HRP20190730T1 - Spoj pirazola i njegova farmaceutska upotreba - Google Patents
Spoj pirazola i njegova farmaceutska upotreba Download PDFInfo
- Publication number
- HRP20190730T1 HRP20190730T1 HRP20190730TT HRP20190730T HRP20190730T1 HR P20190730 T1 HRP20190730 T1 HR P20190730T1 HR P20190730T T HRP20190730T T HR P20190730TT HR P20190730 T HRP20190730 T HR P20190730T HR P20190730 T1 HRP20190730 T1 HR P20190730T1
- Authority
- HR
- Croatia
- Prior art keywords
- alkyl group
- group
- groups
- alkoxy
- halogen
- Prior art date
Links
- -1 Pyrazole compound Chemical class 0.000 title 1
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 claims 55
- 125000000623 heterocyclic group Chemical group 0.000 claims 27
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 claims 26
- 229910052736 halogen Inorganic materials 0.000 claims 22
- 150000001875 compounds Chemical class 0.000 claims 21
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 20
- 150000003839 salts Chemical class 0.000 claims 19
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims 16
- 229910052799 carbon Inorganic materials 0.000 claims 16
- IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Substances N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 14
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims 10
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims 10
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 10
- 125000005842 heteroatom Chemical group 0.000 claims 10
- 229910052757 nitrogen Inorganic materials 0.000 claims 10
- 229910052760 oxygen Inorganic materials 0.000 claims 10
- 239000001301 oxygen Chemical group 0.000 claims 10
- 229910052717 sulfur Chemical group 0.000 claims 10
- 239000011593 sulfur Chemical group 0.000 claims 10
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 claims 9
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 claims 7
- 125000000041 C6-C10 aryl group Chemical group 0.000 claims 7
- 206010012601 diabetes mellitus Diseases 0.000 claims 7
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims 6
- 125000005843 halogen group Chemical group 0.000 claims 5
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 5
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 claims 4
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 claims 3
- 125000006719 (C6-C10) aryl (C1-C6) alkyl group Chemical group 0.000 claims 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 3
- 230000002265 prevention Effects 0.000 claims 3
- 125000001424 substituent group Chemical group 0.000 claims 3
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims 2
- 125000004648 C2-C8 alkenyl group Chemical group 0.000 claims 2
- 125000004414 alkyl thio group Chemical group 0.000 claims 2
- 125000004470 heterocyclooxy group Chemical group 0.000 claims 2
- 125000006625 (C3-C8) cycloalkyloxy group Chemical group 0.000 claims 1
- 125000004649 C2-C8 alkynyl group Chemical group 0.000 claims 1
- 108091006277 SLC5A1 Proteins 0.000 claims 1
- 102000058090 Sodium-Glucose Transporter 1 Human genes 0.000 claims 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 claims 1
- 125000005194 alkoxycarbonyloxy group Chemical group 0.000 claims 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 claims 1
- 239000003795 chemical substances by application Substances 0.000 claims 1
- 125000000392 cycloalkenyl group Chemical group 0.000 claims 1
- 239000003112 inhibitor Substances 0.000 claims 1
- 239000000825 pharmaceutical preparation Substances 0.000 claims 1
- 229920006395 saturated elastomer Polymers 0.000 claims 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2011188121 | 2011-08-31 | ||
| US201161573433P | 2011-09-06 | 2011-09-06 | |
| EP17157922.0A EP3199533B1 (en) | 2011-08-31 | 2012-08-30 | Pyrazole compound and pharmaceutical use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HRP20190730T1 true HRP20190730T1 (hr) | 2019-07-12 |
Family
ID=66948704
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HRP20190730TT HRP20190730T1 (hr) | 2011-08-31 | 2019-04-16 | Spoj pirazola i njegova farmaceutska upotreba |
Country Status (7)
| Country | Link |
|---|---|
| ES (1) | ES2720366T3 (es) |
| HR (1) | HRP20190730T1 (es) |
| HU (1) | HUE043268T2 (es) |
| LT (1) | LT3199533T (es) |
| ME (1) | ME03416B (es) |
| PT (1) | PT3199533T (es) |
| TR (1) | TR201906461T4 (es) |
-
2012
- 2012-08-30 LT LTEP17157922.0T patent/LT3199533T/lt unknown
- 2012-08-30 ME MEP-2019-130A patent/ME03416B/me unknown
- 2012-08-30 HU HUE17157922A patent/HUE043268T2/hu unknown
- 2012-08-30 PT PT17157922T patent/PT3199533T/pt unknown
- 2012-08-30 ES ES17157922T patent/ES2720366T3/es active Active
- 2012-08-30 TR TR2019/06461T patent/TR201906461T4/tr unknown
-
2019
- 2019-04-16 HR HRP20190730TT patent/HRP20190730T1/hr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PT3199533T (pt) | 2019-05-28 |
| TR201906461T4 (tr) | 2019-05-21 |
| LT3199533T (lt) | 2019-06-25 |
| HUE043268T2 (hu) | 2019-08-28 |
| ME03416B (me) | 2020-01-20 |
| ES2720366T3 (es) | 2019-07-19 |
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