU P0102808 A2 HUP0102808 A2 HU P0102808A2
- Authority
- HU
- Hungary
- Prior art keywords
- alkoxy
- alkyl
- heterocyclic group
- group
- methyl
- Prior art date
Links
- RFEJUZJILGIRHQ-XRIOVQLTSA-N 2,3-dihydroxybutanedioic acid;3-[(2s)-1-methylpyrrolidin-2-yl]pyridine Chemical compound OC(=O)C(O)C(O)C(O)=O.OC(=O)C(O)C(O)C(O)=O.CN1CCC[C@H]1C1=CC=CN=C1 RFEJUZJILGIRHQ-XRIOVQLTSA-N 0.000 title abstract 2
- 239000013057 ectoparasiticide Substances 0.000 title abstract 2
- 239000003795 chemical substances by application Substances 0.000 title 1
- 108010002156 Depsipeptides Proteins 0.000 abstract 4
- 125000000623 heterocyclic group Chemical group 0.000 abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 3
- -1 nitro- Chemical class 0.000 abstract 3
- 125000004183 alkoxy alkyl group Chemical group 0.000 abstract 2
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 229910052717 sulfur Inorganic materials 0.000 abstract 2
- MYMOFIZGZYHOMD-UHFFFAOYSA-N Dioxygen Chemical compound O=O MYMOFIZGZYHOMD-UHFFFAOYSA-N 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000005002 aryl methyl group Chemical group 0.000 abstract 1
- 244000078703 ectoparasite Species 0.000 abstract 1
- 125000005114 heteroarylalkoxy group Chemical group 0.000 abstract 1
- 125000004446 heteroarylalkyl group Chemical group 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
- 239000011593 sulfur Substances 0.000 abstract 1
- 125000004434 sulfur atom Chemical group 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/84—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms six-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,4
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N2300/00—Combinations or mixtures of active ingredients covered by classes A01N27/00 - A01N65/48 with other active or formulation relevant ingredients, e.g. specific carrier materials or surfactants, covered by classes A01N25/00 - A01N65/48
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Inorganic Insulating Materials (AREA)
Abstract
A találmány ciklusos depszipeptidek, különösen 24-tagúciklodepszipeptidek alkalmazása ektoparaziták leküzdésére. A találmánytovábbá depszipeptideket tartalmazó ektoparaziticid készítményekre isvonatkozik. A ciklusos depszipeptidek az (I) általános képletnekfelelnek meg, amelyben X1, X2, X3 és X4 jelentése egymástólfüggetlenül oxigén- vagy kénatom, R1 jelentése hidrogénatom,alkilcsoport, halogénatom, hidroxil-, alkoxi-, alkoxi-alkil-,metilcsoporton keresztül kapcsolódó heterociklusos csoport,heteroaril-alkoxi-, nitro-, NR3R4 vagy -SO2-NR3R4 csoport; R2jelentése hidrogén- vagy halogénatom, alkil-, hidroxil-, alkoxi-,alkoxi-alkil-, metilcsoporton keresztül kapcsolódó heterociklusoscsoport, heteroaril-alkoxi-, nitro-, -NR3R4 vagy -SO2-NR3R4 csoport;R3 és R4 egymástól függetlenül hidrogénatom, alkil-, formil-, alkoxi-karbonil-, aril-metil-, metilcsoporton keresztül kapcsolódóheterociklusos csoport vagy R3 és R4 együtt telített vagy telítetlen,1-3 további heteroatomot tartalmazó heterociklusos csoportot alkot,azzal a megszorítással, hogy R1=R2=H esetén az X1, X2, X3 és X4 közüllegalább egynek a jelentése kénatom. Ó
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19828043A DE19828043A1 (de) | 1998-06-24 | 1998-06-24 | Ektoparasitizide Mittel |
PCT/EP1999/004029 WO1999066794A1 (de) | 1998-06-24 | 1999-06-11 | Ektoparasitizide mittel |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP0102808A2 true HUP0102808A2 (hu) | 2001-11-28 |
HUP0102808A3 HUP0102808A3 (en) | 2002-12-28 |
Family
ID=7871810
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU0102808A HUP0102808A3 (en) | 1998-06-24 | 1999-06-11 | Ectoparasiticide agents |
Country Status (16)
Country | Link |
---|---|
US (1) | US6630569B1 (hu) |
EP (1) | EP1089625B1 (hu) |
JP (1) | JP4404484B2 (hu) |
KR (1) | KR20010043938A (hu) |
CN (1) | CN1306394A (hu) |
AT (1) | ATE229269T1 (hu) |
AU (1) | AU751711B2 (hu) |
BR (1) | BR9912199A (hu) |
CA (1) | CA2336129C (hu) |
DE (2) | DE19828043A1 (hu) |
DK (1) | DK1089625T3 (hu) |
ES (1) | ES2186371T3 (hu) |
HU (1) | HUP0102808A3 (hu) |
NZ (1) | NZ509105A (hu) |
PT (1) | PT1089625E (hu) |
WO (1) | WO1999066794A1 (hu) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE19962147A1 (de) * | 1999-12-22 | 2001-06-28 | Bayer Ag | Schädlingsbekämpfungsmittel / PF 1022-221 |
DE19962145A1 (de) | 1999-12-22 | 2001-06-28 | Bayer Ag | Schädlingsbekämpfungsmittel/Depsipeptide |
WO2008006058A2 (en) * | 2006-07-06 | 2008-01-10 | Stepan Company | Alkyl lactyllactate solvent compositions |
WO2008006076A2 (en) | 2006-07-06 | 2008-01-10 | Stepan Company | Alkyl lactyllactates and processes of making the same |
ES2632392T3 (es) | 2007-08-17 | 2017-09-12 | Novartis Ag | Depsipéptidos cíclicos |
US8614289B2 (en) | 2011-04-20 | 2013-12-24 | Novartis Ag | Processes for the manufacture of macrocyclic depsipeptides and new intermediates |
US8680054B2 (en) * | 2011-04-20 | 2014-03-25 | Novartis Ag | Suspension type topical formulations comprising cyclic depsipeptide |
MX2014014838A (es) * | 2012-06-13 | 2015-02-12 | Meiji Seika Pharma Co Ltd | Nuevos derivados de depsipeptidos ciclicos y agentes para el control de organismos dañinos que comprenden los mismos. |
US9067978B2 (en) | 2012-10-09 | 2015-06-30 | Novartis Ag | Solution phase processes for the manufacture of macrocyclic depsipeptides and new intermediates |
US8987413B2 (en) | 2012-10-09 | 2015-03-24 | Novartis Ag | Aldehyde acetal based processes for the manufacture of macrocyclic depsipeptides and new intermediates |
NZ737610A (en) | 2015-05-20 | 2023-07-28 | Boehringer Ingelheim Animal Health Usa Inc | Anthelmintic depsipeptide compounds |
US10344056B2 (en) | 2015-12-28 | 2019-07-09 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic depsipeptide compounds |
MX2019005628A (es) | 2016-11-16 | 2019-12-18 | Boehringer Ingelheim Animal Health Usa Inc | Compuestos depsipeptidos antihelminticos. |
UA125155C2 (uk) * | 2017-11-29 | 2022-01-19 | Зоетіс Сервісіс Ллк | Анти-ендопаразитарні депсипептиди |
MX2020011980A (es) | 2018-05-10 | 2021-03-26 | Zoetis Services Llc | Depsipéptidos endoparasiticidas. |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU669883B2 (en) | 1992-03-17 | 1996-06-27 | Astellas Pharma Inc. | Depsipeptide derivative, production thereof and use thereof |
JPH05271013A (ja) * | 1992-03-27 | 1993-10-19 | Meiji Seika Kaisha Ltd | 環状デプシペプチド物質を有効成分とする害虫防除剤 |
DE4412492A1 (de) * | 1994-04-12 | 1995-10-19 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen |
CN1196056A (zh) * | 1995-09-07 | 1998-10-14 | 法玛西雅厄普约翰公司 | 环化蠕虫抑制剂 |
-
1998
- 1998-06-24 DE DE19828043A patent/DE19828043A1/de not_active Withdrawn
-
1999
- 1999-06-11 AU AU46078/99A patent/AU751711B2/en not_active Ceased
- 1999-06-11 HU HU0102808A patent/HUP0102808A3/hu unknown
- 1999-06-11 EP EP99929178A patent/EP1089625B1/de not_active Expired - Lifetime
- 1999-06-11 ES ES99929178T patent/ES2186371T3/es not_active Expired - Lifetime
- 1999-06-11 PT PT99929178T patent/PT1089625E/pt unknown
- 1999-06-11 CN CN99807711A patent/CN1306394A/zh active Pending
- 1999-06-11 AT AT99929178T patent/ATE229269T1/de active
- 1999-06-11 US US09/719,626 patent/US6630569B1/en not_active Expired - Lifetime
- 1999-06-11 JP JP2000555494A patent/JP4404484B2/ja not_active Expired - Fee Related
- 1999-06-11 DE DE59903759T patent/DE59903759D1/de not_active Expired - Lifetime
- 1999-06-11 KR KR1020007013506A patent/KR20010043938A/ko not_active Application Discontinuation
- 1999-06-11 DK DK99929178T patent/DK1089625T3/da active
- 1999-06-11 WO PCT/EP1999/004029 patent/WO1999066794A1/de not_active Application Discontinuation
- 1999-06-11 CA CA002336129A patent/CA2336129C/en not_active Expired - Fee Related
- 1999-06-11 BR BR9912199-9A patent/BR9912199A/pt not_active Application Discontinuation
- 1999-06-11 NZ NZ509105A patent/NZ509105A/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
ATE229269T1 (de) | 2002-12-15 |
BR9912199A (pt) | 2001-04-10 |
PT1089625E (pt) | 2003-04-30 |
CN1306394A (zh) | 2001-08-01 |
DE19828043A1 (de) | 1999-12-30 |
EP1089625A1 (de) | 2001-04-11 |
NZ509105A (en) | 2002-12-20 |
DE59903759D1 (de) | 2003-01-23 |
KR20010043938A (ko) | 2001-05-25 |
HUP0102808A3 (en) | 2002-12-28 |
CA2336129C (en) | 2008-12-02 |
JP4404484B2 (ja) | 2010-01-27 |
DK1089625T3 (da) | 2003-03-24 |
ES2186371T3 (es) | 2003-05-01 |
CA2336129A1 (en) | 1999-12-29 |
AU751711B2 (en) | 2002-08-22 |
EP1089625B1 (de) | 2002-12-11 |
US6630569B1 (en) | 2003-10-07 |
AU4607899A (en) | 2000-01-10 |
WO1999066794A1 (de) | 1999-12-29 |
JP2002518415A (ja) | 2002-06-25 |
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