HUE058746T2 - Antiproliferációs vegyületek és felhasználásuk - Google Patents

Antiproliferációs vegyületek és felhasználásuk

Info

Publication number
HUE058746T2
HUE058746T2 HUE19726792A HUE19726792A HUE058746T2 HU E058746 T2 HUE058746 T2 HU E058746T2 HU E19726792 A HUE19726792 A HU E19726792A HU E19726792 A HUE19726792 A HU E19726792A HU E058746 T2 HUE058746 T2 HU E058746T2
Authority
HU
Hungary
Prior art keywords
antiproliferation
compounds
antiproliferation compounds
Prior art date
Application number
HUE19726792A
Other languages
English (en)
Hungarian (hu)
Inventor
Henry Yu
Michael Clark
Guy Bemis
Michael Boyd
Kishan Chandupatla
Philip Collier
Hongbo Deng
Huijun Dong
Warren Dorsch
Russell Hoover
Mac Johnson
Shashank Kulkarni
Marina Penney
Steven Ronkin
Darin Takemoto
Qing Tang
Nathan Waal
Tiansheng Wang
David J Lauffer
Pan Li
Original Assignee
Merck Patent Gmbh
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh, Vertex Pharma filed Critical Merck Patent Gmbh
Publication of HUE058746T2 publication Critical patent/HUE058746T2/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • C07D491/044Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/048Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10Spiro-condensed systems
    • C07D491/107Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10Spiro-condensed systems
    • C07D491/113Spiro-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
HUE19726792A 2018-04-24 2019-04-23 Antiproliferációs vegyületek és felhasználásuk HUE058746T2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201862661719P 2018-04-24 2018-04-24

Publications (1)

Publication Number Publication Date
HUE058746T2 true HUE058746T2 (hu) 2022-09-28

Family

ID=66655429

Family Applications (2)

Application Number Title Priority Date Filing Date
HUE19726792A HUE058746T2 (hu) 2018-04-24 2019-04-23 Antiproliferációs vegyületek és felhasználásuk
HUE22161962A HUE067936T2 (hu) 2018-04-24 2019-04-23 Proliferáció-gátló vegyületek és alkalmazásuk

Family Applications After (1)

Application Number Title Priority Date Filing Date
HUE22161962A HUE067936T2 (hu) 2018-04-24 2019-04-23 Proliferáció-gátló vegyületek és alkalmazásuk

Country Status (27)

Country Link
US (4) US10815225B2 (https=)
EP (2) EP3784666B1 (https=)
JP (2) JP7304892B2 (https=)
KR (1) KR102813581B1 (https=)
CN (1) CN112236428B (https=)
AR (1) AR114496A1 (https=)
AU (1) AU2019261308B2 (https=)
BR (1) BR112020020940A2 (https=)
CA (1) CA3098335A1 (https=)
CY (1) CY1125433T1 (https=)
DK (2) DK4043460T3 (https=)
ES (2) ES2987356T3 (https=)
FI (1) FI4043460T3 (https=)
HR (2) HRP20241163T1 (https=)
HU (2) HUE058746T2 (https=)
IL (2) IL278142B2 (https=)
LT (1) LT3784666T (https=)
MX (1) MX2020011089A (https=)
PL (2) PL3784666T3 (https=)
PT (2) PT3784666T (https=)
RS (1) RS63281B1 (https=)
SG (1) SG11202009500QA (https=)
SI (1) SI3784666T1 (https=)
SM (1) SMT202200308T1 (https=)
TW (1) TWI813673B (https=)
WO (1) WO2019209759A1 (https=)
ZA (1) ZA202006071B (https=)

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* Cited by examiner, † Cited by third party
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HRP20241163T1 (hr) 2018-04-24 2024-11-22 Merck Patent Gmbh Antiproliferacijski spojevi i njihova uporaba
WO2020010451A1 (en) * 2018-07-10 2020-01-16 Trillium Therapeutics Inc. Heteroaromatic-fused imidazolyl amides, compositions and uses thereof as sting agonists
WO2020236834A1 (en) * 2019-05-20 2020-11-26 Seshadri Raju Modified z stents for iliac vein stenting
CN118496197A (zh) 2019-12-20 2024-08-16 拜耳公司 取代的噻吩甲酰胺、噻吩甲酸及其衍生物
WO2024073502A1 (en) * 2022-09-28 2024-04-04 Accutar Biotechnology Inc. Heterocyclic compounds as e3 ligase inhibitors
TW202547516A (zh) * 2024-04-26 2025-12-16 大陸商正大天晴藥業集團股份有限公司 稠合雙環化合物及其用途

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PE20020354A1 (es) 2000-09-01 2002-06-12 Novartis Ag Compuestos de hidroxamato como inhibidores de histona-desacetilasa (hda)
DE60217322T2 (de) 2001-04-27 2007-10-04 Zenyaku Kogyo K.K. Heterocyclische verbindung und antitumormittel, das diese als wirkstoff enthält
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
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Also Published As

Publication number Publication date
EP3784666A1 (en) 2021-03-03
HRP20220710T1 (hr) 2022-07-22
DK4043460T3 (da) 2024-08-26
CN112236428A (zh) 2021-01-15
IL278142B2 (en) 2023-11-01
KR102813581B1 (ko) 2025-05-29
JP2023101824A (ja) 2023-07-21
IL278142B1 (en) 2023-07-01
US20230150993A1 (en) 2023-05-18
JP2021522242A (ja) 2021-08-30
SG11202009500QA (en) 2020-11-27
HRP20241163T1 (hr) 2024-11-22
ES2919572T3 (es) 2022-07-27
SI3784666T1 (sl) 2022-07-29
DK3784666T3 (da) 2022-06-20
FI4043460T3 (fi) 2025-05-09
IL301501B1 (en) 2024-06-01
CA3098335A1 (en) 2019-10-31
ES2987356T3 (es) 2024-11-14
EP4043460B1 (en) 2024-06-05
PT3784666T (pt) 2022-06-06
IL278142A (en) 2020-11-30
IL301501A (en) 2023-05-01
TWI813673B (zh) 2023-09-01
US20190322658A1 (en) 2019-10-24
RS63281B1 (sr) 2022-06-30
WO2019209759A1 (en) 2019-10-31
KR20210005151A (ko) 2021-01-13
BR112020020940A2 (pt) 2021-03-02
PL3784666T3 (pl) 2022-07-18
ZA202006071B (en) 2024-01-31
LT3784666T (lt) 2022-06-10
CN112236428B (zh) 2025-04-01
SMT202200308T1 (it) 2022-09-14
IL301501B2 (en) 2024-10-01
AU2019261308A1 (en) 2020-10-22
EP3784666B1 (en) 2022-03-16
US20250188070A1 (en) 2025-06-12
MX2020011089A (es) 2020-11-06
TW202012400A (zh) 2020-04-01
CY1125433T1 (el) 2025-05-09
US11440907B1 (en) 2022-09-13
AU2019261308B2 (en) 2022-09-08
PT4043460T (pt) 2024-09-10
EP4043460A1 (en) 2022-08-17
PL4043460T3 (pl) 2024-10-28
HUE067936T2 (hu) 2024-11-28
US12195453B2 (en) 2025-01-14
AR114496A1 (es) 2020-09-09
US10815225B2 (en) 2020-10-27
JP7304892B2 (ja) 2023-07-07

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