ES2186371T3 - Agentes endoparasiticidas. - Google Patents
Agentes endoparasiticidas.Info
- Publication number
- ES2186371T3 ES2186371T3 ES99929178T ES99929178T ES2186371T3 ES 2186371 T3 ES2186371 T3 ES 2186371T3 ES 99929178 T ES99929178 T ES 99929178T ES 99929178 T ES99929178 T ES 99929178T ES 2186371 T3 ES2186371 T3 ES 2186371T3
- Authority
- ES
- Spain
- Prior art keywords
- carbon atoms
- methoxy
- alkoxy
- alkyl
- mean
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- -1 tert-butyloxy Chemical group 0.000 abstract 11
- 125000004432 carbon atom Chemical group C* 0.000 abstract 10
- 125000003545 alkoxy group Chemical group 0.000 abstract 4
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 239000001257 hydrogen Substances 0.000 abstract 4
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 4
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 125000005344 pyridylmethyl group Chemical group [H]C1=C([H])C([H])=C([H])C(=N1)C([H])([H])* 0.000 abstract 3
- 229910052717 sulfur Inorganic materials 0.000 abstract 3
- 239000011593 sulfur Substances 0.000 abstract 3
- 125000006223 tetrahydrofuranylmethyl group Chemical group 0.000 abstract 3
- 125000005301 thienylmethyl group Chemical group [H]C1=C([H])C([H])=C(S1)C([H])([H])* 0.000 abstract 3
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 2
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 2
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 2
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
- 229910052799 carbon Inorganic materials 0.000 abstract 2
- 229910052731 fluorine Inorganic materials 0.000 abstract 2
- 239000011737 fluorine Substances 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 125000005114 heteroarylalkoxy group Chemical group 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 2
- 125000004184 methoxymethyl group Chemical group [H]C([H])([H])OC([H])([H])* 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
- 229910052757 nitrogen Inorganic materials 0.000 abstract 2
- 229910052760 oxygen Inorganic materials 0.000 abstract 2
- 239000001301 oxygen Substances 0.000 abstract 2
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000005002 aryl methyl group Chemical group 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 244000078703 ectoparasite Species 0.000 abstract 1
- 125000005448 ethoxyethyl group Chemical group [H]C([H])([H])C([H])([H])OC([H])([H])C([H])([H])* 0.000 abstract 1
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000002950 monocyclic group Chemical group 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 125000003367 polycyclic group Chemical group 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/84—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms six-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,4
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N2300/00—Combinations or mixtures of active ingredients covered by classes A01N27/00 - A01N65/48 with other active or formulation relevant ingredients, e.g. specific carrier materials or surfactants, covered by classes A01N25/00 - A01N65/48
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Inorganic Insulating Materials (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Empleo de ciclooctadepsipéptidos de la fórmula (I) **(Fórmula)** en la que R1 significa hidrógeno, alquilo con 1 a 4 átomos de carbono, especialmente metilo, hidroxi, halógeno, especialmente flúor, alcoxi con 1 a 4 átomos de carbono, especialmente metoxi o terc.-butiloxi, alcoxi con 1 a 4 átomos de carbono-alquilo con 1 a 4 átomos de carbono, especialmente metoximetilo, metoxietilo, heterociclilmetilo, especialmente piridilmetilo, tetrahidrofuranil-metilo, pirrolidinilmetilo, furilmetilo, tienilmetilo, heteroaril-alcoxi con 1 a 2 átomos de carbono, especialmente piridil-metoxi, tetrahidrofuril-metoxi, pirrolidinil-metoxi y furil-metoxi, nitro, -NR3R4 , -SO2-NR3R4 , R2 significa hidrógeno, alquilo con 1 a 4 átomos de carbono, especialmente metilo, hidroxi, halógeno, especialmente flúor, alcoxi con 1 a 4 átomos de carbono, especialmente metoxi o terc.-butiloxi, alcoxi con 1 a 4 átomos de carbono-alquilo con 1 a 4 átomos de carbono, especialmente metoximetilo, etoxietilo, heterociclilmetilo, especialmente piridilmetilo, tetrahidrofuranil-metilo, pirrolidinilmetilo, furilmetil. tienilmetilo, heteroaril-alcoxi con 1 a 2 átomos de carbono, especialmente piridil-metoxi, tetrahidrofuranil-metoxi, pirrolidinil-metoxi y furilmetoxi, nitro, -NRR, -SO2-NR3R4 , R3 y R4 significan, independientemente entre si, respectivamente hidrógeno, alquilo con 1 a 4 átomos de carbono, substituido en caso dado, formilo, alcoxicarbonilo con 1 a 4 átomos de carbono, arilmetilo substituido en caso dado, especialmente bencilo, o heterociclilmetilo, especialmente piridilmetilo, tetrahidrofuranilmetilo, pirrolidinilmetilo, furilmetilo, tienil-metilo, R3 y R4 significan junto con el átomo de nitrógeno, con el que están enlazados, un heterociclo, en caso dado substituido, mono- o policíclico, en caso dado puenteado y/o espirocíclico, saturado o insaturado, que puede contener de una a tres heteroátomos mas de la serie formada por nitrógeno, oxígeno y azufre, X1, X2, X3 y X4 significan, independientemente entresi, oxígeno o azufre, significando azufre al menos uno de los restos X1, X2, X3 y X4 en el caso en que R1 y R2 signifiquen, simultáneamente, hidrógeno, para la obtención de agentes para la lucha contra los ectoparásitos.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19828043A DE19828043A1 (de) | 1998-06-24 | 1998-06-24 | Ektoparasitizide Mittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2186371T3 true ES2186371T3 (es) | 2003-05-01 |
Family
ID=7871810
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES99929178T Expired - Lifetime ES2186371T3 (es) | 1998-06-24 | 1999-06-11 | Agentes endoparasiticidas. |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US6630569B1 (es) |
| EP (1) | EP1089625B1 (es) |
| JP (1) | JP4404484B2 (es) |
| KR (1) | KR20010043938A (es) |
| CN (1) | CN1306394A (es) |
| AT (1) | ATE229269T1 (es) |
| AU (1) | AU751711B2 (es) |
| BR (1) | BR9912199A (es) |
| CA (1) | CA2336129C (es) |
| DE (2) | DE19828043A1 (es) |
| DK (1) | DK1089625T3 (es) |
| ES (1) | ES2186371T3 (es) |
| HU (1) | HUP0102808A3 (es) |
| NZ (1) | NZ509105A (es) |
| PT (1) | PT1089625E (es) |
| WO (1) | WO1999066794A1 (es) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19962147A1 (de) | 1999-12-22 | 2001-06-28 | Bayer Ag | Schädlingsbekämpfungsmittel / PF 1022-221 |
| DE19962145A1 (de) * | 1999-12-22 | 2001-06-28 | Bayer Ag | Schädlingsbekämpfungsmittel/Depsipeptide |
| WO2008006058A2 (en) * | 2006-07-06 | 2008-01-10 | Stepan Company | Alkyl lactyllactate solvent compositions |
| ES2395676T3 (es) | 2006-07-06 | 2013-02-14 | Stepan Company | Procedimientos de preparación de lactil lactatos de alquilo |
| PT2183273T (pt) | 2007-08-17 | 2017-05-22 | Novartis Ag | Depsipéptidos cíclicos |
| AR086168A1 (es) | 2011-04-20 | 2013-11-27 | Novartis Ag | Procesos para la elaboracion de depsipeptidos macrociclicos e intermediarios |
| US8680054B2 (en) | 2011-04-20 | 2014-03-25 | Novartis Ag | Suspension type topical formulations comprising cyclic depsipeptide |
| NZ703217A (en) * | 2012-06-13 | 2016-11-25 | Meiji Seika Pharma Co Ltd | Novel cyclic depsipeptide derivatives and harmful organism control agents comprising the same |
| US8987413B2 (en) | 2012-10-09 | 2015-03-24 | Novartis Ag | Aldehyde acetal based processes for the manufacture of macrocyclic depsipeptides and new intermediates |
| US9067978B2 (en) | 2012-10-09 | 2015-06-30 | Novartis Ag | Solution phase processes for the manufacture of macrocyclic depsipeptides and new intermediates |
| RS62130B1 (sr) * | 2015-05-20 | 2021-08-31 | Boehringer Ingelheim Animal Health Usa Inc | Antihelmintička depsipeptidna jedinjenja |
| RU2715556C2 (ru) | 2015-12-28 | 2020-03-02 | Мериал, Инк. | Противогельминтные депсипептидные соединения |
| WO2018093920A1 (en) | 2016-11-16 | 2018-05-24 | Merial, Inc. | Anthelmintic depsipeptide compounds |
| KR102467784B1 (ko) * | 2017-11-29 | 2022-11-17 | 조에티스 서비시즈 엘엘씨 | 체내기생충성 뎁시펩티드 |
| JP7260564B2 (ja) * | 2018-05-10 | 2023-04-18 | ゾエティス・サービシーズ・エルエルシー | 内部寄生性デプシペプチド |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1993019053A1 (fr) | 1992-03-17 | 1993-09-30 | Fujisawa Pharmaceutical Co., Ltd. | Derive de depsipeptide, production et utilisation |
| JPH05271013A (ja) * | 1992-03-27 | 1993-10-19 | Meiji Seika Kaisha Ltd | 環状デプシペプチド物質を有効成分とする害虫防除剤 |
| DE4412492A1 (de) * | 1994-04-12 | 1995-10-19 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen |
| KR19990044489A (ko) * | 1995-09-07 | 1999-06-25 | 로렌스 티. 마이젠헬더 | 환식 구충제 |
-
1998
- 1998-06-24 DE DE19828043A patent/DE19828043A1/de not_active Withdrawn
-
1999
- 1999-06-11 CN CN99807711A patent/CN1306394A/zh active Pending
- 1999-06-11 US US09/719,626 patent/US6630569B1/en not_active Expired - Lifetime
- 1999-06-11 ES ES99929178T patent/ES2186371T3/es not_active Expired - Lifetime
- 1999-06-11 KR KR1020007013506A patent/KR20010043938A/ko not_active Application Discontinuation
- 1999-06-11 DK DK99929178T patent/DK1089625T3/da active
- 1999-06-11 WO PCT/EP1999/004029 patent/WO1999066794A1/de not_active Application Discontinuation
- 1999-06-11 AT AT99929178T patent/ATE229269T1/de active
- 1999-06-11 CA CA002336129A patent/CA2336129C/en not_active Expired - Fee Related
- 1999-06-11 AU AU46078/99A patent/AU751711B2/en not_active Ceased
- 1999-06-11 EP EP99929178A patent/EP1089625B1/de not_active Expired - Lifetime
- 1999-06-11 PT PT99929178T patent/PT1089625E/pt unknown
- 1999-06-11 BR BR9912199-9A patent/BR9912199A/pt not_active Application Discontinuation
- 1999-06-11 NZ NZ509105A patent/NZ509105A/xx not_active IP Right Cessation
- 1999-06-11 JP JP2000555494A patent/JP4404484B2/ja not_active Expired - Fee Related
- 1999-06-11 HU HU0102808A patent/HUP0102808A3/hu unknown
- 1999-06-11 DE DE59903759T patent/DE59903759D1/de not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| WO1999066794A1 (de) | 1999-12-29 |
| DK1089625T3 (da) | 2003-03-24 |
| CN1306394A (zh) | 2001-08-01 |
| US6630569B1 (en) | 2003-10-07 |
| PT1089625E (pt) | 2003-04-30 |
| JP4404484B2 (ja) | 2010-01-27 |
| CA2336129C (en) | 2008-12-02 |
| AU751711B2 (en) | 2002-08-22 |
| ATE229269T1 (de) | 2002-12-15 |
| DE59903759D1 (de) | 2003-01-23 |
| BR9912199A (pt) | 2001-04-10 |
| EP1089625A1 (de) | 2001-04-11 |
| DE19828043A1 (de) | 1999-12-30 |
| KR20010043938A (ko) | 2001-05-25 |
| AU4607899A (en) | 2000-01-10 |
| HUP0102808A3 (en) | 2002-12-28 |
| CA2336129A1 (en) | 1999-12-29 |
| HUP0102808A2 (hu) | 2001-11-28 |
| JP2002518415A (ja) | 2002-06-25 |
| EP1089625B1 (de) | 2002-12-11 |
| NZ509105A (en) | 2002-12-20 |
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