HRP20100577T1 - Uporaba agomelatina za dobivanje lijeka s ciljem liječenja općeg poremećaja anksioznosti - Google Patents

Uporaba agomelatina za dobivanje lijeka s ciljem liječenja općeg poremećaja anksioznosti Download PDF

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Publication number
HRP20100577T1
HRP20100577T1 HR20100577T HRP20100577T HRP20100577T1 HR P20100577 T1 HRP20100577 T1 HR P20100577T1 HR 20100577 T HR20100577 T HR 20100577T HR P20100577 T HRP20100577 T HR P20100577T HR P20100577 T1 HRP20100577 T1 HR P20100577T1
Authority
HR
Croatia
Prior art keywords
agomelatine
anxiety disorder
pharmaceutically acceptable
hydrates
generalised anxiety
Prior art date
Application number
HR20100577T
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English (en)
Inventor
Delalleau Bruno
Fabiano Agnes
Millan Mark
Mocaer Elisabeth
Original Assignee
Les Laboratoires Servier
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37308935&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20100577(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Les Laboratoires Servier filed Critical Les Laboratoires Servier
Publication of HRP20100577T1 publication Critical patent/HRP20100577T1/hr

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/04Nitro compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Uporaba agomelatina ili N-[2-(7-metoksi-1-naftil)etil]acetamida ili jednog od njegovih hidrata, kristalnih oblika i adicijskih soli s farmaceutski prihvatljivom kiselinom ili lužinom, kao jednim djelatnim sastojkom, naznačena time, da je za dobivanje lijeka namijenjenog za liječenje općeg poremećaja anksioznosti. Patent sadrži još 3 patentna zahtjeva.

Claims (4)

1. Uporaba agomelatina ili N-[2-(7-metoksi-1-naftil)etil]acetamida ili jednog od njegovih hidrata, kristalnih oblika i adicijskih soli s farmaceutski prihvatljivom kiselinom ili lužinom, kao jednim djelatnim sastojkom, naznačena time, da je za dobivanje lijeka namijenjenog za liječenje općeg poremećaja anksioznosti.
2. Uporaba u skladu s patentnim zahtjevom 1, naznačena time da je agomelatin dobiven u kristalnom obliku II.
3. Farmaceutske smjese koje, kao djelatni sastojci, sadrže agomelatin, ili jedan od njegovih hidrata, kristalnih oblika i adicijskih soli s farmaceutski prihvatljivom kiselinom ili lužinom, same ili u kombinaciji s jednim ili više farmaceutski prihvatljivih ekscipijensa, naznačeno time, da su za uporabu u liječenju općeg poremećaja anksioznosti.
4. Farmaceutska smjesa u skladu s patentnim zahtjevom 3, naznačena time da je agomelatin dobiven u kristalnom obliku II.
HR20100577T 2006-04-07 2010-10-21 Uporaba agomelatina za dobivanje lijeka s ciljem liječenja općeg poremećaja anksioznosti HRP20100577T1 (hr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0603083A FR2899472B1 (fr) 2006-04-07 2006-04-07 Utilisation de l'agomelatine pour l'obtention de medicaments destines au traitement du trouble anxiete generalisee

Publications (1)

Publication Number Publication Date
HRP20100577T1 true HRP20100577T1 (hr) 2010-11-30

Family

ID=37308935

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20100577T HRP20100577T1 (hr) 2006-04-07 2010-10-21 Uporaba agomelatina za dobivanje lijeka s ciljem liječenja općeg poremećaja anksioznosti

Country Status (44)

Country Link
US (1) US7960438B2 (hr)
EP (1) EP1842535B1 (hr)
JP (1) JP4880031B2 (hr)
KR (1) KR20070100657A (hr)
CN (1) CN101049290B (hr)
AP (1) AP2488A (hr)
AR (1) AR060349A1 (hr)
AT (1) ATE477798T1 (hr)
AU (1) AU2007201527B2 (hr)
BR (1) BRPI0701601A (hr)
CA (1) CA2584060C (hr)
CO (1) CO5840252A1 (hr)
CR (1) CR9019A (hr)
CY (1) CY1111287T1 (hr)
DE (1) DE602007008494D1 (hr)
DK (1) DK1842535T3 (hr)
EA (1) EA012608B1 (hr)
ES (1) ES2351062T3 (hr)
FR (1) FR2899472B1 (hr)
GE (1) GEP20094743B (hr)
GT (1) GT200700032A (hr)
HK (1) HK1108367A1 (hr)
HR (1) HRP20100577T1 (hr)
IL (1) IL182407A (hr)
JO (1) JO3440B1 (hr)
MA (1) MA28987B1 (hr)
ME (1) ME01865B (hr)
MX (1) MX2007004100A (hr)
MY (1) MY143269A (hr)
NI (1) NI200700084A (hr)
NO (1) NO20071774L (hr)
NZ (1) NZ554347A (hr)
PE (1) PE20080174A1 (hr)
PL (1) PL1842535T3 (hr)
PT (1) PT1842535E (hr)
RS (1) RS51485B (hr)
SA (1) SA07280161B1 (hr)
SG (1) SG136881A1 (hr)
SI (1) SI1842535T1 (hr)
TN (1) TNSN07118A1 (hr)
TW (1) TWI374736B (hr)
UY (1) UY30262A1 (hr)
WO (1) WO2007116136A1 (hr)
ZA (1) ZA200702865B (hr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101481321B (zh) * 2009-02-27 2012-04-18 上海医药工业研究院 阿戈美拉汀卤化氢复合物及其制备方法
CN101585779B (zh) * 2009-03-10 2014-04-02 上海医药工业研究院 阿戈美拉汀的晶型vi及其制备方法和应用
FR2956031B1 (fr) * 2010-02-11 2012-03-02 Servier Lab Utilisation de l'agomelatine pour l'obtention de medicaments destines au traitement du trouble obsessionnel compulsif (toc)
CN102190595A (zh) * 2010-03-17 2011-09-21 上海医药工业研究院 阿戈美拉汀溴化氢水合物及其制备方法
CN102190594A (zh) * 2010-03-17 2011-09-21 上海医药工业研究院 阿戈美拉汀氯化氢水合物及其制备方法
PH12012000132A1 (en) * 2011-06-09 2014-10-20 Servier Lab New co-crystals of agomelatine, a process for their preparation and pharmaceutical compositions containing them
FR2978916B1 (fr) * 2011-08-10 2013-07-26 Servier Lab Composition pharmaceutique solide pour administration buccale d'agomelatine
EP2810647A1 (en) 2013-06-06 2014-12-10 Zentiva, a.s. Pharmaceutical formulations comprising agomelatine in the form of agomelatine co-crystal with an organic acid
EP2810656B1 (en) 2013-06-06 2017-08-02 Zentiva, a.s. Agomelatine formulations comprising agomelatine in the form of co-crystals
IT201900002913A1 (it) 2019-03-01 2020-09-01 Nicola Pescosolido Composto utile per il trattamento del glaucoma
CN110867197A (zh) * 2019-10-23 2020-03-06 吴杰 语音交互过程中实时打断语音机器人的方法及设备

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2658818B1 (fr) * 1990-02-27 1993-12-31 Adir Cie Nouveaux derives a structure naphtalenique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
SG45100A1 (en) * 1994-03-07 1998-01-16 Ibm Improvements in image processing
DE19532842C1 (de) * 1995-09-05 1996-12-19 Ibm Bildaufnahmesystem
AR047553A1 (es) * 2003-07-04 2006-01-25 Lundbeck & Co As H La combinacion de un inhibidor de reabsorcion de serotonina y agomelatina
AU2004308962A1 (en) * 2003-12-24 2005-07-14 Sepracor Inc. Melatonin combination therapy for improving sleep quality
FR2866335B1 (fr) * 2004-02-13 2006-05-26 Servier Lab Nouveau procede de synthese de l'agomelatine
JP2008531714A (ja) * 2005-03-04 2008-08-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 不安障害の治療用及び/又は予防用の医薬組成物
US7358395B2 (en) * 2005-08-03 2008-04-15 Les Laboratories Servier Crystalline form V of agomelatine, a process for its preparation and pharmaceutical compositions containing it
US7635721B2 (en) * 2005-08-03 2009-12-22 Les Laboratoires Servier Crystalline form III of agomelatine, a process for its preparation and pharmaceutical compositions containing it
TW200735878A (en) * 2005-11-18 2007-10-01 Astrazeneca Ab Pharmaceutical compositions

Also Published As

Publication number Publication date
FR2899472A1 (fr) 2007-10-12
IL182407A0 (en) 2008-01-20
ME01865B (me) 2011-04-30
PL1842535T3 (pl) 2011-01-31
FR2899472B1 (fr) 2008-09-12
MA28987B1 (fr) 2007-11-01
PE20080174A1 (es) 2008-03-29
EA200700574A2 (ru) 2007-10-26
JO3440B1 (ar) 2019-10-20
US7960438B2 (en) 2011-06-14
EP1842535B1 (fr) 2010-08-18
UY30262A1 (es) 2007-05-31
WO2007116136A1 (fr) 2007-10-18
KR20070100657A (ko) 2007-10-11
SG136881A1 (en) 2007-11-29
AP2488A (en) 2012-10-03
RS51485B (en) 2011-04-30
CA2584060A1 (fr) 2007-10-07
JP2009532446A (ja) 2009-09-10
CO5840252A1 (es) 2007-12-31
HK1108367A1 (en) 2008-05-09
AP2007003953A0 (en) 2007-04-30
TW200808295A (en) 2008-02-16
AU2007201527A1 (en) 2007-10-25
EA012608B1 (ru) 2009-10-30
PT1842535E (pt) 2010-09-28
ZA200702865B (en) 2008-07-30
ES2351062T3 (es) 2011-01-31
BRPI0701601A (pt) 2007-12-11
SA07280161B1 (ar) 2010-10-23
DK1842535T3 (da) 2010-11-15
US20070238792A1 (en) 2007-10-11
AU2007201527B2 (en) 2012-08-09
SI1842535T1 (sl) 2010-10-29
AR060349A1 (es) 2008-06-11
TNSN07118A1 (fr) 2008-06-02
GT200700032A (es) 2007-10-31
JP4880031B2 (ja) 2012-02-22
EA200700574A3 (ru) 2007-12-28
IL182407A (en) 2016-02-29
MY143269A (en) 2011-04-15
CA2584060C (fr) 2011-04-26
CN101049290B (zh) 2012-10-31
NZ554347A (en) 2008-08-29
GEP20094743B (en) 2009-07-27
EP1842535A1 (fr) 2007-10-10
DE602007008494D1 (de) 2010-09-30
CY1111287T1 (el) 2015-08-05
NI200700084A (es) 2008-04-24
CR9019A (es) 2008-10-28
CN101049290A (zh) 2007-10-10
TWI374736B (en) 2012-10-21
NO20071774L (no) 2007-10-08
MX2007004100A (es) 2009-02-16
ATE477798T1 (de) 2010-09-15

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