HK1002030A1 - Heterocyclic derivatives of acylaminothiazole their preparation and pharmaceutical compositions containing them - Google Patents

Heterocyclic derivatives of acylaminothiazole their preparation and pharmaceutical compositions containing them

Info

Publication number
HK1002030A1
HK1002030A1 HK98101048A HK98101048A HK1002030A1 HK 1002030 A1 HK1002030 A1 HK 1002030A1 HK 98101048 A HK98101048 A HK 98101048A HK 98101048 A HK98101048 A HK 98101048A HK 1002030 A1 HK1002030 A1 HK 1002030A1
Authority
HK
Hong Kong
Prior art keywords
acylaminothiazole
preparation
pharmaceutical compositions
compositions containing
heterocyclic derivatives
Prior art date
Application number
HK98101048A
Other languages
English (en)
Inventor
Jean-Pierre Bras
Daniel Frehel
Danielle Gully
Gerard Valette
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26227714&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1002030(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from FR8916122A external-priority patent/FR2655344B1/fr
Priority claimed from FR9005669A external-priority patent/FR2661677B1/fr
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of HK1002030A1 publication Critical patent/HK1002030A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
HK98101048A 1989-12-06 1998-02-11 Heterocyclic derivatives of acylaminothiazole their preparation and pharmaceutical compositions containing them HK1002030A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8916122A FR2655344B1 (fr) 1989-12-06 1989-12-06 Derives heterocycliques d'acylaminothiazoles, leur preparation et compositions pharmaceutiques en contenant.
FR9005669A FR2661677B1 (fr) 1990-05-04 1990-05-04 Derives heterocycliques d'acylaminothiazoles, leur preparation et compositions pharmaceutiques en contenant.

Publications (1)

Publication Number Publication Date
HK1002030A1 true HK1002030A1 (en) 1998-07-24

Family

ID=26227714

Family Applications (1)

Application Number Title Priority Date Filing Date
HK98101048A HK1002030A1 (en) 1989-12-06 1998-02-11 Heterocyclic derivatives of acylaminothiazole their preparation and pharmaceutical compositions containing them

Country Status (20)

Country Link
US (2) US5189049A (no)
EP (1) EP0432040B2 (no)
JP (2) JP2760903B2 (no)
KR (1) KR0147281B1 (no)
AR (1) AR248138A1 (no)
AT (1) ATE109145T1 (no)
AU (1) AU628696B2 (no)
CA (1) CA2031463C (no)
DE (1) DE69011059T3 (no)
DK (1) DK0432040T3 (no)
ES (1) ES2057490T5 (no)
FI (1) FI94249C (no)
GR (1) GR3025940T3 (no)
HK (1) HK1002030A1 (no)
HU (2) HU218276B (no)
IE (1) IE68593B1 (no)
IL (1) IL96577A (no)
LV (1) LV5802B4 (no)
MX (1) MX9203027A (no)
NO (1) NO179584C (no)

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FR2768737B1 (fr) * 1997-09-19 2000-05-19 Sanofi Sa Derives de carboxamidothiazoles, leur preparation, les compositions pharmaceutiques en contenant
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DE19908538A1 (de) 1999-02-26 2000-08-31 Aventis Pharma Gmbh Polycyclische 2-Amino-Thiazol Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen
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US20080039379A1 (en) * 2003-05-27 2008-02-14 Waratah Pharmaceuticals, Inc. Compositions Comprising Gastrin Compounds and Their Use in Diabetes
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Also Published As

Publication number Publication date
FI905941A (fi) 1991-06-07
KR910011814A (ko) 1991-08-07
ATE109145T1 (de) 1994-08-15
IL96577A (en) 1994-06-24
ES2057490T5 (es) 1998-03-16
EP0432040B2 (fr) 1997-12-17
AU628696B2 (en) 1992-09-17
JPH10130147A (ja) 1998-05-19
CA2031463C (en) 2000-07-25
LV5802B4 (lv) 1997-08-20
HU211866A9 (en) 1995-12-28
JP2760903B2 (ja) 1998-06-04
USRE37094E1 (en) 2001-03-13
EP0432040A1 (fr) 1991-06-12
JPH03279374A (ja) 1991-12-10
HU218276B (en) 2000-07-28
DE69011059T3 (de) 1998-04-09
KR0147281B1 (ko) 1998-08-17
AR248138A1 (es) 1995-06-30
NO905255D0 (no) 1990-12-05
IL96577A0 (en) 1991-09-16
FI905941A0 (fi) 1990-12-03
FI94249C (fi) 1995-08-10
HUT59400A (en) 1992-05-28
JP3035253B2 (ja) 2000-04-24
EP0432040B1 (fr) 1994-07-27
NO179584B (no) 1996-07-29
IE68593B1 (en) 1996-06-26
CA2031463A1 (en) 1991-06-07
DK0432040T3 (da) 1994-10-31
DE69011059T2 (de) 1995-03-02
HU908075D0 (en) 1991-06-28
ES2057490T3 (es) 1994-10-16
AU6777990A (en) 1991-06-20
GR3025940T3 (en) 1998-04-30
DE69011059D1 (de) 1994-09-01
NO179584C (no) 1996-11-06
FI94249B (fi) 1995-04-28
US5189049A (en) 1993-02-23
MX9203027A (es) 1992-07-01
LV5802A4 (lv) 1997-02-20
NO905255L (no) 1991-06-07
IE904310A1 (en) 1991-06-19

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Legal Events

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PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)