HUP0101041A2 - Fungicid hatású N-szulfonil és N-szulfinil-fenil-glicinamid-származékok, intermedierjeik, előállításuk és alkalmazásuk - Google Patents

Fungicid hatású N-szulfonil és N-szulfinil-fenil-glicinamid-származékok, intermedierjeik, előállításuk és alkalmazásuk

Info

Publication number
HUP0101041A2
HUP0101041A2 HU0101041A HUP0101041A HUP0101041A2 HU P0101041 A2 HUP0101041 A2 HU P0101041A2 HU 0101041 A HU0101041 A HU 0101041A HU P0101041 A HUP0101041 A HU P0101041A HU P0101041 A2 HUP0101041 A2 HU P0101041A2
Authority
HU
Hungary
Prior art keywords
phenylethyl
phenyl
sulfonylaminoacetamide
optionally substituted
group
Prior art date
Application number
HU0101041A
Other languages
English (en)
Inventor
André Jeanguenat
Martin Zeller
Original Assignee
Novartis Ag.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag. filed Critical Novartis Ag.
Publication of HUP0101041A2 publication Critical patent/HUP0101041A2/hu
Publication of HUP0101041A3 publication Critical patent/HUP0101041A3/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C307/00Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C307/04Diamides of sulfuric acids
    • C07C307/06Diamides of sulfuric acids having nitrogen atoms of the sulfamide groups bound to acyclic carbon atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N41/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom
    • A01N41/02Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom containing a sulfur-to-oxygen double bond
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N41/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom
    • A01N41/02Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom containing a sulfur-to-oxygen double bond
    • A01N41/04Sulfonic acids; Derivatives thereof
    • A01N41/06Sulfonic acid amides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/04Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C237/08Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated having the nitrogen atom of at least one of the carboxamide groups bound to an acyclic carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/03Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C311/06Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/62Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
    • C07C323/63Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/24Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/28Halogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/02Ortho- or ortho- and peri-condensed systems
    • C07C2603/04Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/18Fluorenes; Hydrogenated fluorenes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Furan Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Indole Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)

Abstract

A találmány tárgya (I) általános képletű, új a-aminosav-amidvegyületek valamint lehetséges izomerjeik, ezen izomerek keverékei. Aképletben n jelentése egész szám, melynek értéke 0 vagy 1; R1jelentése adott esetben szubsztituált alkil, alkenil, alkinil,cikloalkil, cikloalkil-alkil, aril- vagy aril-alkilcsoport; vagy NRaRbcsoport, ahol Ra és Rb jelentése egymástól függetlenül hidrogénatom,alkilcsoport, vagy együtt egy alkilén hidat képeznek; R2 jelentésehidrogénatom vagy alkilcsoport; R3 jelentése adott esetbenszubsztituált aril- vagy heteroarilcsoport; A jelentésealkiléncsoport; és B jelentése adott esetben szubsztituáltarilcsoport; a következő vegyületek kivételével 2-fenil-N-(1-fenil-etil)-2-(4-metil-fenil)-szulfonil-amino-acetamid 2-fenil-N-(1-fenil-etil)-2-(4-klór-fenil)-szulfonil-amino-acetamid, 2-fenil-N-(1-fenil-etil)-2-(4-nitro-Ifenil)-szulfonil-amino-acetamid, 2-fenil-N-(1-fenil-etil)-2-(4-metoxi-fenil)-szulfonil-amino-acetamid, 2-fenil-N-(1-fenil-etil)-2-(4-fluor-fenil)-szulfonil-amino-acetamid, 2-fenil-N-(1-fenil-etil)-2-fenil-szulfonil-amino-acetamid és 2-fenil-N-(1-fenil-etil)-2-metán-szulfonil-amino-acetamid. A találmány szerinti új vegyületeknövényeknél fitopatogén mikroorganizmusok, főként gombák okoztafertőzések ellen alkalmazhatók. A találmány magába foglalja a (VI)általános képletű - ahol R2, R3, A és B jelentése az előzőekbenmegadott - intermediereket és ezek előállítását is. Ó
HU0101041A 1998-02-27 1999-02-25 Fungicidal n-sulphonyl and n-sulphinyl phenylglycinamide, intermediates, preparation and use thereof HUP0101041A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9804265.8A GB9804265D0 (en) 1998-02-27 1998-02-27 Organic compounds
PCT/EP1999/001216 WO1999043644A1 (en) 1998-02-27 1999-02-25 N-sulphonyl and n-sulphinyl phenylglycinamide___________________

Publications (2)

Publication Number Publication Date
HUP0101041A2 true HUP0101041A2 (hu) 2001-07-30
HUP0101041A3 HUP0101041A3 (en) 2002-03-28

Family

ID=10827756

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0101041A HUP0101041A3 (en) 1998-02-27 1999-02-25 Fungicidal n-sulphonyl and n-sulphinyl phenylglycinamide, intermediates, preparation and use thereof

Country Status (21)

Country Link
US (1) US6391918B1 (hu)
EP (1) EP1071660B1 (hu)
JP (1) JP2002504536A (hu)
KR (1) KR100633719B1 (hu)
CN (1) CN1226284C (hu)
AR (1) AR018123A1 (hu)
AT (1) ATE231489T1 (hu)
AU (1) AU3030299A (hu)
BR (1) BR9909239B1 (hu)
CA (1) CA2320838A1 (hu)
CR (1) CR5971A (hu)
DE (1) DE69905027T2 (hu)
ES (1) ES2191422T3 (hu)
GB (1) GB9804265D0 (hu)
GT (1) GT199900024A (hu)
HU (1) HUP0101041A3 (hu)
PL (1) PL342620A1 (hu)
TR (1) TR200002485T2 (hu)
TW (1) TW583162B (hu)
WO (1) WO1999043644A1 (hu)
ZA (1) ZA991575B (hu)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9826649D0 (en) 1998-12-03 1999-01-27 Novartis Ag Organic compounds
GB0011944D0 (en) * 2000-05-17 2000-07-05 Novartis Ag Organic compounds
GB0022338D0 (en) * 2000-09-12 2000-10-25 Novartis Ag Organic Compounds
GB0320345D0 (en) 2003-08-29 2003-10-01 Syngenta Participations Ag Organic compounds
WO2005068416A1 (ja) * 2003-12-12 2005-07-28 Sumitomo Chemical Company, Limited アミド化合物及びそれを用いた植物病害の防除方法
JP2006298785A (ja) * 2005-04-18 2006-11-02 Mitsui Chemicals Inc ジアミン誘導体、その製造方法およびそれらを有効成分とする殺菌剤
GB0516705D0 (en) * 2005-08-15 2005-09-21 Syngenta Participations Ag Process
CN113649067B (zh) * 2021-08-13 2023-08-11 万华化学(四川)有限公司 一种有机光催化剂、制备方法及其在合成2,3,5-三甲基氢醌二酯中的应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0493683A1 (en) * 1990-12-20 1992-07-08 American Cyanamid Company Fungicidal amino acid amides
CA2186510A1 (en) 1994-05-04 1995-11-16 Martin Zeller N-sulphonyl and n-sulphinyl amino acid amides as microbiocides
ATE218539T1 (de) * 1997-02-25 2002-06-15 Syngenta Participations Ag N-sulphonyl- und n-sulphinylaminosaüreamide als microbiozide
US6221888B1 (en) * 1997-05-29 2001-04-24 Merck & Co., Inc. Sulfonamides as cell adhesion inhibitors

Also Published As

Publication number Publication date
PL342620A1 (en) 2001-06-18
CA2320838A1 (en) 1999-09-02
GT199900024A (es) 2000-08-18
BR9909239B1 (pt) 2010-07-13
ZA991575B (en) 1999-08-27
AR018123A1 (es) 2001-10-31
ES2191422T3 (es) 2003-09-01
ATE231489T1 (de) 2003-02-15
JP2002504536A (ja) 2002-02-12
US6391918B1 (en) 2002-05-21
WO1999043644A1 (en) 1999-09-02
EP1071660B1 (en) 2003-01-22
BR9909239A (pt) 2000-11-14
KR100633719B1 (ko) 2006-10-16
KR20010041345A (ko) 2001-05-15
CR5971A (es) 2000-01-05
HUP0101041A3 (en) 2002-03-28
TW583162B (en) 2004-04-11
CN1291973A (zh) 2001-04-18
DE69905027D1 (de) 2003-02-27
TR200002485T2 (tr) 2001-01-22
CN1226284C (zh) 2005-11-09
DE69905027T2 (de) 2003-10-09
GB9804265D0 (en) 1998-04-22
EP1071660A1 (en) 2001-01-31
AU3030299A (en) 1999-09-15

Similar Documents

Publication Publication Date Title
HUP0401478A2 (hu) Fungicid hatású pirazolil-karboxanilid-származékok
ATE211466T1 (de) Depsipeptide, herstellung und anwendung
HUP0203624A2 (hu) Fungicid hatású pirazolkarboxamidok és pirazoltioamidok, intermedierjeik, előállításuk és alkalmazásuk
HUP0001993A2 (hu) Fungicid hatású (trifluor-metil-alkil)-amino-triazol 0[1,5-a]pirimidin-származékok, előállításuk és alkalmazásuk
HUP9802578A2 (hu) Fenil-ecetsav-származékok, eljárás és intermedierek előállításukhoz, a vegyületeket hatóanyagként tartalmazó fungicid, inszekticid, arachnicid és nematocid készítmények és alkalmazásuk
HUP0100064A2 (hu) Amidszármazékot és klórtalonilt tartalmazó, szinergetikus fungicid kombináció és alkalmazása
ATE270817T1 (de) Fungizide
HUP0300080A2 (hu) Új malonsavszármazékok, eljárás előállításukra, ezek alkalmazása Xa faktor inhibitorként és ezeket tartalmazó gyógyszerkészítmények
HUP0004529A2 (hu) VLA-4 által mediált leukocita adhéziót gátló szulfonilezett dipeptid-származékok, ezeket tartalmazó gyógyászati készítmények, valamint alkalmazásuk
HUP0401293A2 (hu) Új dihidropteridinonok, eljárás előállításukra és alkalmazásuk gyógyszerként
HRP20070286T3 (en) Substituted diketopiperazines and their use as oxytocyn antagonists
HUP0303639A2 (hu) Új amlodipin-kamzilát és eljárás annak előállítására
HUP0105039A2 (hu) Fungicid hatású propargil-éter-származékok, előállításuk és alkalmazásuk
ATE268752T1 (de) Aralkyl-1,2-diaminen mit calcimimetischer wirkung und verfahren zu ihrer herstellung
HUP0101041A2 (hu) Fungicid hatású N-szulfonil és N-szulfinil-fenil-glicinamid-származékok, intermedierjeik, előállításuk és alkalmazásuk
ATE18201T1 (de) Amide mit pharmakologischer wirkung, herstellung und diese verbindungen enthaltende mittel und verwendung.
MXPA04003729A (es) Compuestos de 4-imidazolin-2-ona.
HUP0004588A2 (hu) Szubsztituált 1,2,3,4,5,6-hexahidro-2,6-metano-3-benzazocin-10-ol-származékok, eljárás előállításukra és alkalmazásuk gyógyszerként, valamint a vegyületeket tartalmazó gyógyszerkészítmények
ATE173252T1 (de) Arylmorpholine, herstellung und verwendung
DK1628968T3 (da) 4-imidazolin-2-on-forbindelser
HUP0402544A2 (hu) Kompozíció elektrolit oldathoz és eljárás az előállítására
IE40942B1 (en) Novel n-sulphenylated oxime-carbamates and their use as insecticides, acaricides and nematicides
DE59005674D1 (de) Cyclohexenonverbindungen, Verfahren zu ihrer Herstellung sowie ihre Verwendung als Herbizide oder das Pflanzenwachstum regulierende Mittel.
HUP0105111A1 (hu) 2,5-Helyettesített benzolszulfonilkarbamid- és tiokarbamidszármazékok, eljárás előállításukra, alkalmazásuk, valamint e vegyületeket tartalmazó gyógyászati készítmények
ES8204721A1 (es) Un procedimiento para preparar derivados de halofenil-piri- dilalilamina