BR9909239A - N-sulfonil e n-sulfinil fenilglicinamida - Google Patents

N-sulfonil e n-sulfinil fenilglicinamida

Info

Publication number
BR9909239A
BR9909239A BR9909239-5A BR9909239A BR9909239A BR 9909239 A BR9909239 A BR 9909239A BR 9909239 A BR9909239 A BR 9909239A BR 9909239 A BR9909239 A BR 9909239A
Authority
BR
Brazil
Prior art keywords
phenyl
acetamide
ethyl
sulfonylamino
optionally substituted
Prior art date
Application number
BR9909239-5A
Other languages
English (en)
Other versions
BR9909239B1 (pt
Inventor
Andre Jeanguenat
Martin Zeller
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR9909239A publication Critical patent/BR9909239A/pt
Publication of BR9909239B1 publication Critical patent/BR9909239B1/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N41/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom
    • A01N41/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom containing a sulfur-to-oxygen double bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N41/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom
    • A01N41/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom containing a sulfur-to-oxygen double bond
    • A01N41/04—Sulfonic acids; Derivatives thereof
    • A01N41/06—Sulfonic acid amides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/04—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C237/08—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated having the nitrogen atom of at least one of the carboxamide groups bound to an acyclic carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C307/00—Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C307/04—Diamides of sulfuric acids
    • C07C307/06—Diamides of sulfuric acids having nitrogen atoms of the sulfamide groups bound to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/03—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C311/06—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/62—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
    • C07C323/63—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/28—Halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/18—Fluorenes; Hydrogenated fluorenes

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Furan Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Indole Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)

Abstract

Patente de Invenção: <B>"N-SULFONIL E N-SULFINIL FENILGLICINAMIDA"<D>. Novas amidas de <244>-aminoácido da fórmula I: copiar fórmula da página 70 bem como todos os isómeros e misturas possíveis de isómeros dos mesmos, em que os substituintes são definidos como segue: n é o número zero ou um; R~ 1~ é alquila, alquenila, alquinila, cicloalquila, cicloalquilalquila, arila ou aralquila opcionalmente substituída; ou um grupo NR~ a~R~ b~ em que R~ a~ e R~ b~ são, cada um, independentemente um do outro, hidrogênio, alquila ou juntos formam uma ponte de alquileno; R~ 2~ é hidrogênio ou alquila; R~ 3~ é arila ou heteroarila opcionalmente substituída; A é alquileno; e B é arila opcionalmente substituída; com exceção dos seguintes compostos: 2-fenil-N-(1-fenil-etil)-2-(metilfenil)-sulfonilamino-acetamida, 2-fenil-N-(1-fenil-etil)-2-(4-clorofenil)-sulfonilamino-acetamida, 2-fenil-N-(1-fenil-etil)-2-(4-nitrofenil)-sulfonilamino-acetamida, 2-fenil-N-(1-fenil-etil)-2-(4-metoxifenil)-sulfonilamino-acetamida, 2-fenil-N-(1-fenil-etil)-2-(4-fluorofenil)-sulfonilamino-acetamida, 2-fenil-N-(1-fenil-etil)-2-fenil-sulfonilamino-acetamida e 2-fenil-N-(1-fenil-etil)-2-metano-sulfonilamino-acetamida. Os novos compostos possuem propriedades protetoras da planta e são adequados para a proteção das plantas contra infestações por microorganismos fitopatogênicos, em particular fungos.
BRPI9909239-5A 1998-02-27 1999-02-25 composto e processo para sua preparação, intermediário e processo para sua preparação, bem como método e composição para controle e prevenção de infestação de plantas por microorganismos. BR9909239B1 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9804265.8A GB9804265D0 (en) 1998-02-27 1998-02-27 Organic compounds
PCT/EP1999/001216 WO1999043644A1 (en) 1998-02-27 1999-02-25 N-sulphonyl and n-sulphinyl phenylglycinamide___________________

Publications (2)

Publication Number Publication Date
BR9909239A true BR9909239A (pt) 2000-11-14
BR9909239B1 BR9909239B1 (pt) 2010-07-13

Family

ID=10827756

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9909239-5A BR9909239B1 (pt) 1998-02-27 1999-02-25 composto e processo para sua preparação, intermediário e processo para sua preparação, bem como método e composição para controle e prevenção de infestação de plantas por microorganismos.

Country Status (21)

Country Link
US (1) US6391918B1 (pt)
EP (1) EP1071660B1 (pt)
JP (1) JP2002504536A (pt)
KR (1) KR100633719B1 (pt)
CN (1) CN1226284C (pt)
AR (1) AR018123A1 (pt)
AT (1) ATE231489T1 (pt)
AU (1) AU3030299A (pt)
BR (1) BR9909239B1 (pt)
CA (1) CA2320838A1 (pt)
CR (1) CR5971A (pt)
DE (1) DE69905027T2 (pt)
ES (1) ES2191422T3 (pt)
GB (1) GB9804265D0 (pt)
GT (1) GT199900024A (pt)
HU (1) HUP0101041A3 (pt)
PL (1) PL342620A1 (pt)
TR (1) TR200002485T2 (pt)
TW (1) TW583162B (pt)
WO (1) WO1999043644A1 (pt)
ZA (1) ZA991575B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9826649D0 (en) 1998-12-03 1999-01-27 Novartis Ag Organic compounds
GB0011944D0 (en) * 2000-05-17 2000-07-05 Novartis Ag Organic compounds
GB0022338D0 (en) * 2000-09-12 2000-10-25 Novartis Ag Organic Compounds
GB0320345D0 (en) 2003-08-29 2003-10-01 Syngenta Participations Ag Organic compounds
WO2005068416A1 (ja) * 2003-12-12 2005-07-28 Sumitomo Chemical Company, Limited アミド化合物及びそれを用いた植物病害の防除方法
JP2006298785A (ja) * 2005-04-18 2006-11-02 Mitsui Chemicals Inc ジアミン誘導体、その製造方法およびそれらを有効成分とする殺菌剤
GB0516705D0 (en) * 2005-08-15 2005-09-21 Syngenta Participations Ag Process
CN113649067B (zh) * 2021-08-13 2023-08-11 万华化学(四川)有限公司 一种有机光催化剂、制备方法及其在合成2,3,5-三甲基氢醌二酯中的应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0493683A1 (en) * 1990-12-20 1992-07-08 American Cyanamid Company Fungicidal amino acid amides
JPH10504522A (ja) * 1994-05-04 1998-05-06 ノバルティス アクチエンゲゼルシャフト 殺微生物剤としてのｎ−スルホニルおよびｎ−スルフィニルアミノ酸アミド
JP2001513095A (ja) * 1997-02-25 2001-08-28 ノバルティス アクチェンゲゼルシャフト 殺微生物剤としてのｎ−スルホニル及びｎ−スルフィニルアミノ酸アミド
US6221888B1 (en) * 1997-05-29 2001-04-24 Merck & Co., Inc. Sulfonamides as cell adhesion inhibitors

Also Published As

Publication number Publication date
US6391918B1 (en) 2002-05-21
CN1226284C (zh) 2005-11-09
WO1999043644A1 (en) 1999-09-02
CR5971A (es) 2000-01-05
EP1071660B1 (en) 2003-01-22
HUP0101041A3 (en) 2002-03-28
AR018123A1 (es) 2001-10-31
AU3030299A (en) 1999-09-15
ATE231489T1 (de) 2003-02-15
GT199900024A (es) 2000-08-18
ES2191422T3 (es) 2003-09-01
TR200002485T2 (tr) 2001-01-22
KR100633719B1 (ko) 2006-10-16
TW583162B (en) 2004-04-11
JP2002504536A (ja) 2002-02-12
KR20010041345A (ko) 2001-05-15
PL342620A1 (en) 2001-06-18
GB9804265D0 (en) 1998-04-22
CN1291973A (zh) 2001-04-18
HUP0101041A2 (hu) 2001-07-30
EP1071660A1 (en) 2001-01-31
ZA991575B (en) 1999-08-27
BR9909239B1 (pt) 2010-07-13
DE69905027T2 (de) 2003-10-09
DE69905027D1 (de) 2003-02-27
CA2320838A1 (en) 1999-09-02

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Legal Events

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B25A Requested transfer of rights approved

Owner name: SYNGENTA PARTICIPATIONS AG (CH)

Free format text: TRANSFERIDO DE : NOVARTIS AG (NOVARTIS SA) (NOVARTIS INC.)

B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 13/07/2010, OBSERVADAS AS CONDICOES LEGAIS.

B24H Lapse because of non-payment of annual fees (definitively: art 78 iv lpi)
B24F Patent annual fee: publication cancelled

Free format text: ANULADA A PUBLICACAO CODIGO 24.8 NA RPI NO 2259 DE 22/04/2014 POR TER SIDO INDEVIDA.

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

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Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2607 DE 22-12-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.