HUE033655T2 - Béta-2-adrenoceptor hatású benzotiazolon vegyület sók - Google Patents

Béta-2-adrenoceptor hatású benzotiazolon vegyület sók Download PDF

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Publication number
HUE033655T2
HUE033655T2 HUE13812075A HUE13812075A HUE033655T2 HU E033655 T2 HUE033655 T2 HU E033655T2 HU E13812075 A HUE13812075 A HU E13812075A HU E13812075 A HUE13812075 A HU E13812075A HU E033655 T2 HUE033655 T2 HU E033655T2
Authority
HU
Hungary
Prior art keywords
compound
butoxyphenyl
methylpropan
ylamino
thiazol
Prior art date
Application number
HUE13812075A
Other languages
English (en)
Inventor
Arnaud Grandeury
Nicola Tufilli
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=53386469&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUE033655(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of HUE033655T2 publication Critical patent/HUE033655T2/hu

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62Benzothiazoles
    • C07D277/68Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Claims (6)

  1. Βέϊ»-%~ΜΐΜ®ύψίΜ hMásd teizöiMoIoíiWf^iM sók SZABADALMI lOÉMYBObllíOL. L Az (^.)-7-(2^1 -(4-butoxifc.DÍI)-2-meUlpropán--2-i!aml-Kí.)-- DhkiroxicbI)-5--hidroxibenxoldltiazoi-^ÜID-öft aeetát só egy kristályos formáim
  2. 2. Az Ï. igénypont szerimi kristályos forma, melyet egy^îyap'rëôtgensttgfefûrÂf-rateiésminta lliillg a 8,8 ± 0,2A 16,4 ± 0,2*, 20,8 ± 0,2" énékek közűi kiválásion 2 théta (0) refrakciós szög értékekkel, CuK« sugárzás alkalmazásával mérve.
  3. 3 Gyógy ,verké\zitnten>, mely az L vagy 2, igénypontok bámtelylke szérinö vegyülei gyogyászattlaglatásos mennyiségit táBalmazza, egy vagy több |yögyákzátllag elfogadható; hordozóval egyitt,
  4. 4 Konibibáoiö, niely egy, az 1. mgy 2, igénypont szernüi vegyfo^ Cgy vagy több gvogydszatilag aktív kö-ágenst: ttóateaz.
  5. 5, Az I·.· vagy 2. igénypontok bármelyikémmmti vegyidet, gyógyszetkénktörténö aL katoazásra.
  6. 6, Az I. vagy 2. Igénypöbíok bátMélylke szerinti vegyülét, Izontsorvadásna betegségek kezelésében vagy megelőzésében való alkalntazlpa-: % A: 4 igénypont szerinti vegyüld, ahol az izomaorvadásos betegség a muscuiam dystrophia, használaton kívüliség okozta atrophia, cachexia vagy szarkopénia.
HUE13812075A 2012-08-30 2013-08-29 Béta-2-adrenoceptor hatású benzotiazolon vegyület sók HUE033655T2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IQ23912 2012-08-30

Publications (1)

Publication Number Publication Date
HUE033655T2 true HUE033655T2 (hu) 2017-12-28

Family

ID=53386469

Family Applications (1)

Application Number Title Priority Date Filing Date
HUE13812075A HUE033655T2 (hu) 2012-08-30 2013-08-29 Béta-2-adrenoceptor hatású benzotiazolon vegyület sók

Country Status (27)

Country Link
EP (2) EP2890687B1 (hu)
KR (1) KR20150047586A (hu)
CN (2) CN104736525B (hu)
BR (1) BR112015004127A2 (hu)
CA (1) CA2882877A1 (hu)
CL (1) CL2015000461A1 (hu)
CY (1) CY1120225T1 (hu)
DK (1) DK2890687T3 (hu)
EA (1) EA029946B1 (hu)
ES (1) ES2642003T3 (hu)
HK (1) HK1206015A1 (hu)
HR (1) HRP20171362T1 (hu)
HU (1) HUE033655T2 (hu)
IL (1) IL237382A0 (hu)
LT (1) LT2890687T (hu)
MA (1) MA37872A1 (hu)
MX (1) MX351741B (hu)
MY (1) MY169038A (hu)
NZ (1) NZ705319A (hu)
PE (1) PE20150465A1 (hu)
PL (1) PL2890687T3 (hu)
PT (1) PT2890687T (hu)
SA (1) SA515360076B1 (hu)
SG (2) SG11201501293PA (hu)
SI (1) SI2890687T1 (hu)
TN (1) TN2015000058A1 (hu)
WO (1) WO2014033654A1 (hu)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3192B1 (ar) * 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR040962A1 (es) 2002-08-09 2005-04-27 Novartis Ag Compuestos derivados de tiazol 1,3-2-ona, composicion farmaceutica y proceso de preparacion del compuesto
CA2514733A1 (en) 2003-02-28 2004-09-16 Transform Pharmaceuticals, Inc. Pharmaceutical co-crystal compositions of drugs such as carbamazepine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothiazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen
JP2007537187A (ja) 2004-05-13 2007-12-20 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 呼吸器疾患の治療においてβアゴニストとして使用するためのヒドロキシ置換ベンゾ縮合ヘテロ環化合物
GB0426164D0 (en) * 2004-11-29 2004-12-29 Novartis Ag Organic compounds
JO3192B1 (ar) * 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون
AU2014222362B2 (en) * 2013-02-28 2016-07-21 Novartis Ag Formulation comprising benzothiazolone compound

Also Published As

Publication number Publication date
EA201590452A1 (ru) 2015-07-30
MX2015002656A (es) 2015-05-20
HRP20171362T1 (hr) 2017-11-03
WO2014033654A1 (en) 2014-03-06
IL237382A0 (en) 2015-04-30
PL2890687T3 (pl) 2017-11-30
TN2015000058A1 (en) 2016-06-29
MX351741B (es) 2017-10-26
EP2890687A1 (en) 2015-07-08
KR20150047586A (ko) 2015-05-04
EP2890687B1 (en) 2017-06-28
HK1206015A1 (en) 2015-12-31
SA515360076B1 (ar) 2016-03-20
CY1120225T1 (el) 2018-12-12
PE20150465A1 (es) 2015-04-22
MY169038A (en) 2019-02-07
MA37872A1 (fr) 2018-07-31
BR112015004127A2 (pt) 2017-07-04
SG10201704377PA (en) 2017-06-29
CN104736525B (zh) 2016-08-24
EA029946B1 (ru) 2018-06-29
CL2015000461A1 (es) 2015-05-04
SG11201501293PA (en) 2015-03-30
ES2642003T3 (es) 2017-11-14
SI2890687T1 (sl) 2017-10-30
EP3243817A1 (en) 2017-11-15
CN104736525A (zh) 2015-06-24
LT2890687T (lt) 2017-09-11
NZ705319A (en) 2018-05-25
CA2882877A1 (en) 2014-03-06
PT2890687T (pt) 2017-10-05
DK2890687T3 (en) 2017-10-09
CN106146428A (zh) 2016-11-23

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