HUP0102099A3 - Substituted 2-oxo-alkanoic acid-[2-(indol-3-yl)ethyl]amides, process for producing them and pharmaceutical compositions containing them - Google Patents
Substituted 2-oxo-alkanoic acid-[2-(indol-3-yl)ethyl]amides, process for producing them and pharmaceutical compositions containing themInfo
- Publication number
- HUP0102099A3 HUP0102099A3 HU0102099A HUP0102099A HUP0102099A3 HU P0102099 A3 HUP0102099 A3 HU P0102099A3 HU 0102099 A HU0102099 A HU 0102099A HU P0102099 A HUP0102099 A HU P0102099A HU P0102099 A3 HUP0102099 A3 HU P0102099A3
- Authority
- HU
- Hungary
- Prior art keywords
- indol
- oxo
- amides
- ethyl
- substituted
- Prior art date
Links
- 150000001408 amides Chemical class 0.000 title 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19816780A DE19816780A1 (de) | 1998-04-16 | 1998-04-16 | Substituierte 2-Oxo-alkansäure-[2-(indol-3-yl)-ethyl]amide |
PCT/EP1999/002302 WO1999054301A1 (de) | 1998-04-16 | 1999-04-03 | Substituierte 2-oxo-alkansäure-[2-(indol-3-yl)-ethyl]amide |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP0102099A2 HUP0102099A2 (hu) | 2001-11-28 |
HUP0102099A3 true HUP0102099A3 (en) | 2001-12-28 |
Family
ID=7864659
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU0102099A HUP0102099A3 (en) | 1998-04-16 | 1999-04-03 | Substituted 2-oxo-alkanoic acid-[2-(indol-3-yl)ethyl]amides, process for producing them and pharmaceutical compositions containing them |
Country Status (11)
Country | Link |
---|---|
US (1) | US6255335B1 (hu) |
EP (1) | EP1071664A1 (hu) |
JP (1) | JP2002512226A (hu) |
KR (1) | KR20010052236A (hu) |
CN (1) | CN1297437A (hu) |
AU (1) | AU752273B2 (hu) |
BR (1) | BR9909692A (hu) |
CA (1) | CA2328875A1 (hu) |
DE (1) | DE19816780A1 (hu) |
HU (1) | HUP0102099A3 (hu) |
WO (1) | WO1999054301A1 (hu) |
Families Citing this family (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE0102764D0 (sv) * | 2001-08-17 | 2001-08-17 | Astrazeneca Ab | Compounds |
GB0226930D0 (en) | 2002-11-19 | 2002-12-24 | Astrazeneca Ab | Chemical compounds |
KR20070007103A (ko) * | 2004-02-18 | 2007-01-12 | 아스트라제네카 아베 | 벤즈아미드 유도체 및 이의 글루코키나아제 활성화제로서의용도 |
JP2007523905A (ja) * | 2004-02-18 | 2007-08-23 | アストラゼネカ アクチボラグ | 化合物 |
TW200600086A (en) | 2004-06-05 | 2006-01-01 | Astrazeneca Ab | Chemical compound |
CA2581619A1 (en) * | 2004-10-16 | 2006-04-20 | Astrazeneca Ab | Process for making phenoxy benzamide compounds |
JP2008542247A (ja) * | 2005-05-24 | 2008-11-27 | アストラゼネカ アクチボラグ | グルコキナーゼモジュレーターとしての2−フェニル置換イミダゾール[4,5b]ピリジン/ピラジンおよびプリン誘導体 |
TW200714597A (en) * | 2005-05-27 | 2007-04-16 | Astrazeneca Ab | Chemical compounds |
US20080234273A1 (en) * | 2005-07-09 | 2008-09-25 | Mckerrecher Darren | Heteroaryl Benzamide Derivatives for Use as Glk Activators in the Treatment of Diabetes |
JP4651714B2 (ja) * | 2005-07-09 | 2011-03-16 | アストラゼネカ アクチボラグ | 糖尿病の治療においてglk活性化剤として使用するためのヘテロアリールベンズアミド誘導体 |
JP2009500442A (ja) * | 2005-07-09 | 2009-01-08 | アストラゼネカ アクチボラグ | 2型糖尿病を処置するためのグルコキナーゼのモジュレーターとしての2−ヘテロシクリルオキシベンゾイルアミノヘテロシクリル化合物 |
US9202182B2 (en) * | 2005-08-11 | 2015-12-01 | International Business Machines Corporation | Method and system for analyzing business architecture |
TW200738621A (en) * | 2005-11-28 | 2007-10-16 | Astrazeneca Ab | Chemical process |
TW200825063A (en) * | 2006-10-23 | 2008-06-16 | Astrazeneca Ab | Chemical compounds |
TW200825060A (en) * | 2006-10-26 | 2008-06-16 | Astrazeneca Ab | Chemical compounds |
UY30822A1 (es) * | 2006-12-21 | 2008-07-31 | Astrazeneca Ab | Fnueva forma cristalina de 3-{[5-azetidin-1-ylcabonyl)pyrazin-2-yl]oxy}-5-[1-methylethyloxy]-n-1h-pyrazol-3-ylbenzamida, composiciones conteniéndola, procesos de preparacion y aplicaciones |
BRPI0917589A2 (pt) | 2008-08-04 | 2015-11-17 | Astrazeneca Ab | composto, composição farmacêutica, uso de um composto, método para tratar doenças, processo, combinação farmacêutica, e, reação de metiloxirano-2-carboxilato (ix) com um álcool roh |
GB0902406D0 (en) * | 2009-02-13 | 2009-04-01 | Astrazeneca Ab | Crystalline polymorphic form |
GB0902434D0 (en) * | 2009-02-13 | 2009-04-01 | Astrazeneca Ab | Chemical process |
WO2010116176A1 (en) * | 2009-04-09 | 2010-10-14 | Astrazeneca Ab | Pyrazolo [4, 5-e] pyrimidine derivative and its use to treat diabetes and obesity |
WO2010116177A1 (en) | 2009-04-09 | 2010-10-14 | Astrazeneca Ab | A pyrazolo [4,5-e] pyrimidine derivative and its use to treat diabetes and obesity |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3217011A (en) | 1965-05-07 | 1965-11-09 | Sterling Drug Inc | 1-(indolyglyoxalyl)-piperidines |
US5569668A (en) | 1995-03-29 | 1996-10-29 | Webster; John M. | Indole derivatives with antibacterial and antimycotic properties |
-
1998
- 1998-04-16 DE DE19816780A patent/DE19816780A1/de not_active Withdrawn
-
1999
- 1999-03-03 US US09/673,155 patent/US6255335B1/en not_active Expired - Fee Related
- 1999-04-03 WO PCT/EP1999/002302 patent/WO1999054301A1/de not_active Application Discontinuation
- 1999-04-03 CN CN99805078A patent/CN1297437A/zh active Pending
- 1999-04-03 HU HU0102099A patent/HUP0102099A3/hu unknown
- 1999-04-03 KR KR1020007011057A patent/KR20010052236A/ko not_active Application Discontinuation
- 1999-04-03 JP JP2000544642A patent/JP2002512226A/ja active Pending
- 1999-04-03 CA CA002328875A patent/CA2328875A1/en not_active Abandoned
- 1999-04-03 EP EP99917958A patent/EP1071664A1/de not_active Withdrawn
- 1999-04-03 BR BR9909692-7A patent/BR9909692A/pt not_active IP Right Cessation
- 1999-04-03 AU AU36050/99A patent/AU752273B2/en not_active Ceased
Also Published As
Publication number | Publication date |
---|---|
EP1071664A1 (de) | 2001-01-31 |
JP2002512226A (ja) | 2002-04-23 |
WO1999054301A1 (de) | 1999-10-28 |
AU752273B2 (en) | 2002-09-12 |
US6255335B1 (en) | 2001-07-03 |
CA2328875A1 (en) | 1999-10-28 |
BR9909692A (pt) | 2000-12-19 |
DE19816780A1 (de) | 1999-10-21 |
AU3605099A (en) | 1999-11-08 |
HUP0102099A2 (hu) | 2001-11-28 |
CN1297437A (zh) | 2001-05-30 |
KR20010052236A (ko) | 2001-06-25 |
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