GR37776B - METHOD FOR THE PREPARATION OF BENZOLOSULPHONYLOURIES. - Google Patents

METHOD FOR THE PREPARATION OF BENZOLOSULPHONYLOURIES.

Info

Publication number
GR37776B
GR37776B GR670137776A GR670137776A GR37776B GR 37776 B GR37776 B GR 37776B GR 670137776 A GR670137776 A GR 670137776A GR 670137776 A GR670137776 A GR 670137776A GR 37776 B GR37776 B GR 37776B
Authority
GR
Greece
Prior art keywords
preparation
chlorine
type
endomethylene
benzolosulphonylouries
Prior art date
Application number
GR670137776A
Other languages
Greek (el)
Original Assignee
Farbwerke Hoechst Aktiengesellschaft Vormals Meister Lucius & Bru
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farbwerke Hoechst Aktiengesellschaft Vormals Meister Lucius & Bru filed Critical Farbwerke Hoechst Aktiengesellschaft Vormals Meister Lucius & Bru
Publication of GR37776B publication Critical patent/GR37776B/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/64Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/50Compounds containing any of the groups, X being a hetero atom, Y being any atom
    • C07C311/52Y being a hetero atom
    • C07C311/54Y being a hetero atom either X or Y, but not both, being nitrogen atoms, e.g. N-sulfonylurea

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Manufacture Of Porous Articles, And Recovery And Treatment Of Waste Products (AREA)

Abstract

έθοδος προς παρασκευήν βενζολοσουλφονυλουριών τουτύπου (ΤΥΠΟΣ Ι) εις ον σημαίνουσιν R κατώτερον αλκύλιον, κατά προτίμησινμεθύλιον ή κατώτερον αλκενύλιον, Χ υδρογόνον, φθόριον, χλώριον ή βρώμιον, κατά προτίμησιν χλώριον, κατώτερον αλκύλιον, κατά προτίμησιν μεθύλιον ή κατώτερον αλκοξυ, κατά προτίμησιν μεθοξυ εν της 4- ή 5-θέσει προς την καρβοναμιδομάδα R1 ενδομεθυλενοκυκλοεξενύλιον ή ενδομεθυλενοκυκλοεξύλιον, ενδοαιθυλενοκυκλοεξύλιον, ενδοαιθυλενοκυκλοεξενύλιον, ως και των αλάτων αυτών.process for the preparation of benzenesulphonylureas of the type (TYPE I) εις ον σημαίνουσιν R lower alkyl, preferably methyl or lower alkenyl, Hydrogen, fluorine, chlorine or bromine, preferably chlorine, lower alkyl, preferably methyl or lower alkoxy, preferably methoxy in the 4- or 5-position to the carbonamide group R1 endomethylene cyclohexenyl or endomethylene cyclohexyl, endoethylenecyclohexyl, endoethylenecyclohexenyl, and salts thereof.

GR670137776A 1966-11-29 1967-11-17 METHOD FOR THE PREPARATION OF BENZOLOSULPHONYLOURIES. GR37776B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DEF0050793 1966-11-29
DEF52939A DE1291742B (en) 1966-11-29 1967-07-13 Process for the preparation of benzenesulfonylureas

Publications (1)

Publication Number Publication Date
GR37776B true GR37776B (en) 1969-07-14

Family

ID=25977518

Family Applications (1)

Application Number Title Priority Date Filing Date
GR670137776A GR37776B (en) 1966-11-29 1967-11-17 METHOD FOR THE PREPARATION OF BENZOLOSULPHONYLOURIES.

Country Status (23)

Country Link
JP (1) JPS5015790B1 (en)
AT (5) AT299971B (en)
BE (1) BE707241A (en)
CH (9) CH522608A (en)
CS (7) CS159737B2 (en)
CY (1) CY617A (en)
DE (2) DE1568626C3 (en)
DK (1) DK120539B (en)
ES (1) ES347613A1 (en)
FI (1) FI45963C (en)
FR (2) FR1571292A (en)
GB (1) GB1203425A (en)
GR (1) GR37776B (en)
IL (1) IL28873A (en)
IT (1) IT1056720B (en)
LU (1) LU54967A1 (en)
MC (1) MC696A1 (en)
MY (1) MY7200011A (en)
NL (1) NL6716016A (en)
NO (1) NO122922B (en)
OA (1) OA03381A (en)
SE (1) SE339221B (en)
SU (2) SU460621A3 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3957866A (en) * 1970-09-23 1976-05-18 J. Uriach & Cia S.A. Cyclopentyl carbamide derivative and process for its production
US4072758A (en) * 1970-09-23 1978-02-07 J. Uriach Y Cia, S.A. Compositions and methods for effecting glucoreduction
JPS54175898U (en) * 1978-05-31 1979-12-12
JPS5559632U (en) * 1978-10-20 1980-04-23
CA3059458A1 (en) * 2017-05-24 2018-11-29 The University Of Queensland Novel compounds and uses

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1192192B (en) *

Also Published As

Publication number Publication date
SU473359A3 (en) 1975-06-05
AT289822B (en) 1971-05-10
FI45963B (en) 1972-07-31
CS159737B2 (en) 1975-01-31
AT278845B (en) 1970-02-10
CH522608A (en) 1972-05-15
CH518913A (en) 1972-02-15
CS159738B2 (en) 1975-01-31
CS159740B2 (en) 1975-01-31
FI45963C (en) 1972-11-10
IT1056720B (en) 1982-02-20
CH518915A (en) 1972-02-15
AT278849B (en) 1970-02-10
CH519483A (en) 1972-02-29
DE1568626B2 (en) 1975-04-10
CS159741B2 (en) 1975-01-31
CH519481A (en) 1972-02-29
CH519482A (en) 1972-02-29
DE1291742B (en) 1969-04-03
NL6716016A (en) 1968-05-30
CH518914A (en) 1972-02-15
AT299971B (en) 1972-07-10
SE339221B (en) 1971-10-04
DE1568626C3 (en) 1975-11-20
LU54967A1 (en) 1969-07-04
CY617A (en) 1971-10-25
FR8367M (en) 1971-02-22
BE707241A (en) 1968-05-29
AT278850B (en) 1970-02-10
GB1203425A (en) 1970-08-26
JPS5015790B1 (en) 1975-06-07
MC696A1 (en) 1968-10-21
CH495339A (en) 1970-08-31
OA03381A (en) 1970-12-15
CH519484A (en) 1972-02-29
DE1568626A1 (en) 1970-03-05
ES347613A1 (en) 1969-06-01
DK120539B (en) 1971-06-14
CS159735B2 (en) 1975-01-31
NO122922B (en) 1971-09-06
IL28873A (en) 1973-02-28
SU460621A3 (en) 1975-02-15
FR1571292A (en) 1969-06-20
MY7200011A (en) 1972-12-31
CS159739B2 (en) 1975-01-31
CS159734B2 (en) 1975-01-31

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