HRP20161288T1 - Topikalni farmaceutski pripravci koji sadrže mometazon furoat - Google Patents

Topikalni farmaceutski pripravci koji sadrže mometazon furoat Download PDF

Info

Publication number
HRP20161288T1
HRP20161288T1 HRP20161288TT HRP20161288T HRP20161288T1 HR P20161288 T1 HRP20161288 T1 HR P20161288T1 HR P20161288T T HRP20161288T T HR P20161288TT HR P20161288 T HRP20161288 T HR P20161288T HR P20161288 T1 HRP20161288 T1 HR P20161288T1
Authority
HR
Croatia
Prior art keywords
weight
percent
preparation
preparation according
weight percent
Prior art date
Application number
HRP20161288TT
Other languages
English (en)
Inventor
Fritjof Evers
Henning Mallwitz
Ricarda Meyer
Christoph Willers
Original Assignee
Almirall S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Almirall S.A. filed Critical Almirall S.A.
Publication of HRP20161288T1 publication Critical patent/HRP20161288T1/hr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/04Antipruritics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dermatology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dispersion Chemistry (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Claims (13)

1. Topikalni farmaceutski pripravak, naznačen time, da sadržava, u odnosu na ukupnu masu pripravka: a) 0,01 do 0,2 težinskih postotaka mometazon furoata, b) 5 do 18 težinskih postotaka heksilen glikola, c) 20 do 40 težinskih postotaka vode i d) 25 do 70 težinskih postotaka uljne faze, pri čemu je mometazon furoat suspendiran (raspršen) u pripravku.
2. Pripravak u skladu s patentnim zahtjevom 1, naznačen time, da je ukupna količina a) mometazon furoata u rasponu od 0,05 do 0,15 težinskih postotaka, poželjno od 0,08 do 0,12 težinskih postotaka s obzirom na ukupnu težinu pripravka.
3. Pripravak u skladu s bilo kojim od patentnih zahtjeva 1 ili 2, naznačen time, da je ukupna količina b) heksilen glikola u rasponu od 7 do 15 težinskih postotaka, poželjno 8 do 13 težinskih postotaka s obzirom na ukupnu težinu pripravka.
4. Pripravak u skladu s bilo kojim od prethodnih patentnih zahtjeva, naznačen time, da je ukupna količina c) vode u rasponu od 25 do 40 težinskih postotaka, poželjno 25 do 35 težinskih postotaka, još poželjnije 26 do 34 težinskih postotaka s obzirom na ukupnu težinu pripravka.
5. Pripravak u skladu s bilo kojim od patentnih prethodnih zahtjeva, naznačen time, da je ukupna količina d) uljne faze u rasponu od 30 do 65 težinskih postotaka s obzirom na ukupnu težinu pripravka.
6. Pripravak u skladu s patentnim zahtjevom 1, naznačen time, da se sastoji s obzirom na ukupnu težinu pripravka, od: a) 0,01 do 0,2 težinskih postotaka, poželjno 0,05 do 0,15 težinskih postotaka mometazon furoata, b) 5 do 18 težinskih postotaka, poželjno 7 do 15 težinskih postotaka heksilen glikola, c) 20 do 40 težinskih postotaka, poželjno 25 do 35 težinskih postotaka vode i d) 25 do 70 težinskih postotaka, poželjno 30 do 65 težinskih postotaka uljne faze.
7. Pripravak u skladu s patentnim zahtjevom 6, naznačen time, da sadržava, u odnosu na ukupnu masu pripravka: a) 0,05 do 0,15 težinskih postotaka, poželjno 0,08 do 0,12 težinskih postotaka mometazon furoata, b) od 7 do 15 težinskih postotaka, poželjno 8 do 13 težinskih postotaka heksilen glikola, c) 25 do 35 težinskih postotaka, poželjno 26 do 34 težinskih postotaka vode, d1) 32 do 50 težinskih postotaka, poželjno 35 do 48 težinskih postotaka naftnih ugljikovodika, d2) 5 do 12 težinskih postotaka, poželjno 7 do 10 težinskih postotaka C6-C24 masnih alkohola i d3) 0,1 do 5 težinskih postotaka, poželjno 0,5 do 3 težinskih postotaka bilo kojeg poliola osim heksilen glikola.
8. Pripravak u skladu s patentnim zahtjevom 7, naznačen time, da sadržava, u odnosu na ukupnu masu pripravka: a) 0,08 do 0,12 težinskih postotaka mometazon furoata, b) 8 do 13 težinskih postotaka heksilen glikola, c) 26 do 34 težinskih postotaka vode, d1) 35 do 48 težinskih postotaka naftnih ugljikovodika odabranih iz skupine koju čine tekući parafin, bijeli parafin ili njihove smjese, d2) 7 do 10 težinskih postotaka C6-C24 masnih alkohola odabranih iz skupine koju čine lauril alkohol, miristil alkohol, palmitil alkohol, stearil alkohol, oleil alkohol ili njihove smjese i d3) 0,5 do 3 težinskih postotaka glicerola.
9. Pripravak u skladu s bilo kojim od patentnih prethodnih zahtjeva, naznačen time, da pripravak nadalje sadržava sredstva protiv iritiranja, antioksidanse, pufere, sredstva za tvorbu helata, sredstva za ublaživanje, sredstva za pojačavanje penetracije, konzervanse, sredstva za pospješivanje otapanja, sredstva za zgušnjavanje, sredstva za vlaženje ili mješavine istih.
10. Pripravak u skladu s bilo kojim od prethodnih patentnih zahtjeva, naznačen time, da spomenuti pripravak ima pH vrijednost u rasponu od 3,0 do 6,0.
11. Pripravak u skladu s bilo kojim od prethodnih patentnih zahtjeva, naznačen time, da je pripravak formuliran u obliku kreme.
12. Pripravak u skladu s bilo kojim od patentnih zahtjeva 1 do 11, naznačen time, da se rabi u liječenju ili prevenciji psorijaze, atopičnog dermatitisa i drugih kožnih poremećaja ili bolesti.
13. Uporaba pripravka u skladu s bilo kojim od patentnih zahtjeva 1 do 11, naznačena time, da je namijenjena proizvodnji lijeka za liječenje ili prevenciju psorijaze, atopičnog dermatitisa i drugih kožnih poremećaja ili bolesti.
HRP20161288TT 2010-05-26 2016-10-06 Topikalni farmaceutski pripravci koji sadrže mometazon furoat HRP20161288T1 (hr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP10382146A EP2394653A1 (en) 2010-05-26 2010-05-26 Topical pharmaceutical compositions comprising mometasone furoate
US36505010A 2010-07-16 2010-07-16
PCT/EP2011/002369 WO2011147536A2 (en) 2010-05-26 2011-05-13 Topical pharmaceutical compositions
EP11719487.8A EP2575822B1 (en) 2010-05-26 2011-05-13 Topical pharmaceutical compositions comprising mometasone furoate

Publications (1)

Publication Number Publication Date
HRP20161288T1 true HRP20161288T1 (hr) 2016-11-18

Family

ID=42797321

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20161288TT HRP20161288T1 (hr) 2010-05-26 2016-10-06 Topikalni farmaceutski pripravci koji sadrže mometazon furoat

Country Status (33)

Country Link
US (2) US20140200203A1 (hr)
EP (2) EP2394653A1 (hr)
JP (1) JP5743241B2 (hr)
KR (1) KR101790371B1 (hr)
CN (1) CN102883725B (hr)
AR (1) AR081765A1 (hr)
AU (1) AU2011257586B2 (hr)
BR (1) BR112012030006A2 (hr)
CA (1) CA2794553C (hr)
CL (1) CL2012003282A1 (hr)
CO (1) CO6640244A2 (hr)
DK (1) DK2575822T3 (hr)
EA (1) EA022967B1 (hr)
ES (1) ES2595250T3 (hr)
HK (1) HK1177893A1 (hr)
HR (1) HRP20161288T1 (hr)
HU (1) HUE029818T2 (hr)
IL (1) IL222163B (hr)
LT (1) LT2575822T (hr)
ME (1) ME02555B (hr)
MX (1) MX2012013642A (hr)
MY (1) MY160377A (hr)
NZ (1) NZ602730A (hr)
PL (1) PL2575822T3 (hr)
PT (1) PT2575822T (hr)
RS (1) RS55233B1 (hr)
SG (2) SG184405A1 (hr)
SI (1) SI2575822T1 (hr)
SM (1) SMT201600342B (hr)
TW (1) TWI473615B (hr)
UY (1) UY33404A (hr)
WO (1) WO2011147536A2 (hr)
ZA (1) ZA201208420B (hr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2394653A1 (en) 2010-05-26 2011-12-14 Almirall, S.A. Topical pharmaceutical compositions comprising mometasone furoate
WO2015005419A1 (ja) * 2013-07-11 2015-01-15 株式会社ポーラファルマ 使用時泡状を呈する外用組成物
GB2540764A (en) * 2015-07-24 2017-02-01 Fontus Health Ltd Topical composition
SG11201908351TA (en) * 2017-03-10 2019-10-30 Edmond J Lavoie Indole derivatives as efflux pump inhibitors
EP3492068A1 (en) * 2017-12-01 2019-06-05 NCP NewCare Products GmbH Composition for treating onychomycosis
CN114767630A (zh) * 2022-06-06 2022-07-22 黑龙江中医药大学 一种治疗变应性鼻炎的药物组合物及其用途

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4808610A (en) 1986-10-02 1989-02-28 Schering Corporation Mometasone furoate anti-inflammatory cream composition using hexylene glycol
US4775529A (en) 1987-05-21 1988-10-04 Schering Corporation Steroid lotion
AU6974191A (en) 1989-12-20 1991-07-18 Schering Corporation Stable cream and lotion bases for lipophilic drug compositions
DE69433923T2 (de) 1993-12-21 2005-07-21 Schering Corp. Salbe enthaltend mometason-furoat und salicylsäure zur topischen behandlung von psoriasis
US5696105A (en) * 1996-03-14 1997-12-09 Hackler; Walter A. Antifungal nail composition
JP3676674B2 (ja) 1997-10-09 2005-07-27 シェーリング コーポレイション 噴霧のためのモメタゾンフロエート懸濁液
TR200201343A2 (tr) 2002-05-17 2003-12-22 Orva İlaç Sanayi̇ Ve Ti̇caret A. Ş. Kortikosteroid ve antiseptik içeren farmasötik bileşim
WO2004105686A2 (en) 2003-05-23 2004-12-09 Taro Pharmaceuticals U.S.A., Inc. Novel topical steroid cream formulations
DE102006034883A1 (de) 2006-07-25 2008-01-31 Hermal Kurt Herrmann Gmbh & Co. Ohg Pharmazeutische Zusammensetzung enthaltend Mometasonfuroat
EP2120868A4 (en) 2007-04-11 2010-08-25 Perrigo Israel Phamaceuticals LOW-DOSED MOMETASON FORMULATIONS
EP2394653A1 (en) 2010-05-26 2011-12-14 Almirall, S.A. Topical pharmaceutical compositions comprising mometasone furoate

Also Published As

Publication number Publication date
ME02555B (me) 2017-02-20
US20140200203A1 (en) 2014-07-17
AU2011257586B2 (en) 2014-04-17
TWI473615B (zh) 2015-02-21
AR081765A1 (es) 2012-10-17
DK2575822T3 (en) 2016-10-17
SI2575822T1 (sl) 2016-11-30
CN102883725A (zh) 2013-01-16
KR101790371B1 (ko) 2017-10-25
RS55233B1 (sr) 2017-02-28
SG10201502252YA (en) 2015-05-28
SMT201600342B (it) 2017-01-10
ES2595250T3 (es) 2016-12-28
EP2394653A1 (en) 2011-12-14
IL222163B (en) 2018-01-31
CO6640244A2 (es) 2013-03-22
ZA201208420B (en) 2013-09-25
JP5743241B2 (ja) 2015-07-01
JP2013530149A (ja) 2013-07-25
EP2575822B1 (en) 2016-07-06
HK1177893A1 (zh) 2013-08-30
HUE029818T2 (en) 2017-04-28
AU2011257586A1 (en) 2012-11-01
LT2575822T (lt) 2016-10-10
EA201291335A1 (ru) 2013-04-30
CL2012003282A1 (es) 2013-01-25
US9907807B2 (en) 2018-03-06
US20160038512A1 (en) 2016-02-11
CA2794553C (en) 2018-01-02
EA022967B1 (ru) 2016-03-31
TW201204367A (en) 2012-02-01
BR112012030006A2 (pt) 2016-08-02
MY160377A (en) 2017-03-15
UY33404A (es) 2011-12-01
EP2575822A2 (en) 2013-04-10
NZ602730A (en) 2014-03-28
PT2575822T (pt) 2016-10-06
WO2011147536A3 (en) 2012-06-07
MX2012013642A (es) 2013-05-06
CN102883725B (zh) 2015-04-01
PL2575822T3 (pl) 2017-01-31
SG184405A1 (en) 2012-11-29
CA2794553A1 (en) 2011-12-01
KR20130086137A (ko) 2013-07-31
WO2011147536A2 (en) 2011-12-01

Similar Documents

Publication Publication Date Title
HRP20161288T1 (hr) Topikalni farmaceutski pripravci koji sadrže mometazon furoat
BR112014029766A2 (pt) composições contendo álcoois graxos, tensoativos catiônicos e n-acil-n-metilglucaminas
BR112014029769A2 (pt) composição contendo n-metil-n-acilglucamina
Behmanesh et al. Effects of olive oil sitz bath on improvement of perineal injury after delivery.
BR112019004971A2 (pt) gel para cuidados pessoais e método
NZ717262A (en) Composition having microbiological stability comprising water and saturated fats
NZ702472A (en) Oil/water-emulsion-type topical compositions containing a retinoid
BR112015032029A2 (pt) uso de uma composição compreendendo óleo de peixe e suco para o tratamento de inflamação
MY192590A (en) Liquid skin-cleansing agent composition
HRP20191059T1 (hr) Skup aktivnih sastojaka za topikalnu primjenu u restrukturiranju izmijenjene kožne barijere poslije kožnih bolesti
TR201903470T4 (tr) Kişisel hijyen için formülasyon.
BR112014007274A2 (pt) preparação cosmética ou dermatológica para aplicação sobre a pele molhada ou úmida e método para cuidar da pele
BR112015027436A8 (pt) composição tópica e veículo para administração de ingredientes farmaceuticamente ou cosmeticamente ativos
BR112014031306A2 (pt) composição farmacêutica e respectivos usos
HRP20200504T1 (hr) Lokalni preparati farmaceutskih i medicinskih proizvoda koji sadrže kombinacije sukralfata, hijaluronske kiseline, arginina i prirodnog hidratantnog sredstva
ES2541379B1 (es) Cosmética natural de bellota
ES2562085B1 (es) Crema para el tratamiento de pieles con estados descamativos y procedimiento de fabricación de dicha crema
CN104721088A (zh) 一种护手霜
PL428523A1 (pl) Kompozycja zawierająca luteinę, zastosowanie kompozycji oraz sposób wytwarzania kompozycji
PL402321A1 (pl) Preparat do pielęgnacji skóry rąk
TH153704A (th) องค์ประกอบทางเภสัชกรรมสำหรับใช้เฉพาะที่
PE20141538A1 (es) Composicion para ser aplicada a la piel, y uso de la misma
Gallagher et al. Comparison of emollient efficacy-a single centre, randomised, double-blind, bi-lateral comparison of two emollients prescribed in the UK for the management of dry skin conditions such as atopic eczema
PL227467B1 (pl) Kompozycja kosmetyczna
TH154104A (th) ครีมดูแลผิวหนังอ่อนนุ่มที่แทรกซึมเร็ว