HK1120213A1 - Improved hiv protease inhibitors pharmaceutical formulations - Google Patents

Improved hiv protease inhibitors pharmaceutical formulations

Info

Publication number
HK1120213A1
HK1120213A1 HK08112065.7A HK08112065A HK1120213A1 HK 1120213 A1 HK1120213 A1 HK 1120213A1 HK 08112065 A HK08112065 A HK 08112065A HK 1120213 A1 HK1120213 A1 HK 1120213A1
Authority
HK
Hong Kong
Prior art keywords
hiv protease
pharmaceutical formulations
protease inhibitors
improved hiv
improved
Prior art date
Application number
HK08112065.7A
Other languages
English (en)
Inventor
Laman Alani
Soumojeet Ghosh
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23936923&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1120213(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of HK1120213A1 publication Critical patent/HK1120213A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrrole Compounds (AREA)
HK08112065.7A 2000-01-19 2008-11-04 Improved hiv protease inhibitors pharmaceutical formulations HK1120213A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US48773900A 2000-01-19 2000-01-19

Publications (1)

Publication Number Publication Date
HK1120213A1 true HK1120213A1 (en) 2009-03-27

Family

ID=23936923

Family Applications (1)

Application Number Title Priority Date Filing Date
HK08112065.7A HK1120213A1 (en) 2000-01-19 2008-11-04 Improved hiv protease inhibitors pharmaceutical formulations

Country Status (26)

Country Link
EP (3) EP1917958B1 (de)
JP (1) JP4769400B2 (de)
KR (1) KR100861885B1 (de)
CN (1) CN100536833C (de)
AT (1) ATE395049T1 (de)
AU (2) AU1940501A (de)
BG (1) BG66112B1 (de)
BR (1) BR0011864A (de)
CA (1) CA2395987C (de)
CY (3) CY1108197T1 (de)
CZ (1) CZ304118B6 (de)
DE (1) DE60038899D1 (de)
DK (3) DK1917958T3 (de)
ES (3) ES2387579T3 (de)
HK (1) HK1120213A1 (de)
HU (1) HU229778B1 (de)
IL (2) IL150265A0 (de)
MX (1) MXPA02007097A (de)
NO (1) NO331400B1 (de)
NZ (1) NZ519724A (de)
PT (3) PT2269591T (de)
SI (3) SI1917958T1 (de)
SK (1) SK287143B6 (de)
TR (1) TR201809435T4 (de)
WO (1) WO2001052821A1 (de)
ZA (1) ZA200205109B (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5767429B2 (ja) 1999-11-12 2015-08-19 アッヴィ・インコーポレイテッド 固体分散剤中の結晶化阻害剤
US8025899B2 (en) 2003-08-28 2011-09-27 Abbott Laboratories Solid pharmaceutical dosage form
GB0615211D0 (en) * 2006-07-31 2006-09-06 Ge Healthcare Uk Ltd Asymmetric flouro-substituted polymethine dyes
US20110224435A1 (en) * 2007-08-07 2011-09-15 Ranbaxy Laboratories Limited Process for preparation of amorphous lopinavir
EP2714683A4 (de) 2011-05-27 2014-11-05 Hetero Research Foundation Amorphes, co-gefälltes ritonavir
GB201808563D0 (en) 2018-05-24 2018-07-11 Univ Manchester Treatments
GB201808564D0 (en) 2018-05-24 2018-07-11 Douglas Pharmaceuticals Ltd Treatments

Family Cites Families (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US594836A (en) * 1897-11-30 Corner-brace
US5354866A (en) 1989-05-23 1994-10-11 Abbott Laboratories Retroviral protease inhibiting compounds
US5552558A (en) 1989-05-23 1996-09-03 Abbott Laboratories Retroviral protease inhibiting compounds
GB8927913D0 (en) 1989-12-11 1990-02-14 Hoffmann La Roche Amino acid derivatives
EP0558603B1 (de) 1990-11-19 1998-08-26 Monsanto Company Retrovirale protease inhibitoren
CA2056911C (en) 1990-12-11 1998-09-22 Yuuichi Nagano Hiv protease inhibitors
EP0532466A3 (en) 1991-09-12 1993-06-16 Ciba-Geigy Ag Derivatives of 5-amino-4-hydroxy-hexanoic acid and their therapeutical use
ATE216371T1 (de) 1991-10-11 2002-05-15 Du Pont Pharm Co Cyclische harnstoffe und analoga verwendbar als retrovirale proteasehemmer
US5413999A (en) 1991-11-08 1995-05-09 Merck & Co., Inc. HIV protease inhibitors useful for the treatment of AIDS
DK0541168T3 (da) 1991-11-08 1998-05-11 Merck & Co Inc HIV-proteaseinhibitorer, som er egnede til behandling af AIDS
EP0560268B1 (de) 1992-03-13 1995-01-04 Bio-Mega/Boehringer Ingelheim Research Inc. Substituierte Pipecoline-Säurederivate als HIV-Protease-Hemmer
CA2131182C (en) 1992-05-20 2005-04-26 John S. Ng Method for making intermediates useful in synthesis of retroviral protease inhibitors
US5559256A (en) 1992-07-20 1996-09-24 E. R. Squibb & Sons, Inc. Aminediol protease inhibitors
IS2334B (is) 1992-09-08 2008-02-15 Vertex Pharmaceuticals Inc., (A Massachusetts Corporation) Aspartyl próteasi hemjari af nýjum flokki súlfonamíða
US5484926A (en) 1993-10-07 1996-01-16 Agouron Pharmaceuticals, Inc. HIV protease inhibitors
DK0727419T3 (da) 1992-12-29 2002-06-10 Abbott Lab Mellemprodukter til fremstilling af forbindelser, som inhiberer retroviral protease
WO1995006061A1 (en) 1993-08-20 1995-03-02 G.D. Searle & Co. Retroviral protease inhibitors and combinations thereof
IL110752A (en) * 1993-09-13 2000-07-26 Abbott Lab Liquid semi-solid or solid pharmaceutical composition for an HIV protease inhibitor
US5559158A (en) 1993-10-01 1996-09-24 Abbott Laboratories Pharmaceutical composition
US5491253A (en) 1993-10-22 1996-02-13 Abbott Laboratories Process for the preparation of a substituted 2,5-diamino-3-hydroxyhexane
IL111991A (en) 1994-01-28 2000-07-26 Abbott Lab Liquid pharmaceutical composition of HIV protease inhibitors in organic solvent
IL129871A (en) 1994-05-06 2003-11-23 Pharmacia & Upjohn Inc Process for preparing 4-phenyl-substituted octanoyl-oxazolidin-2-one intermediates that are useful for preparing pyran-2-ones useful for treating retroviral infections
US5567823A (en) 1995-06-06 1996-10-22 Abbott Laboratories Process for the preparation of an HIV protease inhibiting compound
US6037157A (en) 1995-06-29 2000-03-14 Abbott Laboratories Method for improving pharmacokinetics
EP1295874A3 (de) * 1995-12-13 2003-04-02 Abbott Laboratories Retrovirale Protease hemmende Verbindungen
US5914332A (en) 1995-12-13 1999-06-22 Abbott Laboratories Retroviral protease inhibiting compounds
US6160122A (en) 1996-06-28 2000-12-12 Abbott Laboratories Process for the preparation of a disubstituted thiazole
ZA9710071B (en) * 1996-11-21 1998-05-25 Abbott Lab Pharmaceutical composition.
TR200103488T2 (tr) * 1999-06-04 2002-04-22 Abbott Laboratories Geliştirilmiş farmasötik formülasyonlar.

Also Published As

Publication number Publication date
PT1917958E (pt) 2012-08-16
ES2676151T3 (es) 2018-07-17
EP1917958B1 (de) 2012-06-13
BG106976A (bg) 2003-05-30
EP1917958A2 (de) 2008-05-07
ZA200205109B (en) 2003-10-31
DK1917958T3 (da) 2012-09-24
CN100536833C (zh) 2009-09-09
EP2269591B1 (de) 2018-04-04
ES2304990T3 (es) 2008-11-01
KR20020082210A (ko) 2002-10-30
IL150265A0 (en) 2002-12-01
NO20023455D0 (no) 2002-07-18
SK287143B6 (sk) 2010-01-07
MXPA02007097A (es) 2003-01-28
IL150265A (en) 2015-02-26
SI2269591T1 (en) 2018-08-31
AU2006235895B2 (en) 2009-08-13
KR100861885B1 (ko) 2008-10-09
HUP0302070A2 (hu) 2003-09-29
CZ304118B6 (cs) 2013-11-06
DK2269591T3 (en) 2018-07-16
TR201809435T4 (tr) 2018-07-23
SI1248600T1 (sl) 2008-08-31
EP1917958A3 (de) 2008-08-27
CZ20022663A3 (cs) 2002-11-13
BR0011864A (pt) 2004-07-20
JP4769400B2 (ja) 2011-09-07
AU2006235895A1 (en) 2006-11-30
NO20023455L (no) 2002-09-18
SI1917958T1 (sl) 2012-10-30
DK1248600T3 (da) 2008-09-08
AU1940501A (en) 2001-07-31
HUP0302070A3 (en) 2007-02-28
NZ519724A (en) 2004-07-30
PL361396A1 (en) 2004-10-04
CY1112995T1 (el) 2016-04-13
PT1248600E (pt) 2008-08-25
CY1108197T1 (el) 2014-02-12
WO2001052821A1 (en) 2001-07-26
PT2269591T (pt) 2018-07-09
EP1248600B1 (de) 2008-05-14
CY1120408T1 (el) 2019-07-10
ATE395049T1 (de) 2008-05-15
SK11102002A3 (sk) 2002-12-03
CN1424907A (zh) 2003-06-18
BG66112B1 (bg) 2011-05-31
HU229778B1 (hu) 2014-07-28
JP2003533435A (ja) 2003-11-11
EP1248600A1 (de) 2002-10-16
NO331400B1 (no) 2011-12-19
EP2269591A2 (de) 2011-01-05
EP2269591A3 (de) 2011-07-27
ES2387579T3 (es) 2012-09-26
CA2395987A1 (en) 2001-07-26
CA2395987C (en) 2009-12-22
DE60038899D1 (de) 2008-06-26

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Legal Events

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