HK1077582A1 - Aryl 5-thio beta-d-glucopyranside derivatives and remedies for diabetes containing sthe same - Google Patents

Aryl 5-thio beta-d-glucopyranside derivatives and remedies for diabetes containing sthe same

Info

Publication number
HK1077582A1
HK1077582A1 HK05109578A HK05109578A HK1077582A1 HK 1077582 A1 HK1077582 A1 HK 1077582A1 HK 05109578 A HK05109578 A HK 05109578A HK 05109578 A HK05109578 A HK 05109578A HK 1077582 A1 HK1077582 A1 HK 1077582A1
Authority
HK
Hong Kong
Prior art keywords
glucopyranside
remedies
aryl
derivatives
diabetes containing
Prior art date
Application number
HK05109578A
Other languages
English (en)
Inventor
Masakazu Sato
Hiroyuki Kakinuma
Hajime Asanuma
Original Assignee
Taiso Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiso Pharmaceutical Co Ltd filed Critical Taiso Pharmaceutical Co Ltd
Publication of HK1077582A1 publication Critical patent/HK1077582A1/xx

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/06Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
HK05109578A 2002-08-09 2005-10-27 Aryl 5-thio beta-d-glucopyranside derivatives and remedies for diabetes containing sthe same HK1077582A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002233015 2002-08-09
JP2003097839 2003-04-01

Publications (1)

Publication Number Publication Date
HK1077582A1 true HK1077582A1 (en) 2006-02-17

Family

ID=31719867

Family Applications (2)

Application Number Title Priority Date Filing Date
HK05109578A HK1077582A1 (en) 2002-08-09 2005-10-27 Aryl 5-thio beta-d-glucopyranside derivatives and remedies for diabetes containing sthe same
HK05111661A HK1079532A1 (en) 2002-08-09 2005-12-17 Process for selective production of aryl 5-thio-beta-d-aldohexopyranosides

Family Applications After (1)

Application Number Title Priority Date Filing Date
HK05111661A HK1079532A1 (en) 2002-08-09 2005-12-17 Process for selective production of aryl 5-thio-beta-d-aldohexopyranosides

Country Status (19)

Country Link
US (2) US7414072B2 (fr)
EP (2) EP1528066A4 (fr)
JP (2) JP3813160B2 (fr)
KR (2) KR20050056194A (fr)
CN (2) CN1312165C (fr)
AU (2) AU2003254903B9 (fr)
BR (1) BR0310006A (fr)
CA (2) CA2478889A1 (fr)
HK (2) HK1077582A1 (fr)
HR (1) HRP20040814A2 (fr)
MX (2) MXPA05000725A (fr)
NO (2) NO20043733L (fr)
NZ (1) NZ535229A (fr)
PL (2) PL375298A1 (fr)
RU (1) RU2322449C2 (fr)
TW (2) TW200409778A (fr)
UA (1) UA77300C2 (fr)
WO (2) WO2004014931A1 (fr)
ZA (1) ZA200407187B (fr)

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TW200606129A (en) * 2004-07-26 2006-02-16 Chugai Pharmaceutical Co Ltd Novel cyclohexane derivative, its prodrug, its salt and diabetic therapeutic agent containing the same
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Also Published As

Publication number Publication date
KR20050018642A (ko) 2005-02-23
CN100341885C (zh) 2007-10-10
ZA200407187B (en) 2006-02-22
CA2478889A1 (fr) 2004-02-19
WO2004014930A1 (fr) 2004-02-19
MXPA04009265A (es) 2005-01-25
KR20050056194A (ko) 2005-06-14
PL372865A1 (en) 2005-08-08
UA77300C2 (en) 2006-11-15
US7414072B2 (en) 2008-08-19
PL375298A1 (en) 2005-11-28
US7250522B2 (en) 2007-07-31
US20050256317A1 (en) 2005-11-17
KR100588457B1 (ko) 2006-06-12
TW200406396A (en) 2004-05-01
JPWO2004014930A1 (ja) 2005-12-02
CN1675233A (zh) 2005-09-28
TWI274055B (en) 2007-02-21
EP1528066A1 (fr) 2005-05-04
MXPA05000725A (es) 2005-04-08
CN1312165C (zh) 2007-04-25
NZ535229A (en) 2006-05-26
CA2493491A1 (fr) 2004-02-19
BR0310006A (pt) 2005-02-15
US20050209309A1 (en) 2005-09-22
NO20043733L (no) 2004-10-20
JP3813160B2 (ja) 2006-08-23
AU2003254903A1 (en) 2004-02-25
EP1528066A4 (fr) 2007-05-02
HRP20040814A2 (en) 2005-06-30
AU2003254904A1 (en) 2004-02-25
RU2322449C2 (ru) 2008-04-20
TW200409778A (en) 2004-06-16
RU2004135914A (ru) 2005-05-10
CN1639180A (zh) 2005-07-13
AU2003254903B9 (en) 2008-08-21
HK1079532A1 (en) 2006-04-07
AU2003254903B2 (en) 2008-07-31
JPWO2004014931A1 (ja) 2005-12-02
WO2004014931A1 (fr) 2004-02-19
NO20050650L (no) 2005-03-04
EP1541578A1 (fr) 2005-06-15

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Effective date: 20110808