HU9402832D0 - Imidazol-4-yl-piperidine derivatives, process for producing them and pharmaceutical use of them - Google Patents

Imidazol-4-yl-piperidine derivatives, process for producing them and pharmaceutical use of them

Info

Publication number
HU9402832D0
HU9402832D0 HU9402832A HU9402832A HU9402832D0 HU 9402832 D0 HU9402832 D0 HU 9402832D0 HU 9402832 A HU9402832 A HU 9402832A HU 9402832 A HU9402832 A HU 9402832A HU 9402832 D0 HU9402832 D0 HU 9402832D0
Authority
HU
Hungary
Prior art keywords
imidazol
producing
pharmaceutical use
piperidine derivatives
piperidine
Prior art date
Application number
HU9402832A
Other languages
English (en)
Other versions
HUT71120A (en
Inventor
Samir Jegham
Gerard Defosse
Luc Even
Thomas Andrew Purcell
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of HU9402832D0 publication Critical patent/HU9402832D0/hu
Publication of HUT71120A publication Critical patent/HUT71120A/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HU9402832A 1993-10-04 1994-10-03 Imidazol-4-yl-piperidine derivatives, process for producing them and pharmaceutical compositions containing them HUT71120A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9311771A FR2710915B1 (fr) 1993-10-04 1993-10-04 Dérivés de pipéridine, leur préparation et leur utilisation en thérapeutique.

Publications (2)

Publication Number Publication Date
HU9402832D0 true HU9402832D0 (en) 1995-01-30
HUT71120A HUT71120A (en) 1995-11-28

Family

ID=9451496

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9402832A HUT71120A (en) 1993-10-04 1994-10-03 Imidazol-4-yl-piperidine derivatives, process for producing them and pharmaceutical compositions containing them

Country Status (18)

Country Link
US (1) US5589476A (hu)
EP (1) EP0646583A1 (hu)
JP (1) JPH07179466A (hu)
KR (1) KR950011435A (hu)
CN (1) CN1109471A (hu)
AU (1) AU7432994A (hu)
CA (1) CA2133491A1 (hu)
CZ (1) CZ241994A3 (hu)
FI (1) FI944600A (hu)
FR (1) FR2710915B1 (hu)
HU (1) HUT71120A (hu)
IL (1) IL111148A0 (hu)
NO (1) NO943682L (hu)
NZ (1) NZ264596A (hu)
PL (1) PL305288A1 (hu)
RU (1) RU94036003A (hu)
SK (1) SK119494A3 (hu)
ZA (1) ZA947710B (hu)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5500423A (en) * 1994-09-09 1996-03-19 Hoechst-Roussel Pharmaceuticals Inc. 5,6-dihydro-4H-imidazo[4,5,1-ij]quinolines
FR2731708B1 (fr) * 1995-03-13 1997-04-30 Synthelabo Derives de piperidine, leur procede de preparation et leur application en therapeutique
AU6921196A (en) * 1995-09-18 1997-04-09 Glaxo Group Limited 5-ht3 receptor antagonists for dyskinesia
FR2747678B1 (fr) * 1996-04-22 1998-05-22 Synthelabo Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique
FR2753196B1 (fr) * 1996-09-12 1998-10-23 Synthelabo Derives d'indazole tricyclique, leur preparation et leur application en therapeutique
NZ509832A (en) * 1998-08-21 2003-11-28 Novartis Ag New oral formulation for 5-HT4 agonists or antagonists
IT1303123B1 (it) 1998-10-13 2000-10-30 Rotta Research Lab Derivati basici di benz(e)isoindol-1-oni e pirrolo(3,4-c)chinolin-1-oni ad attivita' 5ht3 antagonista, loro preparazione ed
GB9918425D0 (en) * 1999-08-04 1999-10-06 Novartis Ag Organic compounds
FR2816619B1 (fr) * 2000-11-15 2003-01-31 Sanofi Synthelabo Derives de benzimidazole, leur preparation et leur application en therapeutique
ES2233671T3 (es) * 2000-08-08 2005-06-16 Sanofi-Aventis Derivados de benzimidazol, su preparacion y aplicacion en terapeutica.
FR2812878B1 (fr) * 2000-08-08 2002-10-11 Sanofi Synthelabo Derives de benzimidazole, leur preparation et leur application en therapeutique
FR2816942B1 (fr) * 2000-11-23 2003-05-09 Sanofi Synthelabo Derives de benzimidazole, leur preparation et leur application en therapeutique
FR2816941B1 (fr) * 2000-11-23 2003-01-31 Sanofi Synthelabo Derives de benzimidazole, leur preparation et leur application en therapeutique
US20040242635A1 (en) * 2001-03-30 2004-12-02 Painter Rachel J. Encapsulated dyes in cosmetic compositions
AU2003240742A1 (en) * 2002-06-07 2003-12-22 Altana Pharma Ag 4,5-dihydro-imidazo (4,5,1-ij) quinolin-6-ones derivatives and their use as poly (adp-ribosyl) transferase (parp) inhibitors
EA038494B1 (ru) 2013-03-15 2021-09-07 Инсайт Холдингс Корпорейшн Трициклические гетероциклы как ингибиторы белков бэт
US9290514B2 (en) 2013-07-08 2016-03-22 Incyte Holdings Corporation Tricyclic heterocycles as BET protein inhibitors
US9315501B2 (en) 2013-11-26 2016-04-19 Incyte Corporation Bicyclic heterocycles as BET protein inhibitors
WO2015081203A1 (en) 2013-11-26 2015-06-04 Incyte Corporation Bicyclic heterocycles as bet protein inhibitors
US9309246B2 (en) 2013-12-19 2016-04-12 Incyte Corporation Tricyclic heterocycles as BET protein inhibitors
SI3674302T1 (sl) 2014-04-23 2023-07-31 Incyte Holdings Corporation 1h-pirolo(2,3-c)piridin-7(6h)-oni in pirazolo(3,4-c)piridin-7(6h)-oni kot zaviralci proteinov bet
EP3194406B8 (en) 2014-09-15 2021-03-31 Incyte Corporation Tricyclic heterocycles for use as bet protein inhibitors
US20170121347A1 (en) 2015-10-29 2017-05-04 Incyte Corporation Amorphous solid form of a bet protein inhibitor
UA125476C2 (uk) 2016-06-20 2022-03-23 Інсайт Корпорейшн Спосіб отримання 2,2,4-триметил-8-(6-метил-7-оксо-6,7-дигідро-1н-піроло[2,3-c]піридин-4-іл)-6-(метилсульфоніл)-2н-бензо[b][1,4]оксазин-3(4н)-ону і проміжних сполук
US11833155B2 (en) 2020-06-03 2023-12-05 Incyte Corporation Combination therapy for treatment of myeloproliferative neoplasms

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4939138A (en) * 1988-12-29 1990-07-03 Sterling Drug Inc. 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines
FR2674855B1 (fr) * 1991-04-03 1994-01-14 Synthelabo Derives de piperidine, leur preparation et leur application en therapeutique.

Also Published As

Publication number Publication date
AU7432994A (en) 1995-04-13
RU94036003A (ru) 1996-08-10
ZA947710B (en) 1995-08-10
FR2710915B1 (fr) 1995-11-24
NO943682L (no) 1995-04-05
CN1109471A (zh) 1995-10-04
FI944600A (fi) 1995-04-05
IL111148A0 (en) 1994-12-29
FR2710915A1 (fr) 1995-04-14
SK119494A3 (en) 1995-05-10
PL305288A1 (en) 1995-04-18
NO943682D0 (no) 1994-10-03
JPH07179466A (ja) 1995-07-18
CA2133491A1 (en) 1995-04-05
NZ264596A (en) 1995-11-27
FI944600A0 (fi) 1994-10-03
US5589476A (en) 1996-12-31
KR950011435A (ko) 1995-05-15
HUT71120A (en) 1995-11-28
CZ241994A3 (en) 1995-04-12
EP0646583A1 (fr) 1995-04-05

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Legal Events

Date Code Title Description
DFC4 Cancellation of temporary protection due to refusal