HK1081954A1 - Novel 1,4-diazabicycloalkane derivatives, their preparation and use - Google Patents

Novel 1,4-diazabicycloalkane derivatives, their preparation and use

Info

Publication number
HK1081954A1
HK1081954A1 HK06102123A HK06102123A HK1081954A1 HK 1081954 A1 HK1081954 A1 HK 1081954A1 HK 06102123 A HK06102123 A HK 06102123A HK 06102123 A HK06102123 A HK 06102123A HK 1081954 A1 HK1081954 A1 HK 1081954A1
Authority
HK
Hong Kong
Prior art keywords
novel
preparation
diazabicycloalkane derivatives
diazabicycloalkane
derivatives
Prior art date
Application number
HK06102123A
Other languages
English (en)
Inventor
Dan Peters
Gunnar M Olsen
Elsebet Ostergaard Nielsen
Tino Dyhring Jorgensen
Philip K Ahring
Original Assignee
Neurosearch As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/DK2003/000639 external-priority patent/WO2004029053A1/en
Application filed by Neurosearch As filed Critical Neurosearch As
Publication of HK1081954A1 publication Critical patent/HK1081954A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
HK06102123A 2002-09-30 2006-02-17 Novel 1,4-diazabicycloalkane derivatives, their preparation and use HK1081954A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA200201456 2002-09-30
DKPA200201738 2002-11-11
PCT/DK2003/000639 WO2004029053A1 (en) 2002-09-30 2003-09-29 Novel 1,4-diazabicycloalkane derivatives, their preparation and use

Publications (1)

Publication Number Publication Date
HK1081954A1 true HK1081954A1 (en) 2006-05-26

Family

ID=34828377

Family Applications (1)

Application Number Title Priority Date Filing Date
HK06102123A HK1081954A1 (en) 2002-09-30 2006-02-17 Novel 1,4-diazabicycloalkane derivatives, their preparation and use

Country Status (12)

Country Link
JP (1) JP4711391B2 (de)
KR (1) KR20050062575A (de)
CN (1) CN1326857C (de)
BR (1) BR0314183A (de)
HK (1) HK1081954A1 (de)
IL (1) IL166821A (de)
IS (1) IS7829A (de)
MX (1) MXPA05003344A (de)
NO (1) NO20052124L (de)
PT (1) PT1551835E (de)
RU (1) RU2323218C2 (de)
SI (1) SI1551835T1 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3019B1 (ar) * 2006-04-19 2016-09-05 Janssen Pharmaceutica Nv ثلاثي مستبدل 4،2،1-ثلاثي زولات
KR101458194B1 (ko) * 2006-05-30 2014-11-03 뉴로서치 에이/에스 신규한 1，4―디아자―비사이클로［3．2．2］노닐 옥사디아졸릴 유도체 및 이의 의학적 용도
US8492378B2 (en) 2006-08-03 2013-07-23 Takeda Pharmaceutical Company Limited GSK-3β inhibitor
US20100056565A1 (en) * 2007-02-15 2010-03-04 Argenta Discovery Limited Heterocyclic Derivatives as M3 Muscarinic Receptors
BR112014012056B1 (pt) 2011-11-18 2021-12-14 Heptares Therapeutics Limited Compostos agonistas do receptor m1 muscarínico, composição farmacêutica compreendendo os ditos compostos e uso dos mesmos para tratar um distúrbio cognitivo ou psicótico ou para tratamento ou diminuição da severidade da dor aguda, crônica, neuropática ou inflamatória
CN110946865B (zh) * 2015-12-10 2024-01-26 Ptc医疗公司 用于治疗亨廷顿病的方法
CN108752286B (zh) * 2016-09-18 2021-05-11 广西师范大学 1，2，8-氧代二氮杂环壬烷衍生物及其合成方法和应用
GB201617454D0 (en) 2016-10-14 2016-11-30 Heptares Therapeutics Limited Pharmaceutical compounds
GB201810239D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ226000A (en) * 1987-09-10 1991-06-25 Merck Sharp & Dohme Oxadiazolyl-azabicycloheptanes and pharmaceutical compositions
US5478939A (en) * 1994-07-20 1995-12-26 American Cyanamid Company (R,R) and (S,S) 2,5-diazabicyclo [2,2,1]heptane derivatives
FR2786770B1 (fr) * 1998-12-04 2001-01-19 Synthelabo Derives de 1,4-diazabicyclo[3.2.2.]nonane, leur preparation et leur application en therapeutique
BR0012327A (pt) * 1999-07-09 2002-07-02 Ortho Mcneil Pharm Inc Pirrolidinas e piperidinas neurotróficas, e composições e métodos relacionados
FR2804430B1 (fr) * 2000-01-28 2002-03-22 Sanofi Synthelabo Derives de 4-heteroaryl-1,4-diazabicyclo[3.2.2] nonane, leur preparation et leur application en therapeutique
FR2809732B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo DERIVES DE 4(-2-PHENYLTHIAZOL-5-yl)-1,4-DIAZABICYCLO-[3.2.2] NONANE, LEUR PREPARATION ET LEUR APPLICATION ENTHERAPEUTIQUE
FR2809731B1 (fr) * 2000-05-31 2002-07-19 Sanofi Synthelabo Derives de 1,4-diazabicyclo-[3.2.2] nonane-pheylisoxazole, leur preparation et leur application en therapeutique
US20020086871A1 (en) * 2000-12-29 2002-07-04 O'neill Brian Thomas Pharmaceutical composition for the treatment of CNS and other disorders
FR2832713B1 (fr) * 2001-11-23 2004-02-13 Sanofi Synthelabo Derives de 4-(1,3,4-thiadiazol-2-yl)-1,4-diazabicyclo[3.2.2] nonane, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
KR20050062575A (ko) 2005-06-23
PT1551835E (pt) 2007-03-30
NO20052124L (no) 2005-06-29
IL166821A0 (en) 2006-01-15
RU2005105048A (ru) 2005-11-20
IL166821A (en) 2009-06-15
CN1684965A (zh) 2005-10-19
JP2006503062A (ja) 2006-01-26
BR0314183A (pt) 2005-08-09
JP4711391B2 (ja) 2011-06-29
SI1551835T1 (sl) 2007-06-30
RU2323218C2 (ru) 2008-04-27
IS7829A (is) 2005-04-28
CN1326857C (zh) 2007-07-18
NO20052124D0 (no) 2005-04-29
MXPA05003344A (es) 2005-11-23

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20110929