HK1011355A1 - Amino alkanoic esters of rapamycin - Google Patents

Amino alkanoic esters of rapamycin

Info

Publication number
HK1011355A1
HK1011355A1 HK98112279A HK98112279A HK1011355A1 HK 1011355 A1 HK1011355 A1 HK 1011355A1 HK 98112279 A HK98112279 A HK 98112279A HK 98112279 A HK98112279 A HK 98112279A HK 1011355 A1 HK1011355 A1 HK 1011355A1
Authority
HK
Hong Kong
Prior art keywords
hydrogen
arylalkyl
rapamycin
alkyl
image
Prior art date
Application number
HK98112279A
Other languages
English (en)
Inventor
Amedeo Arturo Failli
Robert John Steffan
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of HK1011355A1 publication Critical patent/HK1011355A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
HK98112279A 1993-12-29 1998-11-24 Amino alkanoic esters of rapamycin HK1011355A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/174,120 US5389639A (en) 1993-12-29 1993-12-29 Amino alkanoic esters of rapamycin
PCT/US1994/014960 WO1995018133A1 (en) 1993-12-29 1994-12-28 Amino alkanoic esters of rapamycin

Publications (1)

Publication Number Publication Date
HK1011355A1 true HK1011355A1 (en) 1999-07-09

Family

ID=22634919

Family Applications (1)

Application Number Title Priority Date Filing Date
HK98112279A HK1011355A1 (en) 1993-12-29 1998-11-24 Amino alkanoic esters of rapamycin

Country Status (14)

Country Link
US (1) US5389639A (xx)
EP (1) EP0737197B1 (xx)
JP (1) JPH09507236A (xx)
KR (1) KR100338582B1 (xx)
AT (1) ATE217312T1 (xx)
AU (1) AU1519895A (xx)
CA (1) CA2179307A1 (xx)
DE (1) DE69430586T2 (xx)
DK (1) DK0737197T3 (xx)
ES (1) ES2177627T3 (xx)
HK (1) HK1011355A1 (xx)
PT (1) PT737197E (xx)
SG (1) SG47843A1 (xx)
WO (1) WO1995018133A1 (xx)

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Also Published As

Publication number Publication date
ES2177627T3 (es) 2002-12-16
DE69430586D1 (de) 2002-06-13
DK0737197T3 (da) 2002-08-26
JPH09507236A (ja) 1997-07-22
US5389639A (en) 1995-02-14
PT737197E (pt) 2002-09-30
EP0737197A1 (en) 1996-10-16
EP0737197B1 (en) 2002-05-08
ATE217312T1 (de) 2002-05-15
SG47843A1 (en) 1998-04-17
CA2179307A1 (en) 1995-07-06
WO1995018133A1 (en) 1995-07-06
DE69430586T2 (de) 2002-11-21
AU1519895A (en) 1995-07-17
KR100338582B1 (ko) 2002-10-12

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Legal Events

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PF Patent in force
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20051228