HK1223615A1 - 多環氨基甲酰基吡啶酮化合物和其用於治療 感染的用途 - Google Patents

多環氨基甲酰基吡啶酮化合物和其用於治療 感染的用途

Info

Publication number
HK1223615A1
HK1223615A1 HK16111945.5A HK16111945A HK1223615A1 HK 1223615 A1 HK1223615 A1 HK 1223615A1 HK 16111945 A HK16111945 A HK 16111945A HK 1223615 A1 HK1223615 A1 HK 1223615A1
Authority
HK
Hong Kong
Prior art keywords
hiv
polycyclic
treatment
carbamoylpyridone compounds
infections
Prior art date
Application number
HK16111945.5A
Other languages
English (en)
Inventor
Ji Mingzhe
Alejandra Trejo Martin Teresa
C Desai Manoj
Jin Haolun
Pyun Hyung-Jung
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of HK1223615A1 publication Critical patent/HK1223615A1/zh

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
HK16111945.5A 2013-07-12 2016-10-17 多環氨基甲酰基吡啶酮化合物和其用於治療 感染的用途 HK1223615A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361845807P 2013-07-12 2013-07-12
PCT/US2014/046415 WO2015006733A1 (en) 2013-07-12 2014-07-11 Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections

Publications (1)

Publication Number Publication Date
HK1223615A1 true HK1223615A1 (zh) 2017-08-04

Family

ID=51257630

Family Applications (2)

Application Number Title Priority Date Filing Date
HK18105921.3A HK1246295A1 (zh) 2013-07-12 2016-10-17 多環氨基甲酰基吡啶酮化合物和其用於治療hiv感染的用途
HK16111945.5A HK1223615A1 (zh) 2013-07-12 2016-10-17 多環氨基甲酰基吡啶酮化合物和其用於治療 感染的用途

Family Applications Before (1)

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HK18105921.3A HK1246295A1 (zh) 2013-07-12 2016-10-17 多環氨基甲酰基吡啶酮化合物和其用於治療hiv感染的用途

Country Status (18)

Country Link
US (6) US9458159B2 (zh)
EP (2) EP3252053B1 (zh)
JP (1) JP6411492B2 (zh)
AU (3) AU2014286995B2 (zh)
CA (1) CA2918055C (zh)
CY (1) CY1119545T1 (zh)
DK (1) DK3019499T3 (zh)
ES (2) ES2647216T3 (zh)
HK (2) HK1246295A1 (zh)
HR (1) HRP20171807T1 (zh)
HU (1) HUE037343T2 (zh)
LT (1) LT3019499T (zh)
NO (1) NO2865735T3 (zh)
PL (1) PL3019499T3 (zh)
PT (1) PT3019499T (zh)
RS (1) RS56539B1 (zh)
SI (2) SI3252053T1 (zh)
WO (1) WO2015006733A1 (zh)

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JP7453399B2 (ja) 2020-02-24 2024-03-19 ギリアード サイエンシーズ， インコーポレイテッド Ｈｉｖ感染症を治療するための四環式化合物及びその使用
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