HUE066520T2 - Eljárás 5-bróm-2-(3-klór-piridin-2-il)-2H-pirazol-3-karbonsav szintézis közttermékének elõállítására - Google Patents
Eljárás 5-bróm-2-(3-klór-piridin-2-il)-2H-pirazol-3-karbonsav szintézis közttermékének elõállításáraInfo
- Publication number
- HUE066520T2 HUE066520T2 HUE22161905A HUE22161905A HUE066520T2 HU E066520 T2 HUE066520 T2 HU E066520T2 HU E22161905 A HUE22161905 A HU E22161905A HU E22161905 A HUE22161905 A HU E22161905A HU E066520 T2 HUE066520 T2 HU E066520T2
- Authority
- HU
- Hungary
- Prior art keywords
- pyrazole
- pyridin
- bromo
- chloro
- synthesis
- Prior art date
Links
- FORBXGROTPOMEH-UHFFFAOYSA-N 5-bromo-2-(3-chloropyridin-2-yl)pyrazole-3-carboxylic acid Chemical compound OC(=O)C1=CC(Br)=NN1C1=NC=CC=C1Cl FORBXGROTPOMEH-UHFFFAOYSA-N 0.000 title 1
- 230000015572 biosynthetic process Effects 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
- 238000003786 synthesis reaction Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962916840P | 2019-10-18 | 2019-10-18 | |
US202062982248P | 2020-02-27 | 2020-02-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
HUE066520T2 true HUE066520T2 (hu) | 2024-08-28 |
Family
ID=73198483
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HUE20804069A HUE062047T2 (hu) | 2019-10-18 | 2020-10-16 | Eljárás 5-bróm-2-(3-klór-piridin-2-il)-2H-pirazol-3-karbonsav elõállítására |
HUE20804381A HUE062237T2 (hu) | 2019-10-18 | 2020-10-16 | Eljárások 5-bróm-2-(3-klór-piridin-2-il)-2H-pirazol-3-karbonsav elõállítására |
HUE22161905A HUE066520T2 (hu) | 2019-10-18 | 2020-10-16 | Eljárás 5-bróm-2-(3-klór-piridin-2-il)-2H-pirazol-3-karbonsav szintézis közttermékének elõállítására |
Family Applications Before (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HUE20804069A HUE062047T2 (hu) | 2019-10-18 | 2020-10-16 | Eljárás 5-bróm-2-(3-klór-piridin-2-il)-2H-pirazol-3-karbonsav elõállítására |
HUE20804381A HUE062237T2 (hu) | 2019-10-18 | 2020-10-16 | Eljárások 5-bróm-2-(3-klór-piridin-2-il)-2H-pirazol-3-karbonsav elõállítására |
Country Status (16)
Country | Link |
---|---|
US (2) | US20220396560A1 (hu) |
EP (5) | EP3976591B1 (hu) |
JP (2) | JP2022552273A (hu) |
KR (2) | KR20220086612A (hu) |
CN (2) | CN114650987B (hu) |
AU (2) | AU2020366037A1 (hu) |
BR (2) | BR112022007102A2 (hu) |
HU (3) | HUE062047T2 (hu) |
IL (5) | IL294551B2 (hu) |
MA (2) | MA56053A (hu) |
MX (2) | MX2022004627A (hu) |
PL (3) | PL3976589T3 (hu) |
TW (2) | TW202128631A (hu) |
UY (1) | UY38925A (hu) |
WO (2) | WO2021076835A1 (hu) |
ZA (2) | ZA202204277B (hu) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX2022004636A (es) * | 2019-10-18 | 2022-06-08 | Fmc Corp | Metodos para la preparacion del acido 5-bromo-2-(3-cloropiridin-2- il)-2h-pirazol-3-carboxilico. |
CN115557931B (zh) * | 2022-10-20 | 2024-05-14 | 浙江新安化工集团股份有限公司 | 一种3-溴-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酸的合成方法 |
Family Cites Families (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2060816C3 (de) * | 1970-12-10 | 1980-09-04 | Merck Patent Gmbh, 6100 Darmstadt | 4-Phenylpiperidinderivate Verfahren zu ihrer Herstellung und pharmazeutische Zubereitungen enthaltend diese Verbindungen |
UA81791C2 (uk) * | 2003-01-28 | 2008-02-11 | Е.І. Дю Пон Дэ Нэмур Энд Компани | Ціаноантраніламідні сполуки, композиція та спосіб регулювання кількості шкідників |
PE20060285A1 (es) * | 2004-03-30 | 2006-05-08 | Aventis Pharma Inc | Piridonas sustituidas como inhibidores de pol(adp-ribosa)-polimerasa (parp) |
MY140912A (en) * | 2004-07-26 | 2010-01-29 | Du Pont | Mixtures of anthranilamide invertebrate pest control agents |
US7087755B1 (en) * | 2004-11-12 | 2006-08-08 | Frontier Scientific, Inc. | Substituted pyridines |
MX2009006266A (es) * | 2006-12-13 | 2009-06-22 | Pfizer Prod Inc | Procedimientos de preparacion de 3-(4-(2,4-difluorobenciloxi)-3-br omo-6-metil-2-oxopiridin-1 (2h)-il)-n,4-dimetilbenzamida. |
CL2008000979A1 (es) * | 2007-04-11 | 2008-10-17 | Sumitomo Chemical Co | Proceso para producir un compuesto derivado de 2-piridin-2-il-2h-pirazol-3-fenilamida; compuestos intermediarios; el compuesto en si; composicion plaguicida que contiene a dicho compuesto; uso de dicho compuesto como plaguicida; y metodo para control |
JP2008280340A (ja) * | 2007-04-12 | 2008-11-20 | Sumitomo Chemical Co Ltd | ヒドラジド化合物及びそれを含有する有害節足動物防除剤 |
JP2009023991A (ja) * | 2007-06-20 | 2009-02-05 | Ishihara Sangyo Kaisha Ltd | アントラニルアミド系化合物の製造方法 |
CN102746327A (zh) * | 2007-08-14 | 2012-10-24 | 住友化学株式会社 | 肼化合物的制造方法、以及肼化合物的制造中间体及其制造方法 |
TW201245155A (en) * | 2010-09-01 | 2012-11-16 | Du Pont | Fungicidal pyrazoles |
CN102651485B (zh) * | 2011-02-28 | 2016-03-30 | 丰田自动车株式会社 | 可充镁电池、电解液在可充镁电池中的应用、以及用于可充镁电池的电解液 |
US9475812B2 (en) * | 2011-06-04 | 2016-10-25 | Xuanzhu Pharma Co., Ltd. | Pyridonaphthyridine type dual PI3K and mTOR inhibitor and its preparation and use |
WO2013105100A1 (en) * | 2012-01-09 | 2013-07-18 | Symed Labs Limited | Processes for the preparation of 5-chloro-n-({(5s)-2-oxo-3-[4-(3-oxo-4-morpholinyl)phenyl]-1,3-oxazolidin-5-yl}methyl)-2-thiophene-carboxamide and intermediates thereof |
CN105669643A (zh) * | 2013-12-05 | 2016-06-15 | 江西天人生态股份有限公司 | 一类基于鱼泥丁受体的邻甲酰氨基苯甲酰胺衍生物及其制备方法和用途 |
EA032581B1 (ru) * | 2014-04-14 | 2019-06-28 | Грюненталь Гмбх | Гетероарилзамещенные гетероциклилсульфоны |
TW201726128A (zh) * | 2015-10-08 | 2017-08-01 | 歌林達有限公司 | 經吡唑基取代之四氫哌喃基碸 |
JP2018534283A (ja) * | 2015-10-16 | 2018-11-22 | ウィリアム マーシュ ライス ユニバーシティWilliam Marsh Rice University | エポシロン類似体、合成方法、処置方法、およびその薬物結合体 |
ES2882526T3 (es) * | 2016-12-21 | 2021-12-02 | Bayer Cropscience Ag | Procedimiento para la preparación de un derivado de N-¬2-(2-piridinil)etil|carboxamida |
GB201721969D0 (en) * | 2017-12-27 | 2018-02-07 | Bp Oil Int | Methods for preparing fuel additives |
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2020
- 2020-10-16 PL PL20804069.1T patent/PL3976589T3/pl unknown
- 2020-10-16 US US17/769,810 patent/US20220396560A1/en active Pending
- 2020-10-16 HU HUE20804069A patent/HUE062047T2/hu unknown
- 2020-10-16 US US17/769,787 patent/US20220259178A1/en active Pending
- 2020-10-16 HU HUE20804381A patent/HUE062237T2/hu unknown
- 2020-10-16 EP EP20804381.0A patent/EP3976591B1/en active Active
- 2020-10-16 MA MA056053A patent/MA56053A/fr unknown
- 2020-10-16 UY UY0001038925A patent/UY38925A/es unknown
- 2020-10-16 CN CN202080072845.5A patent/CN114650987B/zh active Active
- 2020-10-16 AU AU2020366037A patent/AU2020366037A1/en active Pending
- 2020-10-16 JP JP2022521266A patent/JP2022552273A/ja active Pending
- 2020-10-16 EP EP20804069.1A patent/EP3976589B1/en active Active
- 2020-10-16 IL IL294551A patent/IL294551B2/en unknown
- 2020-10-16 WO PCT/US2020/055888 patent/WO2021076835A1/en unknown
- 2020-10-16 PL PL20804381.0T patent/PL3976591T3/pl unknown
- 2020-10-16 MX MX2022004627A patent/MX2022004627A/es unknown
- 2020-10-16 AU AU2020366212A patent/AU2020366212A1/en active Pending
- 2020-10-16 IL IL291939A patent/IL291939B2/en unknown
- 2020-10-16 KR KR1020227016245A patent/KR20220086612A/ko active Search and Examination
- 2020-10-16 TW TW109135805A patent/TW202128631A/zh unknown
- 2020-10-16 MA MA056055A patent/MA56055A/fr unknown
- 2020-10-16 CN CN202080072852.5A patent/CN114641471A/zh active Pending
- 2020-10-16 PL PL22161905.9T patent/PL4043451T3/pl unknown
- 2020-10-16 BR BR112022007102A patent/BR112022007102A2/pt unknown
- 2020-10-16 BR BR112022007215A patent/BR112022007215A2/pt unknown
- 2020-10-16 HU HUE22161905A patent/HUE066520T2/hu unknown
- 2020-10-16 IL IL299818A patent/IL299818B1/en unknown
- 2020-10-16 JP JP2022521265A patent/JP2022552272A/ja active Pending
- 2020-10-16 MX MX2022004631A patent/MX2022004631A/es unknown
- 2020-10-16 WO PCT/US2020/055897 patent/WO2021076839A1/en unknown
- 2020-10-16 KR KR1020227016372A patent/KR20220084347A/ko active Search and Examination
- 2020-10-16 EP EP23166843.5A patent/EP4219455A1/en active Pending
- 2020-10-16 TW TW109135811A patent/TW202116748A/zh unknown
- 2020-10-16 IL IL298694A patent/IL298694A/en unknown
- 2020-10-16 EP EP23168298.0A patent/EP4253380A3/en not_active Withdrawn
- 2020-10-16 EP EP22161905.9A patent/EP4043451B1/en active Active
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2022
- 2022-04-10 IL IL292090A patent/IL292090B2/en unknown
- 2022-04-14 ZA ZA2022/04277A patent/ZA202204277B/en unknown
- 2022-04-14 ZA ZA2022/04278A patent/ZA202204278B/en unknown
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