HU9201254D0 - Rapamicine-carbamates and medical preparations containing them as active agents - Google Patents
Rapamicine-carbamates and medical preparations containing them as active agentsInfo
- Publication number
- HU9201254D0 HU9201254D0 HU9201254A HU9201254A HU9201254D0 HU 9201254 D0 HU9201254 D0 HU 9201254D0 HU 9201254 A HU9201254 A HU 9201254A HU 9201254 A HU9201254 A HU 9201254A HU 9201254 D0 HU9201254 D0 HU 9201254D0
- Authority
- HU
- Hungary
- Prior art keywords
- rapamicine
- carbamates
- active agents
- preparations containing
- medical preparations
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/08—Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Transplantation (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/686,728 US5118678A (en) | 1991-04-17 | 1991-04-17 | Carbamates of rapamycin |
US07/837,048 US5194447A (en) | 1992-02-18 | 1992-02-18 | Sulfonylcarbamates of rapamycin |
Publications (1)
Publication Number | Publication Date |
---|---|
HU9201254D0 true HU9201254D0 (en) | 1992-07-28 |
Family
ID=27103855
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU9201254A HU9201254D0 (en) | 1991-04-17 | 1992-04-13 | Rapamicine-carbamates and medical preparations containing them as active agents |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP0509795A2 (hu) |
JP (1) | JPH05112573A (hu) |
KR (1) | KR920019798A (hu) |
AU (1) | AU642592B2 (hu) |
CZ (1) | CZ117392A3 (hu) |
FI (1) | FI921595A (hu) |
HU (1) | HU9201254D0 (hu) |
IE (1) | IE921249A1 (hu) |
MX (1) | MX9201710A (hu) |
NO (1) | NO921449L (hu) |
NZ (1) | NZ242367A (hu) |
SK (1) | SK117392A3 (hu) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5776943A (en) * | 1991-05-14 | 1998-07-07 | American Home Products Corporation | Rapamycin metabolites |
US5118677A (en) * | 1991-05-20 | 1992-06-02 | American Home Products Corporation | Amide esters of rapamycin |
WO1993018043A1 (en) * | 1992-03-05 | 1993-09-16 | American Home Products Corporation | Novel rapamycin 42-sulfonates and 42-(n-carboalkoxy)sulfamates useful as immunosuppressive agents |
GB9307491D0 (en) * | 1993-04-08 | 1993-06-02 | Sandoz Ltd | Organic compounds |
CH686761A5 (de) | 1993-05-27 | 1996-06-28 | Sandoz Ag | Galenische Formulierungen. |
US5527907A (en) * | 1993-11-19 | 1996-06-18 | Abbott Laboratories | Macrolide immunomodulators |
JP4105761B2 (ja) * | 1993-11-19 | 2008-06-25 | アボット・ラボラトリーズ | ラパミシン(マクロライド)の半合成類似体免疫調節剤 |
US5362718A (en) | 1994-04-18 | 1994-11-08 | American Home Products Corporation | Rapamycin hydroxyesters |
US8124630B2 (en) | 1999-01-13 | 2012-02-28 | Bayer Healthcare Llc | ω-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors |
EP1158985B1 (en) | 1999-01-13 | 2011-12-28 | Bayer HealthCare LLC | OMEGA-CARBOXY ARYL SUBSTITUTED DIPHENYL UREAS AS p38 KINASE INHIBITORS |
PT1210350E (pt) * | 1999-08-18 | 2004-10-29 | Wyeth Corp | Esteres de sdz-rad soluveis em agua |
EP1478358B1 (en) | 2002-02-11 | 2013-07-03 | Bayer HealthCare LLC | Sorafenib tosylate for the treatment of diseases characterized by abnormal angiogenesis |
UY28213A1 (es) | 2003-02-28 | 2004-09-30 | Bayer Pharmaceuticals Corp | Nuevos derivados de cianopiridina útiles en el tratamiento de cáncer y otros trastornos. |
CA2526636C (en) | 2003-05-20 | 2012-10-02 | Bayer Pharmaceuticals Corporation | Diaryl ureas for diseases mediated by pdgfr |
CL2004001834A1 (es) | 2003-07-23 | 2005-06-03 | Bayer Pharmaceuticals Corp | Compuesto 4-{4-[3-(4-cloro-3-trifluorometilfenil)-ureido]-3-fluorofenoxi}-piridin-2-metilamida, inhibidor de la raf, vegfr, p38 y pdgfr quinasas, sus sales; composiicon farmaceutica; combinacion farmaceutica; y su uso para tratar trastornos hiperprol |
WO2005042567A1 (en) * | 2003-11-03 | 2005-05-12 | Altachem Pharma Ltd. | Rapamycin peptides conjugates: synthesis and uses thereof |
US8021849B2 (en) | 2004-11-05 | 2011-09-20 | Siemens Healthcare Diagnostics Inc. | Methods and kits for the determination of sirolimus in a sample |
US7241771B2 (en) | 2005-03-07 | 2007-07-10 | Wyeth | Oxepane isomer of 42-O-(2-hydroxy)ethyl-rapamycin |
US7189582B2 (en) | 2005-04-27 | 2007-03-13 | Dade Behring Inc. | Compositions and methods for detection of sirolimus |
SG11202107653RA (en) * | 2019-01-25 | 2021-08-30 | Nodthera Ltd | Carbamate derivatives and uses thereof |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4885171A (en) * | 1978-11-03 | 1989-12-05 | American Home Products Corporation | Use of rapamycin in treatment of certain tumors |
US4316885A (en) * | 1980-08-25 | 1982-02-23 | Ayerst, Mckenna And Harrison, Inc. | Acyl derivatives of rapamycin |
US4650803A (en) * | 1985-12-06 | 1987-03-17 | University Of Kansas | Prodrugs of rapamycin |
JPH05504944A (ja) * | 1989-08-18 | 1993-07-29 | 藤沢薬品工業株式会社 | 巨大環式化合物 |
PT98990A (pt) * | 1990-09-19 | 1992-08-31 | American Home Prod | Processo para a preparacao de esteres de acidos carboxilicos de rapamicina |
US5118677A (en) * | 1991-05-20 | 1992-06-02 | American Home Products Corporation | Amide esters of rapamycin |
-
1992
- 1992-04-10 FI FI921595A patent/FI921595A/fi unknown
- 1992-04-10 NO NO92921449A patent/NO921449L/no unknown
- 1992-04-10 JP JP4090825A patent/JPH05112573A/ja active Pending
- 1992-04-11 KR KR1019920006033A patent/KR920019798A/ko not_active Application Discontinuation
- 1992-04-13 MX MX9201710A patent/MX9201710A/es unknown
- 1992-04-13 HU HU9201254A patent/HU9201254D0/hu unknown
- 1992-04-14 AU AU14880/92A patent/AU642592B2/en not_active Ceased
- 1992-04-15 NZ NZ24236792A patent/NZ242367A/en unknown
- 1992-04-15 EP EP19920303401 patent/EP0509795A2/en not_active Withdrawn
- 1992-04-16 IE IE124992A patent/IE921249A1/en not_active Application Discontinuation
- 1992-04-16 SK SK1173-92A patent/SK117392A3/sk unknown
- 1992-04-16 CZ CS921173A patent/CZ117392A3/cs unknown
Also Published As
Publication number | Publication date |
---|---|
EP0509795A3 (hu) | 1994-03-23 |
NO921449D0 (no) | 1992-04-10 |
FI921595A (fi) | 1992-10-18 |
IE921249A1 (en) | 1992-10-21 |
AU1488092A (en) | 1992-10-22 |
NO921449L (no) | 1992-10-19 |
JPH05112573A (ja) | 1993-05-07 |
SK117392A3 (en) | 1995-04-12 |
EP0509795A2 (en) | 1992-10-21 |
CZ117392A3 (en) | 1993-09-15 |
MX9201710A (es) | 1993-01-01 |
KR920019798A (ko) | 1992-11-20 |
FI921595A0 (fi) | 1992-04-10 |
NZ242367A (en) | 1994-07-26 |
AU642592B2 (en) | 1993-10-21 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
HU9201254D0 (en) | Rapamicine-carbamates and medical preparations containing them as active agents | |
HU906229D0 (en) | Medical preparations | |
ZA897506B (en) | Fungicidally active preparations | |
HU906721D0 (en) | Methylene-diphosphonic acid derivatives and inflammation-preventing preparations containing them as active agents | |
EP0467218A3 (en) | Combinations of active agents for skin care | |
GB9125695D0 (en) | Medical preparations | |
HU00207A9 (en) | Sulfonanilide derivatives and medicine | |
AP9300555A0 (en) | Therapeutic agent and its use | |
HU904007D0 (en) | Medical preparations providing regulated active agent discharge and processes for the preparation thereof | |
HU9201364D0 (en) | Medical preparations contqining bafilomycin microlides | |
NZ227594A (en) | Human interleukin-1alpha and preparations thereof | |
CY1984A (en) | Pharmaceutical formulation containing penciclovir | |
HU9204072D0 (en) | Terazole derivatives and medical preparatives containing them | |
HU905823D0 (en) | Medical preparations | |
ZA939740B (en) | N-arylhydrazine derivatives as insecticidal and acaricidal agents | |
GB2249788B (en) | 3-amino-5-benzylidene-2-thioxo-thiazolidine-4-ones and cosmetic agents containing them | |
HU908294D0 (en) | Fungicide preparations containing pyridyl-cyclopropane as active agent and process for the preparation of the active agents | |
GB9302553D0 (en) | Pharmaceutical preparations and their manufacture and use | |
AU1447892A (en) | Pharmaceutical preparations for the therapy of tumors containing colchicine as the active principle and methods for the use of the same | |
EP0417632A3 (en) | 2-ethoxymethyl-5-hydroxy-gamma-pyrone and melanogenesis-inhibiting endermic preparation containing the same compound as active ingredient | |
HU9203050D0 (en) | Thieno-cyclopentanole-oximes and pharmaceutical preparatives containing them | |
GB9218709D0 (en) | Biologically active health formulation | |
GB9125761D0 (en) | Medical preparations | |
HU9202971D0 (en) | Hetero-polycyclic biocidical compounds and preparatives containing them as active substance | |
IL98276A0 (en) | Use of anaesthetic agents in the manufacture of pharmaceutical preparations for iontophoresis |