HRP20150613T1 - Sol benzojeve kiseline otamiksabana - Google Patents

Sol benzojeve kiseline otamiksabana Download PDF

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Publication number
HRP20150613T1
HRP20150613T1 HRP20150613TT HRP20150613T HRP20150613T1 HR P20150613 T1 HRP20150613 T1 HR P20150613T1 HR P20150613T T HRP20150613T T HR P20150613TT HR P20150613 T HRP20150613 T HR P20150613T HR P20150613 T1 HRP20150613 T1 HR P20150613T1
Authority
HR
Croatia
Prior art keywords
benzoic acid
amino
methyl
acid salt
imino
Prior art date
Application number
HRP20150613TT
Other languages
English (en)
Croatian (hr)
Inventor
Norbert Nagel
Bruno Baumgartner
Harald Berchtold
Timothy Ayers
Original Assignee
Sanofi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi filed Critical Sanofi
Publication of HRP20150613T1 publication Critical patent/HRP20150613T1/hr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/89Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/06Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
    • C07D213/16Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom containing only one pyridine ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HRP20150613TT 2011-03-29 2012-03-27 Sol benzojeve kiseline otamiksabana HRP20150613T1 (hr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP11305348 2011-03-29
US201161500342P 2011-06-23 2011-06-23
EP12711858.6A EP2691371B1 (en) 2011-03-29 2012-03-27 Benzoic acid salt of otamixaban
PCT/EP2012/055364 WO2012130821A1 (en) 2011-03-29 2012-03-27 Benzoic acid salt of otamixaban

Publications (1)

Publication Number Publication Date
HRP20150613T1 true HRP20150613T1 (hr) 2015-07-17

Family

ID=44065390

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20150613TT HRP20150613T1 (hr) 2011-03-29 2012-03-27 Sol benzojeve kiseline otamiksabana

Country Status (21)

Country Link
US (1) US8993602B2 (enExample)
EP (1) EP2691371B1 (enExample)
JP (1) JP5959617B2 (enExample)
KR (1) KR101852226B1 (enExample)
CN (1) CN103562183B (enExample)
AU (1) AU2012234325B2 (enExample)
BR (1) BR112013025105A2 (enExample)
CA (1) CA2830965C (enExample)
CY (1) CY1116659T1 (enExample)
DK (1) DK2691371T3 (enExample)
ES (1) ES2539236T3 (enExample)
HR (1) HRP20150613T1 (enExample)
IL (1) IL228574A (enExample)
MX (1) MX2013011266A (enExample)
MY (1) MY161396A (enExample)
PL (1) PL2691371T3 (enExample)
PT (1) PT2691371E (enExample)
RU (1) RU2597423C2 (enExample)
SG (1) SG193612A1 (enExample)
SI (1) SI2691371T1 (enExample)
WO (1) WO2012130821A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2012234323A1 (en) 2011-03-29 2013-10-17 Sanofi Otamixaban formulations with improved stability
CN106565698B (zh) * 2016-08-15 2019-03-08 南京帕隆材料科技有限公司 取代噻唑类衍生物及其制备方法和用途
CN106518859B (zh) * 2016-08-15 2019-01-18 南京帕隆材料科技有限公司 噻唑类衍生物及其制备方法和用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5424334A (en) 1991-12-19 1995-06-13 G. D. Searle & Co. Peptide mimetic compounds useful as platelet aggregation inhibitors
IL125163A0 (en) * 1996-01-02 1999-01-26 Rhone Poulenc Rorer Pharma Substituted n-[(aminoiminomethyl or aminomethyl) phenyl] propyl amides
US6080767A (en) * 1996-01-02 2000-06-27 Aventis Pharmaceuticals Products Inc. Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides
GB0108903D0 (en) 2000-10-05 2001-05-30 Aventis Pharm Prod Inc Novel crystalline forms of a factor Xa inhibitor
EA020045B1 (ru) * 2007-05-02 2014-08-29 Портола Фармасьютиклз, Инк. Комбинированная терапия соединением, проявляющим активность ингибитора рецептора адф на тромбоцитах
AU2010277725B2 (en) * 2009-07-29 2016-08-18 Sanofi Otamixaban for treatment of elderly and renal impaired non-ST elevation myocardial infarction patients

Also Published As

Publication number Publication date
BR112013025105A2 (pt) 2017-06-06
CA2830965A1 (en) 2012-10-04
HK1189584A1 (en) 2014-06-13
CN103562183A (zh) 2014-02-05
SG193612A1 (en) 2013-11-29
SI2691371T1 (sl) 2015-07-31
WO2012130821A1 (en) 2012-10-04
CY1116659T1 (el) 2017-03-15
MX2013011266A (es) 2014-03-27
AU2012234325B2 (en) 2016-08-11
DK2691371T3 (da) 2015-06-22
CA2830965C (en) 2019-04-09
ES2539236T3 (es) 2015-06-29
EP2691371B1 (en) 2015-03-18
CN103562183B (zh) 2015-12-23
PT2691371E (pt) 2015-07-20
KR20140022851A (ko) 2014-02-25
EP2691371A1 (en) 2014-02-05
US8993602B2 (en) 2015-03-31
US20140024684A1 (en) 2014-01-23
MY161396A (en) 2017-04-14
RU2013148005A (ru) 2015-05-10
IL228574A0 (en) 2013-12-31
JP2014509622A (ja) 2014-04-21
RU2597423C2 (ru) 2016-09-10
JP5959617B2 (ja) 2016-08-02
KR101852226B1 (ko) 2018-04-25
IL228574A (en) 2015-07-30
AU2012234325A1 (en) 2013-10-17
PL2691371T3 (pl) 2015-08-31

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