GB1567515A - Esters of testo-sterone and 5 -dihydro-testosterone - Google Patents

Esters of testo-sterone and 5 -dihydro-testosterone Download PDF

Info

Publication number
GB1567515A
GB1567515A GB2131477A GB2131477A GB1567515A GB 1567515 A GB1567515 A GB 1567515A GB 2131477 A GB2131477 A GB 2131477A GB 2131477 A GB2131477 A GB 2131477A GB 1567515 A GB1567515 A GB 1567515A
Authority
GB
United Kingdom
Prior art keywords
testosterone
alkyl
esters
weight
cyclo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB2131477A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Akzo NV
Original Assignee
Akzo NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/691,103 external-priority patent/US4098802A/en
Application filed by Akzo NV filed Critical Akzo NV
Publication of GB1567515A publication Critical patent/GB1567515A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0018Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa
    • C07J1/0022Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C07J1/0025Esters

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
GB2131477A 1976-05-28 1977-05-20 Esters of testo-sterone and 5 -dihydro-testosterone Expired GB1567515A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/691,103 US4098802A (en) 1975-02-18 1976-05-28 Oral pharmaceutical preparation having androgenic activity

Publications (1)

Publication Number Publication Date
GB1567515A true GB1567515A (en) 1980-05-14

Family

ID=24775172

Family Applications (1)

Application Number Title Priority Date Filing Date
GB2131477A Expired GB1567515A (en) 1976-05-28 1977-05-20 Esters of testo-sterone and 5 -dihydro-testosterone

Country Status (12)

Country Link
JP (1) JPS52148060A (fi)
AR (1) AR214323A1 (fi)
BE (1) BE855163A (fi)
CH (1) CH627761A5 (fi)
DE (1) DE2723876C2 (fi)
DK (1) DK146096C (fi)
ES (1) ES459230A1 (fi)
FI (1) FI57597C (fi)
FR (1) FR2352832A1 (fi)
GB (1) GB1567515A (fi)
NL (1) NL7705790A (fi)
SE (1) SE425493B (fi)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002015938A2 (en) * 2000-08-23 2002-02-28 Akzo Nobel N.V. Testosterone ester formulation for human use
US7718640B2 (en) 2003-03-14 2010-05-18 Bayer-Schering Pharma Ag Methods and pharmaceutical compositions for reliable achievement of acceptable serum testosterone levels
US9012436B2 (en) 2008-04-28 2015-04-21 Diurnal Limited Lipid composition
US11311555B2 (en) 2010-11-30 2022-04-26 Lipocine Inc. High-strength testosterone undecanoate compositions

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20180153904A1 (en) 2010-11-30 2018-06-07 Lipocine Inc. High-strength testosterone undecanoate compositions
US20120148675A1 (en) 2010-12-10 2012-06-14 Basawaraj Chickmath Testosterone undecanoate compositions
TW201521731A (zh) * 2013-03-15 2015-06-16 利波辛股份有限公司 用於口服之脂平衡的長鏈睪固酮酯
US20180147215A1 (en) 2016-11-28 2018-05-31 Lipocine Inc. Oral testosterone undecanoate therapy

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL189235C (nl) * 1974-02-28 1993-02-16 Akzo Nv Werkwijze voor de bereiding van een oraal toe te dienen farmaceutisch preparaat met androgene werking.

Cited By (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002015938A2 (en) * 2000-08-23 2002-02-28 Akzo Nobel N.V. Testosterone ester formulation for human use
WO2002015938A3 (en) * 2000-08-23 2002-08-15 Akzo Nobel Nv Testosterone ester formulation for human use
JP2004506698A (ja) * 2000-08-23 2004-03-04 アクゾ・ノベル・エヌ・ベー ヒトに用いるためのテストステロンエステル製剤
AU2001291775B2 (en) * 2000-08-23 2005-09-08 N.V. Organon Testosterone ester formulation for human use
US7718640B2 (en) 2003-03-14 2010-05-18 Bayer-Schering Pharma Ag Methods and pharmaceutical compositions for reliable achievement of acceptable serum testosterone levels
US8338395B2 (en) 2003-03-14 2012-12-25 Bayer Intellectual Property Gmbh Methods and pharmaceutical compositions for reliable achievement of acceptable serum testosterone levels
US9012436B2 (en) 2008-04-28 2015-04-21 Diurnal Limited Lipid composition
US11311555B2 (en) 2010-11-30 2022-04-26 Lipocine Inc. High-strength testosterone undecanoate compositions
US11364249B2 (en) 2010-11-30 2022-06-21 Lipocine Inc. High-strength testosterone undecanoate compositions
US11364250B2 (en) 2010-11-30 2022-06-21 Lipocine Inc. High-strength testosterone undecanoate compositions

Also Published As

Publication number Publication date
FR2352832B1 (fi) 1980-07-11
ES459230A1 (es) 1978-11-16
FI57597C (fi) 1980-09-10
DE2723876A1 (de) 1977-12-15
SE7706235L (sv) 1977-11-29
JPS52148060A (en) 1977-12-08
FI57597B (fi) 1980-05-30
DK236877A (da) 1977-11-29
DK146096B (da) 1983-06-27
AR214323A1 (es) 1979-05-31
JPS6145637B2 (fi) 1986-10-08
CH627761A5 (en) 1982-01-29
FI771684A (fi) 1977-11-29
FR2352832A1 (fr) 1977-12-23
DK146096C (da) 1983-11-21
DE2723876C2 (de) 1986-10-30
BE855163A (fr) 1977-11-28
NL7705790A (nl) 1977-11-30
SE425493B (sv) 1982-10-04

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Legal Events

Date Code Title Description
PS Patent sealed
PCNP Patent ceased through non-payment of renewal fee