GR35672B - METHOD FOR THE PREPARATION OF NEW AMIDES OF ALIPHPATIC CARBONIC ACIDS. - Google Patents

METHOD FOR THE PREPARATION OF NEW AMIDES OF ALIPHPATIC CARBONIC ACIDS.

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Publication number
GR35672B
GR35672B GR670135672A GR670135672A GR35672B GR 35672 B GR35672 B GR 35672B GR 670135672 A GR670135672 A GR 670135672A GR 670135672 A GR670135672 A GR 670135672A GR 35672 B GR35672 B GR 35672B
Authority
GR
Greece
Prior art keywords
general formula
acid
preparation
crystallization
derivative
Prior art date
Application number
GR670135672A
Other languages
Greek (el)
Original Assignee
J. R. Geigy A.G.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by J. R. Geigy A.G. filed Critical J. R. Geigy A.G.
Publication of GR35672B publication Critical patent/GR35672B/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/75Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/74Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79Acids; Esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Bakery Products And Manufacturing Methods Therefor (AREA)
  • Edible Oils And Fats (AREA)
  • Saccharide Compounds (AREA)

Abstract

έθοδος παρασκευής νέων αμιδίων αλειφατικών καρβονοξέων συμφώνως προς τον γενικόν τύπον Ι: [*] εις ον σημαίνουν R1-CO- το ακυλυπόλοιπον ενός αλκανοξέος ή αλκενοξέος μετά 15-22 ατόμων άνθρακος, R2 εν άτομον αλογόνου, μίαν κατωτέραν αλκυλ-, αλκοξυ-, αλκενυλοξυ-, αλκυλοθειο-, αλκενυλοθειο-, αλκανοϋλαμινο-, ή αλκοξυκαρβονυλομάδα και R3 υδρογόνον ή εν κατώτερον αλκυλυπόλοιπον, και των δια προσθήκης αλάτων αυτών μετ' ανοργάνων και οργανικών οξέων, χαρακτηριζομένη εκ του ότι φέρομεν προς αντίδρασιν εν οξύ του γενικού τύπου ΙΙ: R1 - CO - OH εις ον το R1 - CO - έχει την ανωτέρω αναφερθείσαν σημασίαν, ήεν ικανόν προς αντίδρασιν θεμελιώδες παράγωγον ενός τοιούτου οξέος μετά μιας υποκατεστημένης εις τον πυρήνα αμινοπυριδίνης ή υποκατεστημένης εις τον πυρήνα αλκυλαμινοπυριδίνης του γενικού τύπου ΙΙΙ: [*] εις ον R2 και R3 έχουσι την ανωτέρω αναφερθείσαν σημασίαν, ή μεθ' ενός ικανού προς αντίδρασιν θεμελιώδους παραγώγου αυτού, και εάν επιθυμούμεν προσθέτομεν εις εν λαμβανόμενον αλκεναμίδιον του γενικού τύπου Ι βρώμιον, καθαρίζομεν το προϊόν προσθήκης δια κρυσταλώσεως ή μιας άλλης συνήθους μεθόδου και ακολούθως αποβρωμιούμεν, και/ή εάν επιθυμούμενμετατρέπομεν μίαν λαμβανομένην ένωσιν του γενικούτύπου προς εν δια προσθήκης άλας μεθ' ενός ανοργάνου ή οργανικού οξέος. Process for the preparation of novel aliphatic carboxylic amides according to general formula I: [*] εις ον σημαίνουν R1-CO- is the acyl residue of an alkanoic acid or alkenic acid having 15-22 carbon atoms, R 2 in a halogen atom, a lower alkyl-, alkoxy-, alkenyloxy-, alkylthio-, alkenylthio-, alkanoylamino-, or alkoxycarbonyl group and R3 hydrogen or lower alkyl residue, and addition salts thereof with inorganic and organic acids, characterized in that they are reacted with an acid of general formula II: R1 - CO - OH in which R1 - CO - has the above-mentioned significance, or is capable of reacting a fundamental derivative of such an acid with a nucleoside-substituted amino-pyridine or nucle-substituted alkylaminopyridine of general formula III: [*] to R2 and R3 having the above-mentioned significance, or with a reactive fundamental derivative thereof, and if desired to be added to the alkenamide of general formula I bromine, purify the additive by crystallization or other by crystallization or other , and / or if desired a converted compound of the general formula to a salt for addition with an inorganic or organic acid.

GR670135672A 1966-01-28 1967-01-27 METHOD FOR THE PREPARATION OF NEW AMIDES OF ALIPHPATIC CARBONIC ACIDS. GR35672B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH123666 1966-01-28

Publications (1)

Publication Number Publication Date
GR35672B true GR35672B (en) 1968-10-17

Family

ID=4205652

Family Applications (1)

Application Number Title Priority Date Filing Date
GR670135672A GR35672B (en) 1966-01-28 1967-01-27 METHOD FOR THE PREPARATION OF NEW AMIDES OF ALIPHPATIC CARBONIC ACIDS.

Country Status (13)

Country Link
AT (2) AT267526B (en)
BE (1) BE693264A (en)
CH (2) CH491112A (en)
DE (1) DE1695007A1 (en)
DK (1) DK115260B (en)
ES (1) ES336149A1 (en)
FR (2) FR1510320A (en)
GB (1) GB1179263A (en)
GR (1) GR35672B (en)
IL (1) IL27338A (en)
NL (1) NL6701360A (en)
NO (1) NO122421B (en)
SE (1) SE329848B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1991004027A1 (en) * 1989-09-15 1991-04-04 Pfizer Inc. New n-aryl and n-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme a: cholesterol acyl transferase (acat)
CN105017096B (en) * 2015-07-03 2017-08-08 厦门大学 A kind of Oleoyl monoethanolamide derivative, its preparation method and application

Also Published As

Publication number Publication date
NL6701360A (en) 1967-07-31
DK115260B (en) 1969-09-22
DE1695007A1 (en) 1971-02-25
AT269880B (en) 1969-04-10
FR6382M (en) 1968-10-14
IL27338A (en) 1971-02-25
BE693264A (en) 1967-07-27
AT267526B (en) 1969-01-10
SE329848B (en) 1970-10-26
GB1179263A (en) 1970-01-28
CH491112A (en) 1970-05-31
ES336149A1 (en) 1968-10-16
FR1510320A (en) 1968-01-19
NO122421B (en) 1971-06-28
CH484906A (en) 1970-01-31

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