HRP20040435A2 - Solid pharmaceutical formulation for a piperazineurea derivative - Google Patents
Solid pharmaceutical formulation for a piperazineurea derivative Download PDFInfo
- Publication number
- HRP20040435A2 HRP20040435A2 HR20040435A HRP20040435A HRP20040435A2 HR P20040435 A2 HRP20040435 A2 HR P20040435A2 HR 20040435 A HR20040435 A HR 20040435A HR P20040435 A HRP20040435 A HR P20040435A HR P20040435 A2 HRP20040435 A2 HR P20040435A2
- Authority
- HR
- Croatia
- Prior art keywords
- methyl
- piperazine
- pharmaceutical reagent
- acid
- fluorobenzyl
- Prior art date
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Classifications
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
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- A—HUMAN NECESSITIES
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- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A61K9/2004—Excipients; Inactive ingredients
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- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
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- Immunology (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
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- Cardiology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pulmonology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10152351A DE10152351B4 (de) | 2001-10-18 | 2001-10-18 | Feste Arzneimittelformulierung für ein Piperazinharnstoffderivat |
PCT/EP2002/011229 WO2003035037A1 (de) | 2001-10-18 | 2002-10-07 | Feste arzneimittelformulierung für ein piperazinharnstoffderivat |
Publications (1)
Publication Number | Publication Date |
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HRP20040435A2 true HRP20040435A2 (en) | 2005-06-30 |
Family
ID=7703496
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HR20040435A HRP20040435A2 (en) | 2001-10-18 | 2004-05-17 | Solid pharmaceutical formulation for a piperazineurea derivative |
Country Status (23)
Country | Link |
---|---|
EP (1) | EP1435917A1 (es) |
JP (1) | JP2005506365A (es) |
KR (1) | KR20040047920A (es) |
CN (1) | CN1571660A (es) |
AR (1) | AR037111A1 (es) |
AU (1) | AU2002333896B2 (es) |
BR (1) | BR0213340A (es) |
CA (1) | CA2463951A1 (es) |
CO (1) | CO5580740A2 (es) |
DE (1) | DE10152351B4 (es) |
EC (1) | ECSP045108A (es) |
HR (1) | HRP20040435A2 (es) |
IL (1) | IL161166A0 (es) |
MX (1) | MXPA04003522A (es) |
NO (1) | NO20042022L (es) |
NZ (1) | NZ532287A (es) |
PE (1) | PE20030472A1 (es) |
PL (1) | PL367987A1 (es) |
RS (1) | RS32204A (es) |
RU (1) | RU2311172C2 (es) |
UY (1) | UY27500A1 (es) |
WO (1) | WO2003035037A1 (es) |
ZA (1) | ZA200403781B (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE374181T1 (de) | 2001-06-27 | 2007-10-15 | Smithkline Beecham Corp | Fluorpyrrolidine als dipeptidylpeptidaseinhibitoren |
EP1749519A1 (de) * | 2005-08-05 | 2007-02-07 | Schering Aktiengesellschaft | Arzneiform mit Retardtierter pH-unabhängiger Wirkstofffreisetzung für Wirkstoffe mit starker pH-abhängiger Löslichkeit |
EP2010158B1 (en) * | 2006-04-26 | 2016-02-17 | Alphapharm Pty Ltd. | Controlled release formulations comprising uncoated discrete unit(s) and an extended release matrix |
DE102008047910A1 (de) | 2008-09-19 | 2010-03-25 | Molkerei Meggle Wasserburg Gmbh & Co. Kg | Tablettierhilfsstoff auf Laktose- und Cellulosebasis |
KR101654582B1 (ko) | 2016-05-12 | 2016-09-06 | 그린로드(주) | 원뿔형 부유 고분자 필터, 및 그의 제조장치 및 제조방법, 및 그를 포함하는 수처리 필터 |
RU2729223C1 (ru) * | 2020-05-13 | 2020-08-05 | Мераб Георгиевич Чикобава | Дозированная форма для амплификации нуклеиновых кислот |
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Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6207665B1 (en) * | 1997-06-12 | 2001-03-27 | Schering Aktiengesellschaft | Piperazine derivatives and their use as anti-inflammatory agents |
EA003137B1 (ru) * | 1998-02-05 | 2003-02-27 | Пфайзер Продактс Инк | Новые производные дигидроксигексановой кислоты |
EP1027885B1 (en) * | 1999-02-09 | 2008-07-09 | Pfizer Products Inc. | Basic drug compositions with enhanced bioavailability |
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2001
- 2001-10-18 DE DE10152351A patent/DE10152351B4/de not_active Expired - Fee Related
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2002
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- 2002-10-07 RU RU2004115328/15A patent/RU2311172C2/ru not_active IP Right Cessation
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- 2002-10-07 AU AU2002333896A patent/AU2002333896B2/en not_active Ceased
- 2002-10-07 NZ NZ532287A patent/NZ532287A/en unknown
- 2002-10-07 CA CA002463951A patent/CA2463951A1/en not_active Abandoned
- 2002-10-07 KR KR10-2004-7005591A patent/KR20040047920A/ko not_active Application Discontinuation
- 2002-10-07 RS YU32204A patent/RS32204A/sr unknown
- 2002-10-07 WO PCT/EP2002/011229 patent/WO2003035037A1/de not_active Application Discontinuation
- 2002-10-07 JP JP2003537604A patent/JP2005506365A/ja active Pending
- 2002-10-17 PE PE2002001027A patent/PE20030472A1/es not_active Application Discontinuation
- 2002-10-17 UY UY27500A patent/UY27500A1/es not_active Application Discontinuation
- 2002-10-18 AR ARP020103929A patent/AR037111A1/es unknown
-
2004
- 2004-05-13 CO CO04044345A patent/CO5580740A2/es not_active Application Discontinuation
- 2004-05-14 NO NO20042022A patent/NO20042022L/no not_active Application Discontinuation
- 2004-05-17 EC EC2004005108A patent/ECSP045108A/es unknown
- 2004-05-17 HR HR20040435A patent/HRP20040435A2/hr not_active Application Discontinuation
- 2004-05-17 ZA ZA200403781A patent/ZA200403781B/en unknown
Also Published As
Publication number | Publication date |
---|---|
WO2003035037A1 (de) | 2003-05-01 |
AR037111A1 (es) | 2004-10-20 |
CO5580740A2 (es) | 2005-11-30 |
EP1435917A1 (de) | 2004-07-14 |
DE10152351A1 (de) | 2003-05-08 |
RS32204A (en) | 2006-10-27 |
PE20030472A1 (es) | 2003-06-16 |
KR20040047920A (ko) | 2004-06-05 |
RU2004115328A (ru) | 2005-06-10 |
BR0213340A (pt) | 2004-10-05 |
UY27500A1 (es) | 2003-06-30 |
DE10152351B4 (de) | 2005-09-22 |
AU2002333896A2 (en) | 2003-05-06 |
PL367987A1 (en) | 2005-03-21 |
NZ532287A (en) | 2007-04-27 |
RU2311172C2 (ru) | 2007-11-27 |
AU2002333896B2 (en) | 2007-07-26 |
MXPA04003522A (es) | 2004-07-23 |
NO20042022L (no) | 2004-05-14 |
CA2463951A1 (en) | 2003-05-01 |
JP2005506365A (ja) | 2005-03-03 |
ECSP045108A (es) | 2004-06-28 |
IL161166A0 (en) | 2004-08-31 |
ZA200403781B (en) | 2004-11-29 |
CN1571660A (zh) | 2005-01-26 |
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